Targeting Tumour-Associated Fibroblasts in Cancers
Shah, Kairav, Mallik, Sanchari Basu, Gupta, Praveer, Iyer, Abishek
Published in Frontiers in oncology (22.06.2022)
Published in Frontiers in oncology (22.06.2022)
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Journal Article
HDAC7 Inhibition by Phenacetyl and Phenylbenzoyl Hydroxamates
Mak, Jeffrey Y. W, Wu, Kai-Chen, Gupta, Praveer K, Barbero, Sheila, McLaughlin, Maddison G, Lucke, Andrew J, Tng, Jiahui, Lim, Junxian, Loh, Zhixuan, Sweet, Matthew J, Reid, Robert C, Liu, Ligong, Fairlie, David P
Published in Journal of medicinal chemistry (25.02.2021)
Published in Journal of medicinal chemistry (25.02.2021)
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Inhibitors of class I histone deacetylases attenuate thioacetamide‐induced liver fibrosis in mice by suppressing hepatic type 2 inflammation
Loh, Zhixuan, Fitzsimmons, Rebecca L., Reid, Robert C., Ramnath, Divya, Clouston, Andrew, Gupta, Praveer K., Irvine, Katharine M., Powell, Elizabeth E., Schroder, Kate, Stow, Jennifer L., Sweet, Matthew J., Fairlie, David P., Iyer, Abishek
Published in British journal of pharmacology (01.10.2019)
Published in British journal of pharmacology (01.10.2019)
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Journal Article
Potent Cationic Inhibitors of West Nile Virus NS2B/NS3 Protease With Serum Stability, Cell Permeability and Antiviral Activity
Stoermer, Martin J, Chappell, Keith J, Liebscher, Susann, Jensen, Christina M, Gan, Chun H, Gupta, Praveer K, Xu, Wei-Jun, Young, Paul R, Fairlie, David P
Published in Journal of medicinal chemistry (25.09.2008)
Published in Journal of medicinal chemistry (25.09.2008)
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Journal Article
Towards isozyme-selective HDAC inhibitors for interrogating disease
Gupta, Praveer, Reid, Robert C, Iyer, Abishek, Sweet, Matthew J, Fairlie, David P
Published in Current topics in medicinal chemistry (01.08.2012)
Published in Current topics in medicinal chemistry (01.08.2012)
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Insecticidal activities of histone deacetylase inhibitors against a dipteran parasite of sheep, Lucilia cuprina
Bagnall, Neil H., Hines, Barney M., Lucke, Andrew J., Gupta, Praveer K., Reid, Robert C., Fairlie, David P., Kotze, Andrew C.
Published in International journal for parasitology -- drugs and drug resistance (01.04.2017)
Published in International journal for parasitology -- drugs and drug resistance (01.04.2017)
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Journal Article
Inhibitors selective for HDAC6 in enzymes and cells
Gupta, Praveer K., Reid, Robert C., Liu, Ligong, Lucke, Andrew J., Broomfield, Steve A., Andrews, Melanie R., Sweet, Matthew J., Fairlie, David P.
Published in Bioorganic & medicinal chemistry letters (01.12.2010)
Published in Bioorganic & medicinal chemistry letters (01.12.2010)
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Journal Article
Histone deacetylase enzymes as drug targets for the control of the sheep blowfly, Lucilia cuprina
Kotze, Andrew C., Hines, Barney M., Bagnall, Neil H., Anstead, Clare A., Gupta, Praveer, Reid, Robert C., Ruffell, Angela P., Fairlie, David P.
Published in International journal for parasitology -- drugs and drug resistance (01.12.2015)
Published in International journal for parasitology -- drugs and drug resistance (01.12.2015)
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Journal Article
Comparative α-Helicity of Cyclic Pentapeptides in Water
de Araujo, Aline D., Hoang, Huy N., Kok, W. Mei, Diness, Frederik, Gupta, Praveer, Hill, Timothy A., Driver, Russell W., Price, David A., Liras, Spiros, Fairlie, David P.
