Search Results - "GUDI Girish" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

$Preclinical characterization of ISB 1342, a CD38 × CD3 T-cell engager for relapsed/refractory multiple myeloma$

Preclinical characterization of ISB 1342, a CD38 × CD3 T-cell engager for relapsed/refractory multiple myeloma

by Pouleau, Blandine, Estoppey, Carole, Suere, Perrine, Nallet, Emilie, Laurendon, Amélie, Monney, Thierry, Pais Ferreira, Daniela, Drake, Adam, Carretero-Iglesia, Laura, Macoin, Julie, Berret, Jérémy, Pihlgren, Maria, Doucey, Marie-Agnès, Gudi, Girish S., Menon, Vinu, Udupa, Venkatesha, Maiti, Abhishek, Borthakur, Gautam, Srivastava, Ankita, Blein, Stanislas, Mbow, M. Lamine, Matthes, Thomas, Kaya, Zeynep, Edwards, Claire M., Edwards, James R., Menoret, Emmanuelle, Kervoëlen, Charlotte, Pellat-Deceunynck, Catherine, Moreau, Philippe, Zhukovsky, Eugene, Perro, Mario, Chimen, Myriam
Published in Blood (20.07.2023)

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$Pre-clinical characterization of ISB 1342, a CD38xCD3 T-cell engager for relapsed/refractory multiple myeloma$

Pre-clinical characterization of ISB 1342, a CD38xCD3 T-cell engager for relapsed/refractory multiple myeloma

by Pouleau, Blandine, Estoppey, Carole, Suere, Perrine, Nallet, Emilie, Laurendon, Amélie, Monney, Thierry, Pais Ferreira, Daniela, Drake, Adam, Carretero-Iglesia, Laura, Macoin, Julie, Berret, Jeremy, Pihlgren, Maria, Doucey, Marie-Agnes, Gudi, Girish S, Menon, Vinu, Udupa, Venkatesha, Maiti, Abhishek, Borthakur, Gautam, Srivastava, Ankita, Blein, Stanislas, Mbow, Lamine, Matthes, Thomas, Kaya, Zeynep, Edwards, Claire M, Edwards, James R, Menoret, Emmanuelle, Kervoelen, Charlotte, Pellat-Deceunynck, Catherine, Moreau, Philippe, Zhukovsky, Eugene Alexander, Perro, Mario, Chimen, Myriam
Published in Blood (16.05.2023)

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Single-step Protein A and Protein G avidity purification methods to support bispecific antibody discovery and development

Single-step Protein A and Protein G avidity purification methods to support bispecific antibody discovery and development

by Ollier, Romain, Wassmann, Paul, Monney, Thierry, Ries Fecourt, Christelle, Gn, Sunitha, C A, Vinu, Ayoub, Daniel, Stutz, Cian, Gudi, Girish S, Blein, Stanislas
Published in mAbs (17.11.2019)

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Effect of ritonavir on pharmacokinetics of antimalarial drug combinations in rats

Effect of ritonavir on pharmacokinetics of antimalarial drug combinations in rats

by Sunitha G N, Satyavati Dulipala D, Girish Gudi
Published in International journal of research in pharmaceutical sciences (21.09.2019)

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Discovery of 5-(2-chloro-4′-(1H-imidazol-1-yl)-[1,1′-biphenyl]-4-yl)-1H-tetrazole as potent and orally efficacious S-nitrosoglutathione reductase (GSNOR) inhibitors for the potential treatment of COPD

Discovery of 5-(2-chloro-4′-(1H-imidazol-1-yl)-[1,1′-biphenyl]-4-yl)-1H-tetrazole as potent and orally efficacious S-nitrosoglutathione reductase (GSNOR) inhibitors for the potential treatment of COPD

by Muthukaman, Nagarajan, Deshmukh, Sanjay, Tondlekar, Shital, Tambe, Macchindra, Pisal, Dnyandeo, Sarode, Neelam, Mhatre, Siddharth, Chakraborti, Samitabh, Shah, Daisy, Bhosale, Vikram M., Kulkarni, Abhay, Mahat, Mahamad Yunnus A., Jadhav, Satyawan B., Gudi, Girish S., Khairatkar-Joshi, Neelima, Gharat, Laxmikant A.
Published in Bioorganic & medicinal chemistry letters (15.12.2018)

