New Tetrahydroisoquinoline Derivatives Overcome Pgp Activity in Brain-Blood Barrier and Glioblastoma Multiforme in Vitro
Salaroglio, Iris Chiara, Gazzano, Elena, Kopecka, Joanna, Chegaev, Konstantin, Costamagna, Costanzo, Fruttero, Roberta, Guglielmo, Stefano, Riganti, Chiara
Published in Molecules (Basel, Switzerland) (09.06.2018)
Published in Molecules (Basel, Switzerland) (09.06.2018)
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Mitochondrial Delivery of Phenol Substructure Triggers Mitochondrial Depolarization and Apoptosis of Cancer Cells
Gazzano, Elena, Lazzarato, Loretta, Rolando, Barbara, Kopecka, Joanna, Guglielmo, Stefano, Costamagna, Costanzo, Chegaev, Konstantin, Riganti, Chiara
Published in Frontiers in pharmacology (04.06.2018)
Published in Frontiers in pharmacology (04.06.2018)
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Comparative Study of Different H2S Donors as Vasodilators and Attenuators of Superoxide-Induced Endothelial Damage
Marini, Elisabetta, Rolando, Barbara, Sodano, Federica, Blua, Federica, Concina, Giulia, Guglielmo, Stefano, Lazzarato, Loretta, Chegaev, Konstantin
Published in Antioxidants (01.02.2023)
Published in Antioxidants (01.02.2023)
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Journal Article
Direct introduction of cyano group on furoxan ring
Annaratone, Lorenzo, Guglielmo, Stefano, Chegaev, Konstantin Yu
Published in Mendeleev communications (01.11.2017)
Published in Mendeleev communications (01.11.2017)
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Journal Article
Leishmanicidal Activities of Novel Synthetic Furoxan and Benzofuroxan Derivatives
DUTRA, Luiz Antônio, DE ALMEIDA, Letícia, FRUTTERO, Roberta, GRAMINHA, Marcia A. S, DOS SANTOS, Jean Leandro, PASSALACQUA, Thais G, REIS, Juliana Santana, TORRES, Fabio A. E, MARTINEZ, Isabel, PECCININI, Rosangela Gonçalves, CHUNG MAN CHIN, CHEGAEV, Konstantin, GUGLIELMO, Stefano
Published in Antimicrobial agents and chemotherapy (01.08.2014)
Published in Antimicrobial agents and chemotherapy (01.08.2014)
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Phenylsulfonylfuroxans as Modulators of Multidrug-Resistance-Associated Protein-1 and P-Glycoprotein
Fruttero, Roberta, Crosetti, Marco, Chegaev, Konstantin, Guglielmo, Stefano, Gasco, Alberto, Berardi, Francesco, Niso, Mauro, Perrone, Roberto, Panaro, Maria Antonietta, Colabufo, Nicola Antonio
Published in Journal of medicinal chemistry (12.08.2010)
Published in Journal of medicinal chemistry (12.08.2010)
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Thermosensitive Nanocomposite Hydrogels for Intravitreal Delivery of Cefuroxime
Sapino, Simona, Peira, Elena, Chirio, Daniela, Chindamo, Giulia, Guglielmo, Stefano, Oliaro-Bosso, Simonetta, Barbero, Raffaella, Vercelli, Cristina, Re, Giovanni, Brunella, Valentina, Riedo, Chiara, Fea, Antonio Maria, Gallarate, Marina
Published in Nanomaterials (Basel, Switzerland) (15.10.2019)
Published in Nanomaterials (Basel, Switzerland) (15.10.2019)
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Furoxan-, alkylnitrate-derivatives and related compounds as anti-trypanosomatid agents: Mechanism of action studies
Boiani, Lucı´a, Aguirre, Gabriela, González, Mercedes, Cerecetto, Hugo, Chidichimo, Agustina, Cazzulo, Juan J., Bertinaria, Massimo, Guglielmo, Stefano
Published in Bioorganic & medicinal chemistry (01.09.2008)
Published in Bioorganic & medicinal chemistry (01.09.2008)
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Topical nifedipine with lidocaine ointment vs. active control for treatment of Chronic anal fissure: Results of a prospective, randomized, double-blind study
PERROTTI, Pasquale, BOVE, Antonio, ANTROPOLI, Carmine, MOLINO, Domenico, ANTROPOLI, Massimo, BALZANO, Antonio, DE STEFANO, Guglielmo, ATTENA, Francesco
Published in Diseases of the colon & rectum (01.11.2002)
Published in Diseases of the colon & rectum (01.11.2002)
