The GABAB Receptor—Structure, Ligand Binding and Drug Development
Evenseth, Linn Samira Mari, Gabrielsen, Mari, Sylte, Ingebrigt
Published in Molecules (Basel, Switzerland) (07.07.2020)
Published in Molecules (Basel, Switzerland) (07.07.2020)
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Journal Article
Ligand-guided homology modelling of the GABAB2 subunit of the GABAB receptor
Freyd, Thibaud, Warszycki, Dawid, Mordalski, Stefan, Bojarski, Andrzej J, Sylte, Ingebrigt, Gabrielsen, Mari
Published in PloS one (01.03.2017)
Published in PloS one (01.03.2017)
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Journal Article
In Silico Methods for the Discovery of Orthosteric GABAB Receptor Compounds
Evenseth, Linn, Warszycki, Dawid, Bojarski, Andrzej, Gabrielsen, Mari, Sylte, Ingebrigt
Published in Molecules (Basel, Switzerland) (07.03.2019)
Published in Molecules (Basel, Switzerland) (07.03.2019)
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Journal Article
A short update on the structure of drug binding sites on neurotransmitter transporters
Gabrielsen, Mari, Sylte, Ingebrigt, Dahl, Svein G, Ravna, Aina W
Published in BMC research notes (22.12.2011)
Published in BMC research notes (22.12.2011)
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Journal Article
Homology Modeling of Transporter Proteins
Sylte, Ingebrigt, Gabrielsen, Mari, Kristiansen, Kurt
Published in Methods in molecular biology (Clifton, N.J.) (2023)
Published in Methods in molecular biology (Clifton, N.J.) (2023)
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Journal Article
Exploring Conformational Dynamics of the Extracellular Venus flytrap Domain of the GABA B Receptor: A Path-Metadynamics Study
Evenseth, Linn S M, Ocello, Riccardo, Gabrielsen, Mari, Masetti, Matteo, Recanatini, Maurizio, Sylte, Ingebrigt, Cavalli, Andrea
Published in Journal of chemical information and modeling (27.04.2020)
Published in Journal of chemical information and modeling (27.04.2020)
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Journal Article
Exploring Conformational Dynamics of the Extracellular Venus flytrap Domain of the GABAB Receptor: A Path-Metadynamics Study
Evenseth, Linn S. M, Ocello, Riccardo, Gabrielsen, Mari, Masetti, Matteo, Recanatini, Maurizio, Sylte, Ingebrigt, Cavalli, Andrea
Published in Journal of chemical information and modeling (27.04.2020)
Published in Journal of chemical information and modeling (27.04.2020)
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Journal Article
Ligand-guided homology modelling of the GABA.sub.B2 subunit of the GABA.sub.B receptor
Freyd, Thibaud, Warszycki, Dawid, Mordalski, Stefan, Bojarski, Andrzej J, Sylte, Ingebrigt, Gabrielsen, Mari
Published in PloS one (21.03.2017)
Published in PloS one (21.03.2017)
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Journal Article
The GABA B Receptor-Structure, Ligand Binding and Drug Development
Evenseth, Linn Samira Mari, Gabrielsen, Mari, Sylte, Ingebrigt
Published in Molecules (Basel, Switzerland) (07.07.2020)
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Published in Molecules (Basel, Switzerland) (07.07.2020)
Journal Article
Regulation of liver X receptor target genes by 22-functionalized oxysterols. Synthesis, in silico and in vitro evaluations
Viktorsson, Elvar Örn, Gabrielsen, Mari, Kumarachandran, Nugalya, Sylte, Ingebrigt, Rongved, Pål, Åstrand, Ove Alexander Høgmoen, Kase, Eili Tranheim
Published in Steroids (01.02.2017)
Published in Steroids (01.02.2017)
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Journal Article
Identification of Novel Serotonin Transporter Compounds by Virtual Screening
