Evaluation of endo- and exo-aryl-substitutions and central scaffold modifications on diphenyl substituted alkanes as 5-lipoxygenase activating protein inhibitors
Chu, Lin, Armstrong, Helen M., Chang, Linda L., Cheng, Amy F., Colwell, Lawrence, Cui, Jisong, Evans, Jilly, Galka, Amy, Goulet, Mark T., Hayes, Nancy, Lo, Jane, Menke, John, Ok, Hyun O., Ondeyka, Debra L., Patel, Minal, Quaker, Grace M., Sings, Heather, Witkin, Stephanie L., Zhao, Annie, Ujjainwalla, Feroze
Published in Bioorganic & medicinal chemistry letters (15.06.2012)
Published in Bioorganic & medicinal chemistry letters (15.06.2012)
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Synthesis and structure–activity relationships of pyrido[3,2-b]pyrazin-3(4H)-ones and pteridin-7(8H)-ones as corticotropin-releasing factor-1 receptor antagonists
Dzierba, Carolyn D., Sielecki, Thais M., Arvanitis, Argyrios G., Galka, Amy, Johnson, Tricia L., Takvorian, Amy G., Rafalski, Maria, Kasireddy-Polam, Padmaja, Vig, Shikha, Dasgupta, Bireshwar, Zhang, Ge, Molski, Thaddeus F., Wong, Harvey, Zaczek, Robert C., Lodge, Nicholas J., Combs, Andrew P., Gilligan, Paul J., Trainor, George L., Bronson, Joanne J., Macor, John E.
Published in Bioorganic & medicinal chemistry letters (01.08.2012)
Published in Bioorganic & medicinal chemistry letters (01.08.2012)
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Substituted acyclic sulfonamides as human cannabinoid-1 receptor inverse agonists
Armstrong, Helen E., Galka, Amy, Lin, Linus S., Lanza, Thomas J., Jewell, James P., Shah, Shrenik K., Guthikonda, Ravi, Truong, Quang, Chang, Linda L., Quaker, Grace, Colandrea, Vincent J., Tong, Xinchun, Wang, Junying, Xu, Sherry, Fong, Tung M., Shen, Chun-Pyn, Lao, Julie, Chen, Jing, Shearman, Lauren P., Stribling, D. Sloan, Rosko, Kimberly, Strack, Alison, Ha, Sookhee, der Ploeg, Lex Van, Goulet, Mark T., Hagmann, William K.
Published in Bioorganic & medicinal chemistry letters (15.04.2007)
Published in Bioorganic & medicinal chemistry letters (15.04.2007)
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