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Tetrazole and oxadiazole derivatives as bioisosteres of tariquidar and elacridar: New potent P-gp modulators acting as MDR reversers
Braconi, Laura, Dei, Silvia, Contino, Marialessandra, Riganti, Chiara, Bartolucci, Gianluca, Manetti, Dina, Romanelli, Maria Novella, Perrone, Maria Grazia, Colabufo, Nicola Antonio, Guglielmo, Stefano, Teodori, Elisabetta
Published in European journal of medicinal chemistry (05.11.2023)
Published in European journal of medicinal chemistry (05.11.2023)
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Journal Article
DNA‐Targeted NO Release Photoregulated by Green Light
Parisi, Cristina, Fraix, Aurore, Guglielmo, Stefano, Spyrakis, Francesca, Rolando, Barbara, Lazzarato, Loretta, Fruttero, Roberta, Gasco, Alberto, Sortino, Salvatore
Published in Chemistry : a European journal (27.10.2020)
Published in Chemistry : a European journal (27.10.2020)
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Journal Article
Molecular dynamics simulations reveal the determinants of cyclin-dependent kinase 2 inhibition by 5-nitrosopyrimidine derivatives
Guglielmo, Stefano, Cortese, Daniela, Cano, Celine, Fruttero, Roberta
Published in Journal of biomolecular structure & dynamics (01.09.2020)
Published in Journal of biomolecular structure & dynamics (01.09.2020)
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One molecule two goals: A selective P-glycoprotein modulator increases drug transport across gastro-intestinal barrier and recovers doxorubicin toxicity in multidrug resistant cancer cells
Contino, Marialessandra, Guglielmo, Stefano, Riganti, Chiara, Antonello, Giulia, Perrone, Maria Grazia, Giampietro, Roberta, Rolando, Barbara, Fruttero, Roberta, Colabufo, Nicola A.
Published in European journal of medicinal chemistry (15.12.2020)
Published in European journal of medicinal chemistry (15.12.2020)
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Journal Article
Synthesis and biological activity of furoxan derivatives against Mycobacterium tuberculosis
Fernandes, Guilherme Felipe dos Santos, de Souza, Paula Carolina, Marino, Leonardo Biancolino, Chegaev, Konstantin, Guglielmo, Stefano, Lazzarato, Loretta, Fruttero, Roberta, Chung, Man Chin, Pavan, Fernando Rogério, dos Santos, Jean Leandro
Published in European journal of medicinal chemistry (10.11.2016)
Published in European journal of medicinal chemistry (10.11.2016)
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Journal Article
Design, Biological Evaluation, and Molecular Modeling of Tetrahydroisoquinoline Derivatives: Discovery of A Potent P‑Glycoprotein Ligand Overcoming Multidrug Resistance in Cancer Stem Cells
Riganti, Chiara, Contino, Marialessandra, Guglielmo, Stefano, Perrone, Maria G, Salaroglio, Iris C, Milosevic, Vladan, Giampietro, Roberta, Leonetti, Francesco, Rolando, Barbara, Lazzarato, Loretta, Colabufo, Nicola A, Fruttero, Roberta
Published in Journal of medicinal chemistry (24.01.2019)
Published in Journal of medicinal chemistry (24.01.2019)
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Structural and biological characterization of new hybrid drugs joining an HDAC inhibitor to different NO-donors
Atlante, Sandra, Chegaev, Konstantin, Cencioni, Chiara, Guglielmo, Stefano, Marini, Elisabetta, Borretto, Emily, Gaetano, Carlo, Fruttero, Roberta, Spallotta, Francesco, Lazzarato, Loretta
Published in European journal of medicinal chemistry (20.01.2018)
Published in European journal of medicinal chemistry (20.01.2018)
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Journal Article
Overcoming Multidrug Resistance (MDR): Design, Biological Evaluation and Molecular Modelling Studies of 2,4‐Substituted Quinazoline Derivatives
Braconi, Laura, Teodori, Elisabetta, Contino, Marialessandra, Riganti, Chiara, Bartolucci, Gianluca, Manetti, Dina, Romanelli, Maria Novella, Perrone, Maria Grazia, Colabufo, Nicola Antonio, Guglielmo, Stefano, Dei, Silvia
Published in ChemMedChem (20.06.2022)
Published in ChemMedChem (20.06.2022)
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