4-(2-Chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]5-methyl-N-(2-propynyl)-1, 3-thiazol-2-amine Hydrochloride (SSR125543A), a Potent and Selective Corticotrophin-Releasing Factor1 Receptor Antagonist. II. Characterization in Rodent Models of Stress-Related Disorders
Guy Griebel, Jacques Simiand, Régis Steinberg, Mireille Jung, Danielle Gully, Pierre Roger, Michel Geslin, Bernard Scatton, Jean-Pierre Maffrand, Philippe SoubriÃ
Published in The Journal of pharmacology and experimental therapeutics (01.04.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2002)
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Journal Article
The 100-kDa Neurotensin Receptor Is gp95/Sortilin, A Non-G-Protein-coupled Receptor
Mazella, Jean, Zsürger, Nicole, Navarro, Valérie, Chabry, Joëlle, Kaghad, Mourad, Caput, Daniel, Ferrara, Pascual, Vita, Natalio, Gully, Danielle, Maffrand, Jean-Pierre, Vincent, Jean-Pierre
Published in The Journal of biological chemistry (09.10.1998)
Published in The Journal of biological chemistry (09.10.1998)
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Journal Article
4-(2-Chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]5-methyl-N-(2-propynyl)-1,3-thiazol-2-amine Hydrochloride (SSR125543A): A Potent and Selective Corticotrophin-Releasing Factor1 Receptor Antagonist. I. Biochemical and Pharmacological Characterization
Danielle Gully, Michel Geslin, Laurence Serva, Evelyne Fontaine, Pierre Roger, Christine Lair, Valerie Darre, Claudine Marcy, Pierre-Eric Rouby, Jacques Simiand, Josette Guitard, Georgette Gout, Regis Steinberg, Daniel Rodier, Guy Griebel, Philippe Soubrie, Marc Pascal, Rebecca Pruss, Bernard Scatton, Jean-Pierre Maffrand, Gerard Le Fur
Published in The Journal of pharmacology and experimental therapeutics (01.04.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2002)
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Journal Article
Biochemical and Pharmacological Activities of SR 142948A, a New Potent Neurotensin Receptor Antagonist
Gully, D, Labeeuw, B, Boigegrain, R, Oury-Donat, F, Bachy, A, Poncelet, M, Steinberg, R, Suaud-Chagny, M F, Santucci, V, Vita, N, Pecceu, F, Labbé-Jullié, C, Kitabgi, P, Soubrié, P, Le Fur, G, Maffrand, J P
Published in The Journal of pharmacology and experimental therapeutics (01.02.1997)
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Published in The Journal of pharmacology and experimental therapeutics (01.02.1997)
Journal Article
Arginine 336 and Asparagine 333 of the Human Cholecystokinin-A Receptor Binding Site Interact with the Penultimate Aspartic Acid and the C-terminal Amide of Cholecystokinin
Gigoux, V, Escrieut, C, Fehrentz, J A, Poirot, S, Maigret, B, Moroder, L, Gully, D, Martinez, J, Vaysse, N, Fourmy, D
Published in The Journal of biological chemistry (16.07.1999)
Published in The Journal of biological chemistry (16.07.1999)
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Journal Article
Met-195 of the Cholecystokinin-A Receptor Interacts with the Sulfated Tyrosine of Cholecystokinin and Is Crucial for Receptor Transition to High Affinity State
Gigoux, Véronique, Escrieut, Chantal, Silvente-Poirot, Sandrine, Maigret, Bernard, Gouilleux, Laurent, Fehrentz, Jean-Alain, Gully, Danielle, Moroder, Luis, Vaysse, Nicole, Fourmy, Daniel
Published in The Journal of biological chemistry (05.06.1998)
Published in The Journal of biological chemistry (05.06.1998)
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Journal Article
Identification of Two Amino Acids of the Human Cholecystokinin-A Receptor That Interact with the N-terminal Moiety of Cholecystokinin
Kennedy, Karen, Gigoux, Véronique, Escrieut, Chantal, Maigret, Bernard, Martinez, Jean, Moroder, Luis, Fréhel, Daniel, Gully, Danielle, Vaysse, Nicole, Fourmy, Daniel
Published in The Journal of biological chemistry (31.01.1997)
Published in The Journal of biological chemistry (31.01.1997)
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Journal Article
Dose-Dependent Pain-Facilitatory and -Inhibitory Actions of Neurotensin Are Revealed by SR 48692, a Nonpeptide Neurotensin Antagonist: Influence on the Antinociceptive Effect of Morphine
Smith, D J, Hawranko, A A, Monroe, P J, Gully, D, Urban, M O, Craig, C R, Smith, J P, Smith, D L
Published in The Journal of pharmacology and experimental therapeutics (01.08.1997)
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Published in The Journal of pharmacology and experimental therapeutics (01.08.1997)
Journal Article
SR146131: A New Potent, Orally Active, and Selective Nonpeptide Cholecystokinin Subtype 1 Receptor Agonist. I: In Vitro Studies
Bignon, E, Bachy, A, Boigegrain, R, Brodin, R, Cottineau, M, Gully, D, Herbert, J M, Keane, P, Labie, C, Molimard, J C, Olliero, D, Oury-Donat, F, Petereau, C, Prabonnaud, V, Rockstroh, M P, Schaeffer, P, Servant, O, Thurneyssen, O, Soubrié, P, Pascal, M, Maffrand, J P, Le Fur, G
Published in The Journal of pharmacology and experimental therapeutics (01.05.1999)
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Published in The Journal of pharmacology and experimental therapeutics (01.05.1999)
Journal Article
Inhibition of neurotensin‐induced pancreatic carcinoma growth by a nonpeptide neurotensin receptor antagonist, SR48692
Iwase, Kazuhiro, Evers, B. Mark, Hellmich, Mark R., Kim, Hong Jin, Higashide, Shunichi, Gully, Danielle, Thompson, James C., Townsend, Courtney M.