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Alleviating CYP and hERG liabilities by structure optimization of dihydrofuran-fused tricyclic benzo[d]imidazole series – Potent, selective and orally efficacious microsomal prostaglandin E synthase-1 (mPGES-1) inhibitors: Part-2

Alleviating CYP and hERG liabilities by structure optimization of dihydrofuran-fused tricyclic benzo[d]imidazole series – Potent, selective and orally efficacious microsomal prostaglandin E synthase-1 (mPGES-1) inhibitors: Part-2

by Muthukaman, Nagarajan, Deshmukh, Sanjay, Tambe, Macchindra, Pisal, Dnyandeo, Tondlekar, Shital, Shaikh, Mahamadhanif, Sarode, Neelam, Kattige, Vidya G., Sawant, Pooja, Pisat, Monali, Karande, Vikas, Honnegowda, Srinivasa, Kulkarni, Abhay, Behera, Dayanidhi, Jadhav, Satyawan B., Sangana, Ramchandra R., Gudi, Girish S., Khairatkar-Joshi, Neelima, Gharat, Laxmikant A.
Published in Bioorganic & medicinal chemistry letters (15.04.2018)

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Discovery of furan and dihydrofuran-fused tricyclic benzo[d]imidazole derivatives as potent and orally efficacious microsomal prostaglandin E synthase-1 (mPGES-1) inhibitors: Part-1

Discovery of furan and dihydrofuran-fused tricyclic benzo[d]imidazole derivatives as potent and orally efficacious microsomal prostaglandin E synthase-1 (mPGES-1) inhibitors: Part-1

by Muthukaman, Nagarajan, Tambe, Macchindra, Deshmukh, Sanjay, Pisal, Dnyandeo, Tondlekar, Shital, Shaikh, Mahamadhanif, Sarode, Neelam, Kattige, Vidya G., Pisat, Monali, Sawant, Pooja, Honnegowda, Srinivasa, Karande, Vikas, Kulkarni, Abhay, Behera, Dayanidhi, Jadhav, Satyawan B., Sangana, Ramchandra R., Gudi, Girish S., Khairatkar-Joshi, Neelima, Gharat, Laxmikant A.
Published in Bioorganic & medicinal chemistry letters (01.12.2017)

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Design, Synthesis, and Pharmacological Evaluation of 5,6-Disubstituted Pyridin-2(1H)‑one Derivatives as Phosphodiesterase 10A (PDE10A) Antagonists

Design, Synthesis, and Pharmacological Evaluation of 5,6-Disubstituted Pyridin-2(1H)‑one Derivatives as Phosphodiesterase 10A (PDE10A) Antagonists

by Lingam, V. S. Prasadarao, Dahale, Dnyaneshwar H, Rathi, Vijay E, Shingote, Yogesh B, Thakur, Rajni R, Mindhe, Ajit S, Kummari, Srinivas, Khairatkar-Joshi, Neelima, Bajpai, Malini, Shah, Daisy M, Sapalya, Ratika S, Gullapalli, Srinivas, Gupta, Praveen K, Gudi, Girish S, Jadhav, Satyawan B, Pattem, Rambabu, Thomas, Abraham
Published in Journal of medicinal chemistry (22.10.2015)

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Tricyclic 4,4-dimethyl-3,4-dihydrochromeno[3,4-d]imidazole derivatives as microsomal prostaglandin E-2 synthase-1 (mPGES-1) inhibitors: SAR and in vivo efficacy in hyperalgesia pain model

Tricyclic 4,4-dimethyl-3,4-dihydrochromeno[3,4-d]imidazole derivatives as microsomal prostaglandin E-2 synthase-1 (mPGES-1) inhibitors: SAR and in vivo efficacy in hyperalgesia pain model

by Muthukaman, Nagarajan, Tambe, Macchindra, Shaikh, Mahamadhanif, Pisal, Dnyandeo, Deshmukh, Sanjay, Tondlekar, Shital, Sarode, Neelam, Narayana, Lakshminarayana, Gajera, Jitendra M., Kattige, Vidya G., Honnegowda, Srinivasa, Karande, Vikas, Kulkarni, Abhay, Behera, Dayanidhi, Jadhav, Satyawan B., Gudi, Girish S., Khairatkar-Joshi, Neelima, Gharat, Laxmikant A.
Published in Bioorganic & medicinal chemistry letters (01.06.2017)