Published in Angewandte Chemie (International ed.) (01.07.2014)
Published in Angewandte Chemie (International ed.) (01.07.2014)
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Journal Article
Differential Anti-inflammatory Activity of HDAC Inhibitors in Human Macrophages and Rat Arthritis
Lohman, Rink-Jan, Iyer, Abishek, Fairlie, Thomas J, Cotterell, Adam, Gupta, Praveer, Reid, Robert C, Vesey, David A, Sweet, Matthew J, Fairlie, David P
Published in The Journal of pharmacology and experimental therapeutics (01.02.2016)
Published in The Journal of pharmacology and experimental therapeutics (01.02.2016)
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Journal Article
Comparative [alpha]-Helicity of Cyclic Pentapeptides in Water
deAraujo, Aline D, Hoang, Huy N, Kok, W Mei, Diness, Frederik, Gupta, Praveer, Hill, Timothy A, Driver, Russell W, Price, David A, Liras, Spiros, Fairlie, David P
Published in Angewandte Chemie International Edition (01.07.2014)
Published in Angewandte Chemie International Edition (01.07.2014)
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Journal Article
Histone Deacetylase 7 Promotes Toll-like Receptor 4-dependent Proinflammatory Gene Expression in Macrophages
Shakespear, Melanie R., Hohenhaus, Daniel M., Kelly, Greg M., Kamal, Nabilah A., Gupta, Praveer, Labzin, Larisa I., Schroder, Kate, Garceau, Valerie, Barbero, Sheila, Iyer, Abishek, Hume, David A., Reid, Robert C., Irvine, Katharine M., Fairlie, David P., Sweet, Matthew J.
Published in The Journal of biological chemistry (30.08.2013)
Published in The Journal of biological chemistry (30.08.2013)
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Journal Article
A Versatile Synthetic Approach toward Diversity Libraries using Monosaccharide Scaffolds
Le Thanh, Giang, Abbenante, Giovanni, Adamson, George, Becker, Bernd, Clark, Chris, Condie, Glenn, Falzun, Tania, Grathwohl, Matthias, Gupta, Praveer, Hanson, Michael, Huynh, Ngoc, Katavic, Peter, Kuipers, Krystle, Lam, Ann, Liu, Ligong, Mann, Maretta, Mason, Jeff, McKeveney, Declan, Muldoon, Craig, Pearson, Andrew, Rajaratnam, Premraj, Ryan, Sarah, Tometzki, Gerry, Verquin, Geraldine, Waanders, Jennifer, West, Michael, Wilcox, Neil, Wimmer, Norbert, Yau, Annika, Zuegg, Johannes, Meutermans, Wim
Published in Journal of organic chemistry (01.01.2010)
Published in Journal of organic chemistry (01.01.2010)
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Journal Article
Comparative α-Helicity of Cyclic Pentapeptides in Water
de Araujo, Aline D., Hoang, Huy N., Kok, W. Mei, Diness, Frederik, Gupta, Praveer, Hill, Timothy A., Driver, Russell W., Price, David A., Liras, Spiros, Fairlie, David P.
Published in Angewandte Chemie (01.07.2014)
Published in Angewandte Chemie (01.07.2014)
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Journal Article
Orthogonally Protected Monosaccharide Building Blocks for Solid Phase Production of Diversity Oriented Libraries
Rajaratnam, Premraj, Gupta, Praveer, Katavic, Peter, Kuipers, Krystle, Huyh, Ngoc, Ryan, Sarah, Falzun, Tania, Tometzki, Gerrald B, Bornaghi, Laurent, Le Thanh, Giang, Abbenante, Giovanni, Liu, Ligong, Meutermans, Wim, Wimmer, Norbert, West, Michael L
Published in Australian journal of chemistry (2010)
Published in Australian journal of chemistry (2010)
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