Search Results - "GUILLON, Rémi" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Highly Selective Phosphatidylinositol 4‑Kinase IIIβ Inhibitors and Structural Insight into Their Mode of Action

Highly Selective Phosphatidylinositol 4‑Kinase IIIβ Inhibitors and Structural Insight into Their Mode of Action

by Mejdrová, Ivana, Chalupská, Dominika, Kögler, Martin, Šála, Michal, Plačková, Pavla, Baumlová, Adriana, Hřebabecký, Hubert, Procházková, Eliška, Dejmek, Milan, Guillon, Rémi, Strunin, Dmytro, Weber, Jan, Lee, Gary, Birkus, Gabriel, Mertlíková-Kaiserová, Helena, Boura, Evzen, Nencka, Radim
Published in Journal of medicinal chemistry (14.05.2015)

Get full text

Journal Article

New azole antifungals with a fused triazinone scaffold

New azole antifungals with a fused triazinone scaffold

by Montoir, David, Guillon, Rémi, Gazzola, Sophie, Ourliac-Garnier, Isabelle, Soklou, Kossi Efouako, Tonnerre, Alain, Picot, Carine, Planchat, Aurélien, Pagniez, Fabrice, Le Pape, Patrice, Logé, Cédric
Published in European journal of medicinal chemistry (01.03.2020)

Get full text

Journal Article

Identification of Noncompetitive Inhibitors of Cytosolic 5′-Nucleotidase II Using a Fragment-Based Approach

Identification of Noncompetitive Inhibitors of Cytosolic 5′-Nucleotidase II Using a Fragment-Based Approach

by Marton, Zsuzsanna, Guillon, Rémi, Krimm, Isabelle, Preeti, Rahimova, Rahila, Egron, David, Jordheim, Lars P, Aghajari, Nushin, Dumontet, Charles, Périgaud, Christian, Lionne, Corinne, Peyrottes, Suzanne, Chaloin, Laurent
Published in Journal of medicinal chemistry (24.12.2015)

Get full text

Journal Article

Lead optimization and biological evaluation of fragment-based cN-II inhibitors

Lead optimization and biological evaluation of fragment-based cN-II inhibitors

by Guillon, Rémi, Rahimova, Rahila, Preeti, Egron, David, Rouanet, Sonia, Dumontet, Charles, Aghajari, Nushin, Jordheim, Lars Petter, Chaloin, Laurent, Peyrottes, Suzanne
Published in European journal of medicinal chemistry (15.04.2019)

Get full text

Journal Article

Discovery of a Novel Broad-Spectrum Antifungal Agent Derived from Albaconazole

Discovery of a Novel Broad-Spectrum Antifungal Agent Derived from Albaconazole

by Guillon, Rémi, Pagniez, Fabrice, Picot, Carine, Hédou, Damien, Tonnerre, Alain, Chosson, Elizabeth, Duflos, Muriel, Besson, Thierry, Logé, Cédric, Le Pape, Patrice
Published in ACS medicinal chemistry letters (14.02.2013)

Get full text

Journal Article

Novel synthesis of angular thiazolo[5,4-f] and [4,5-h]quinazolines, preparation of their linear thiazolo[4,5-g] and [5,4-g]quinazoline analogs

Novel synthesis of angular thiazolo[5,4-f] and [4,5-h]quinazolines, preparation of their linear thiazolo[4,5-g] and [5,4-g]quinazoline analogs

by Hédou, Damien, Guillon, Rémi, Lecointe, Charlotte, Logé, Cédric, Chosson, Elizabeth, Besson, Thierry
Published in Tetrahedron (15.04.2013)

Get full text

Journal Article

Synthesis and structure–activity relationships of 2-phenyl-1-[(pyridinyl- and piperidinylmethyl)amino]-3-(1 H-1,2,4-triazol-1-yl)propan-2-ols as antifungal agents

Synthesis and structure–activity relationships of 2-phenyl-1-[(pyridinyl- and piperidinylmethyl)amino]-3-(1 H-1,2,4-triazol-1-yl)propan-2-ols as antifungal agents

by Giraud, Francis, Guillon, Rémi, Logé, Cédric, Pagniez, Fabrice, Picot, Carine, Borgne, Marc Le, Pape, Patrice Le
Published in Bioorganic & medicinal chemistry letters (15.01.2009)

Get full text

Journal Article

Design of new antifungal agents: synthesis and evaluation of 1-[(1 H-indol-5-ylmethyl)amino]-2-phenyl-3-(1 H-1,2,4-triazol-1-yl)propan-2-ols

Design of new antifungal agents: synthesis and evaluation of 1-[(1 H-indol-5-ylmethyl)amino]-2-phenyl-3-(1 H-1,2,4-triazol-1-yl)propan-2-ols

by Guillon, Rémi, Giraud, Francis, Logé, Cédric, Le Borgne, Marc, Picot, Carine, Pagniez, Fabrice, Le Pape, Patrice
Published in Bioorganic & medicinal chemistry letters (15.10.2009)

Get full text

Journal Article

Design, Synthesis, and Biological Evaluation of 1-[(Biarylmethyl)methylamino]-2-(2,4-difluorophenyl)-3-(1H-1,2,4-triazol-1-yl)propan-2-ols as Potent Antifungal Agents: New Insights into Structure-Activity Relationships