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Tricyclic 4,4-dimethyl-3,4-dihydrochromeno[3,4-d]imidazole derivatives as microsomal prostaglandin E2 synthase-1 (mPGES-1) inhibitors: SAR and in vivo efficacy in hyperalgesia pain model

Tricyclic 4,4-dimethyl-3,4-dihydrochromeno[3,4-d]imidazole derivatives as microsomal prostaglandin E2 synthase-1 (mPGES-1) inhibitors: SAR and in vivo efficacy in hyperalgesia pain model

by Muthukaman, Nagarajan, Tambe, Macchindra, Shaikh, Mahamadhanif, Pisal, Dnyandeo, Deshmukh, Sanjay, Tondlekar, Shital, Sarode, Neelam, Narayana, Lakshminarayana, Gajera, Jitendra M., Kattige, Vidya G., Honnegowda, Srinivasa, Karande, Vikas, Kulkarni, Abhay, Behera, Dayanidhi, Jadhav, Satyawan B., Gudi, Girish S., Khairatkar-Joshi, Neelima, Gharat, Laxmikant A.
Published in Bioorganic & medicinal chemistry letters (01.06.2017)

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Discovery of 2-(2-chloro-6-fluorophenyl)amino)-N-(3-fluoro-5-(trifluoromethyl)phenyl)-1-methyl-7,8-dihydro-1H-[1,4]dioxino [2 ',3 ':3,4]benzo[1,2-d]imidazole-5-carboxamide as potent, selective and efficacious microsomal prostaglandin E-2 synthase-1 (mPGES-1) inhibitor

Discovery of 2-(2-chloro-6-fluorophenyl)amino)-N-(3-fluoro-5-(trifluoromethyl)phenyl)-1-methyl-7,8-dihydro-1H-[1,4]dioxino [2 ',3 ':3,4]benzo[1,2-d]imidazole-5-carboxamide as potent, selective and efficacious microsomal prostaglandin E-2 synthase-1 (mPGES-1) inhibitor

by Muthukaman, Nagarajan, Deshmukh, Sanjay, Sarode, Neelam, Tondlekar, Shital, Tambe, Macchindra, Pisal, Dnyandeo, Shaikh, Mahamadhanif, Kattige, Vidya G., Honnegowda, Srinivasa, Karande, Vikas, Kulkarni, Abhay, Jadhav, Satyawan B., Mahat, Mahamad Yunnus A., Gudi, Girish S., Khairatkar-Joshi, Neelima, Gharat, Laxmikant A.
Published in Bioorganic & medicinal chemistry letters (15.12.2016)

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Phase 2b randomized trial of OX40 inhibitor telazorlimab for moderate-to-severe atopic dermatitis

Phase 2b randomized trial of OX40 inhibitor telazorlimab for moderate-to-severe atopic dermatitis

by Rewerska, Barbara, Sher, Lawrence D., Alpizar, Sady, Pauser, Sylvia, Pulka, Grazyna, Mozaffarian, Neelufar, Salhi, Yacine, Martinet, Camille, Jabert, Wafaa, Gudi, Girish, CA, Vinu, GN, Sunitha, Macoin, Julie, Anstett, Victor, Turrini, Riccardo, Doucey, Marie-Agnès, Blein, Stanislas, Konto, Cyril, Machkova, Martina
Published in The journal of allergy and clinical immunology. Global (01.02.2024)

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Synthesis and pharmacological evaluation of novel N-aryl-3,4-dihydro-1′H-spiro[chromene-2,4′-piperidine]-1′-carboxamides as TRPM8 antagonists

Synthesis and pharmacological evaluation of novel N-aryl-3,4-dihydro-1′H-spiro[chromene-2,4′-piperidine]-1′-carboxamides as TRPM8 antagonists

by Chaudhari, Sachin S., Kadam, Ashok B., Khairatkar-Joshi, Neelima, Mukhopadhyay, Indranil, Karnik, Pallavi V., Raghuram, Anupindi, Rao, Shobha S., Vaiyapuri, Thamil Selvan, Wale, Dinesh P., Bhosale, Vikram M., Gudi, Girish S., Sangana, Ramchandra R., Thomas, Abraham
Published in Bioorganic & medicinal chemistry (01.11.2013)