Published in Cancer (01.05.1997)
Published in Cancer (01.05.1997)
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Journal Article
Peripheral biological activity of SR 27897 : a new potent non-peptide antagonist of CCKA receptors
GULLY, D, FREHEL, D, MARCY, C, SPINAZZE, A, LESPY, L, NELIAT, G, MAFFRAND, J.-P, LE FUR, G
Published in European journal of pharmacology (23.02.1993)
Published in European journal of pharmacology (23.02.1993)
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Journal Article
Human Umbilical Vein Endothelial Cells Express High Affinity Neurotensin Receptors Coupled to Intracellular Calcium Release (∗)
Schaeffer, Paul, Laplace, Marie-Claude, Savi, Pierre, Pflieger, Anne-Marie, Gully, Danielle, Herbert, Jean-Marc
Published in The Journal of biological chemistry (17.02.1995)
Published in The Journal of biological chemistry (17.02.1995)
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Journal Article
Negative modulation of nitric oxide production by neurotensin as a putative mechanism of the diuretic action of SR 48692 in rats
Croci, Tiziano, Landi, Marco, Gully, Danielle, Maffrand, Jean‐Pierre, Le Fur, Gérard, Manara, Luciano
Published in British journal of pharmacology (01.04.1997)
Published in British journal of pharmacology (01.04.1997)
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Journal Article
4-(2-Chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]5-methyl-N-(2-propynyl)-1, 3-thiazol-2-amine hydrochloride (SSR125543A), a potent and selective corticotrophin-releasing factor(1) receptor antagonist. II. Characterization in rodent models of stress-related disorders
Griebel, Guy, Simiand, Jacques, Steinberg, Régis, Jung, Mireille, Gully, Danielle, Roger, Pierre, Geslin, Michel, Scatton, Bernard, Maffrand, Jean-Pierre, Soubrié, Philippe
Published in The Journal of pharmacology and experimental therapeutics (01.04.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2002)
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Journal Article
4-(2-Chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]5-methyl-N-(2-propynyl)-1,3-thiazol-2-amine hydrochloride (SSR125543A): a potent and selective corticotrophin-releasing factor(1) receptor antagonist. I. Biochemical and pharmacological characterization
Gully, Danielle, Geslin, Michel, Serva, Laurence, Fontaine, Evelyne, Roger, Pierre, Lair, Christine, Darre, Valerie, Marcy, Claudine, Rouby, Pierre-Eric, Simiand, Jacques, Guitard, Josette, Gout, Georgette, Steinberg, Regis, Rodier, Daniel, Griebel, Guy, Soubrie, Philippe, Pascal, Marc, Pruss, Rebecca, Scatton, Bernard, Maffrand, Jean-Pierre, Le Fur, Gerard
Published in The Journal of pharmacology and experimental therapeutics (01.04.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2002)
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Journal Article
Neurotensin and a non‐peptide neurotensin receptor antagonist control human colon cancer cell growth in cell culture and in cells xenografted into nude mice
Maoret, Jean‐José, Anini, Younes, Rouyer‐Fessard, Christiane, Gully, Danielle, Laburthe, Marc
Published in International journal of cancer (29.01.1999)
Published in International journal of cancer (29.01.1999)
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Journal Article
Biochemical and Pharmacological Profile of a Potent and Selective Nonpeptide Antagonist of the Neurotensin Receptor
Gully, Danielle, Canton, Maryse, Boigegrain, Robert, Jeanjean, Francis, Molimard, Jean-Charles, Poncelet, Martine, Gueudet, Christiane, Heaulme, Michel, Leyris, Roger, Brouard, Aline, Pelaprat, Didier, Labbe-Jullie, Catherine, Mazella, Jean, Soubrie, Philippe, Maffrand, Jean-Pierre, Rostene, William, Kitabgi, Patrick, Le Fur, Gerard
Published in Proceedings of the National Academy of Sciences - PNAS (01.01.1993)
Published in Proceedings of the National Academy of Sciences - PNAS (01.01.1993)
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Journal Article
Arginine 197 of the cholecystokinin-A receptor binding site interacts with the sulfate of the peptide agonist cholecystokinin
GIGOUX, VÉRONIQUE, MAIGRET, BERNARD, ESCRIEUT, CHANTAL, SILVENTE-POIROT, SANDRINE, BOUISSON, MICHÈLE, FEHRENTZ, JEAN-ALAIN, MORODER, LUIS, GULLY, DANIELLE, MARTINEZ, JEAN, VAYSSE, NICOLE, FOURMY, DANIEL
Published in Protein science (01.11.1999)
Published in Protein science (01.11.1999)
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Journal Article
Characterization of binding sites of a new neurotensin receptor antagonist, [ [formula omitted]]SR 142948A, in the rat brain
Betancur, Catalina, Canton, Maryse, Burgos, Alain, Labeeuw, Bernard, Gully, Danielle, Rostène, William, Pélaprat, Didier
Published in European journal of pharmacology (05.02.1998)
Published in European journal of pharmacology (05.02.1998)
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Journal Article
Use of nonpeptide antagonists to explore the physiological roles of neurotensin. Focus on brain neurotensin/dopamine interactions
Rostene, W, Azzi, M, Boudin, H, Lepee, I, Souaze, F, Mendez-Ubach, M, Betancur, C, Gully, D
Published in Annals of the New York Academy of Sciences (24.04.1997)
Published in Annals of the New York Academy of Sciences (24.04.1997)
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