Design, Synthesis, and Biological Evaluation of 1-[(Biarylmethyl)methylamino]-2-(2,4-difluorophenyl)-3-(1H-1,2,4-triazol-1-yl)propan-2-ols as Potent Antifungal Agents: New Insights into Structure-Activity Relationships

by Guillon, Rémi, Pagniez, Fabrice, Rambaud, Charlotte, Picot, Carine, Duflos, Muriel, Logé, Cédric, Le Pape, Patrice
Published in ChemMedChem (04.10.2011)

Get full text

Journal Article

Synthesis and in vitro antifungal evaluation of 2-(2,4-difluorophenyl)-1-[(1H-indol-3-ylmethyl)methylamino]-3-(1H-1,2,4-triazol-1-yl)propan-2-ols

Synthesis and in vitro antifungal evaluation of 2-(2,4-difluorophenyl)-1-[(1H-indol-3-ylmethyl)methylamino]-3-(1H-1,2,4-triazol-1-yl)propan-2-ols

by Guillon, Rémi, Logé, Cédric, Pagniez, Fabrice, Ferchaud-Roucher, Véronique, Duflos, Muriel, Picot, Carine, Pape, Patrice Le
Published in Journal of enzyme inhibition and medicinal chemistry (01.04.2011)

Get full text

Journal Article

Design, Synthesis, and in vitro Antifungal Activity of 1-[(4-Substituted-benzyl)methylamino]-2-(2,4-difluorophenyl)-3-(1H-1,2,4-triazol-1-yl)propan-2-ols

Design, Synthesis, and in vitro Antifungal Activity of 1-[(4-Substituted-benzyl)methylamino]-2-(2,4-difluorophenyl)-3-(1H-1,2,4-triazol-1-yl)propan-2-ols

by Guillon, Rémi, Pagniez, Fabrice, Giraud, Francis, Crépin, Damien, Picot, Carine, Le Borgne, Marc, Morio, Florent, Duflos, Muriel, Logé, Cédric, Le Pape, Patrice
Published in ChemMedChem (02.05.2011)

Get full text

Journal Article

Lead optimization and biological evaluation of fragment-based cN-II inhibitors

Lead optimization and biological evaluation of fragment-based cN-II inhibitors

by Guillon, Rémi, Rahimova, Rahila, Preeti, Preeti, Egron, David, Rouanet, Sonia, Dumontet, Charles, Aghajari, Nushin, Jordheim, Lars Petter, Chaloin, Laurent, Peyrottes, Suzanne
Published in European journal of medicinal chemistry (01.04.2019)

Get full text

Journal Article

ADENINE DERIVATIVES AS PROTEIN KINASE INHIBITORS

ADENINE DERIVATIVES AS PROTEIN KINASE INHIBITORS

by AMIABLE, Claire, SURLERAUX, Dominique, GUILLON, Rémi
Year of Publication 13.09.2023

Get full text

Patent

ADENINE DERIVATIVES AS PROTEIN KINASE INHIBITORS

ADENINE DERIVATIVES AS PROTEIN KINASE INHIBITORS

by AMIABLE, Claire, SURLERAUX, Dominique, GUILLON, Rémi
Year of Publication 13.09.2023

Get full text

Patent

PYRIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS

PYRIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS

by AMIABLE, Claire, SURLERAUX, Dominique, GUILLON, Rémi, LASCHET, Céline
Year of Publication 30.05.2024

Get full text

Patent

Adenine derivatives as protein kinase inhibitors

Adenine derivatives as protein kinase inhibitors

by Amiable, Claire, Surleraux, Dominique, Guillon, Rémi
Year of Publication 01.02.2022

Get full text

Patent

Adenine derivatives as protein kinase inhibitors

Adenine derivatives as protein kinase inhibitors

by Amiable, Claire, Surleraux, Dominique, Guillon, Rémi
Year of Publication 30.09.2021

Get full text

Patent

Adenine derivatives as protein kinase inhibitors

Adenine derivatives as protein kinase inhibitors

by Amiable, Claire, Surleraux, Dominique, Guillon, Rémi
Year of Publication 02.09.2021

Get full text

Patent

Development of Novel Highly Specific FLT3 Targeted Inhibitors for Combination or Sequential Therapy of Acute Myeloid Leukemia

Development of Novel Highly Specific FLT3 Targeted Inhibitors for Combination or Sequential Therapy of Acute Myeloid Leukemia

by Sabir, Misbah, Hellesoy, Monica, Kivioja, Jarno, Engen, Caroline, Amiable, Claire, Popa, Mihaela, Guillon, Remi, Bruserud, Øystein, Heckman, Caroline A, McCormack, Emmet, Surleraux, Dominique, Gjertsen, Bjørn Tore
Published in Blood (08.12.2017)

Get full text

Journal Article

ADENINE DERIVATIVES AS PROTEIN KINASE INHIBITORS

ADENINE DERIVATIVES AS PROTEIN KINASE INHIBITORS

by RÉMI GUILLON, DOMINIQUE SURLERAUX, CLAIRE AMIABLE
Year of Publication 26.02.2020

Get full text

Patent