Gabrielsen, Mari, Kurczab, Rafał, Siwek, Agata, Wolak, Małgorzata, Ravna, Aina W, Kristiansen, Kurt, Kufareva, Irina, Abagyan, Ruben, Nowak, Gabriel, Chilmonczyk, Zdzisław, Sylte, Ingebrigt, Bojarski, Andrzej J
Published in Journal of chemical information and modeling (24.03.2014)
Published in Journal of chemical information and modeling (24.03.2014)
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Journal Article
Homology Modeling of Human [gamma]-Butyric Acid Transporters and the Binding of Pro-Drugs 5-Aminolevulinic Acid and Methyl Aminolevulinic Acid Used in Photodynamic Therapy
Baglo, Yan, Gabrielsen, Mari, Sylte, Ingebrigt, Gederaas, Odrun A
Published in PloS one (07.06.2013)
Published in PloS one (07.06.2013)
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Journal Article
In Silico Methods for the Discovery of Orthosteric GABA B Receptor Compounds
Evenseth, Linn M, Warszycki, Dawid, Bojarski, Andrzej J, Gabrielsen, Mari, Sylte, Ingebrigt
Published in Molecules (Basel, Switzerland) (07.03.2019)
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Published in Molecules (Basel, Switzerland) (07.03.2019)
Journal Article
Synthesis, in vitro and in vivo biological evaluation of new oxysterols as modulators of the liver X receptors
Åstrand, Ove Alexander Høgmoen, Viktorsson, Elvar Örn, Kristensen, Aleksander Lim, Ekeberg, Dag, Røberg-Larsen, Hanne, Wilson, Steven Ray, Gabrielsen, Mari, Sylte, Ingebrigt, Rustan, Arild Christian, Thoresen, G. Hege, Rongved, Pål, Kase, Eili Tranheim
Published in The Journal of steroid biochemistry and molecular biology (01.01.2017)
Published in The Journal of steroid biochemistry and molecular biology (01.01.2017)
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Journal Article
Molecular mechanism of serotonin transporter inhibition elucidated by a new flexible docking protocol
Gabrielsen, Mari, Kurczab, Rafał, Ravna, Aina W., Kufareva, Irina, Abagyan, Ruben, Chilmonczyk, Zdzisław, Bojarski, Andrzej J., Sylte, Ingebrigt
Published in European journal of medicinal chemistry (01.01.2012)
Published in European journal of medicinal chemistry (01.01.2012)
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Journal Article
Homology Modeling of Human gamma -Butyric Acid Transporters and the Binding of Pro-Drugs 5-Aminolevulinic Acid and Methyl Aminolevulinic Acid Used in Photodynamic Therapy. e65200
Baglo, Yan, Gabrielsen, Mari, Sylte, Ingebrigt, Gederaas, Odrun A
Published in PloS one (01.06.2013)
Published in PloS one (01.06.2013)
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Journal Article
Synthesis, Antidepressant Evaluation and Docking Studies of Long-Chain Alkylnitroquipazines as Serotonin Transporter Inhibitors
Gabrielsen, Mari, Wołosewicz, Karol, Zawadzka, Anna, Kossakowski, Jerzy, Nowak, Gabriel, Wolak, Małgorzata, Stachowicz, Katarzyna, Siwek, Agata, Ravna, Aina W., Kufareva, Irina, Kozerski, Lech, Bednarek, Elżbieta, Sitkowski, Jerzy, Bocian, Wojciech, Abagyan, Ruben, Bojarski, Andrzej J., Sylte, Ingebrigt, Chilmonczyk, Zdzisław
Published in Chemical biology & drug design (01.06.2013)
Published in Chemical biology & drug design (01.06.2013)
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Journal Article
Synthesis, in vitro binding studies and docking of long-chain arylpiperazine nitroquipazine analogues, as potential serotonin transporter inhibitors
Jarończyk, Małgorzata, Wołosewicz, Karol, Gabrielsen, Mari, Nowak, Gabriel, Kufareva, Irina, Mazurek, Aleksander P., Ravna, Aina W., Abagyan, Ruben, Bojarski, Andrzej J., Sylte, Ingebrigt, Chilmonczyk, Zdzisław
Published in European journal of medicinal chemistry (01.03.2012)
Published in European journal of medicinal chemistry (01.03.2012)
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Journal Article