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Imidazopyridazinones as novel PDE7 inhibitors: SAR and in vivo studies in Parkinson’s disease model

Imidazopyridazinones as novel PDE7 inhibitors: SAR and in vivo studies in Parkinson’s disease model

by Banerjee, Abhisek, Patil, Sandip, Pawar, Mahesh Y., Gullapalli, Srinivas, Gupta, Praveen K., Gandhi, Maulik N., Bhateja, Deepak K., Bajpai, Malini, Sangana, Ramachandra Rao, Gudi, Girish S., Khairatkar-Joshi, Neelima, Gharat, Laxmikant A.
Published in Bioorganic & medicinal chemistry letters (01.10.2012)

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Discovery of benzo[d]imidazo[5,1-b]thiazole as a new class of phosphodiesterase 10A inhibitors

Discovery of benzo[d]imidazo[5,1-b]thiazole as a new class of phosphodiesterase 10A inhibitors

by Banerjee, Abhisek, Narayana, Lakshminarayana, Raje, Firoj A., Pisal, Dnyandeo V., Kadam, Pradip A., Gullapalli, Srinivas, Kumar, Hemant, More, Sandeep V., Bajpai, Malini, Sangana, Ramachandra Rao, Jadhav, Satyawan, Gudi, Girish S., Khairatkar-Joshi, Neelima, Merugu, Ravi R.T., Voleti, Sreedhara R., Gharat, Laxmikant A.
Published in Bioorganic & medicinal chemistry letters (15.12.2013)

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Discovery of 2-((2-chloro-6-fluorophenyl)amino)-N-(3-fluoro-5-(trifluoromethyl)phenyl)-1-methyl-7,8-dihydro-1H-[1,4]dioxino[2′,3′:3,4]benzo[1,2-d]imidazole-5-carboxamide as potent, selective and efficacious microsomal prostaglandin E2 synthase-1 (mPGES-1) inhibitor

Discovery of 2-((2-chloro-6-fluorophenyl)amino)-N-(3-fluoro-5-(trifluoromethyl)phenyl)-1-methyl-7,8-dihydro-1H-[1,4]dioxino[2′,3′:3,4]benzo[1,2-d]imidazole-5-carboxamide as potent, selective and efficacious microsomal prostaglandin E2 synthase-1 (mPGES-1) inhibitor

by Muthukaman, Nagarajan, Deshmukh, Sanjay, Sarode, Neelam, Tondlekar, Shital, Tambe, Macchindra, Pisal, Dnyandeo, Shaikh, Mahamadhanif, Kattige, Vidya G., Honnegowda, Srinivasa, Karande, Vikas, Kulkarni, Abhay, Jadhav, Satyawan B., Mahat, Mahamad Yunnus A., Gudi, Girish S., Khairatkar-Joshi, Neelima, Gharat, Laxmikant A.
Published in Bioorganic & medicinal chemistry letters (15.12.2016)

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Design, synthesis and pharmacological evaluation of novel polycyclic heteroarene ethers as PDE10A inhibitors: Part I

Design, synthesis and pharmacological evaluation of novel polycyclic heteroarene ethers as PDE10A inhibitors: Part I

by Das, Sanjib, Harde, Rajendra L., Shelke, Dnyaneshwar E., Khairatkar-Joshi, Neelima, Bajpai, Malini, Sapalya, Ratika S., Surve, Harshada V., Gudi, Girish S., Pattem, Rambabu, Behera, Dayanidhi B., Jadhav, Satyawan B., Thomas, Abraham
Published in Bioorganic & medicinal chemistry letters (01.05.2014)

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Isothiazole and isoxazole fused pyrimidones as PDE7 inhibitors: SAR and pharmacokinetic evaluation

Isothiazole and isoxazole fused pyrimidones as PDE7 inhibitors: SAR and pharmacokinetic evaluation

by Banerjee, Abhisek, Yadav, Pravin S., Bajpai, Malini, Sangana, Ramachandra Rao, Gullapalli, Srinivas, Gudi, Girish S., Gharat, Laxmikant A.
Published in Bioorganic & medicinal chemistry letters (01.05.2012)

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Design, synthesis and pharmacological evaluation of novel polycyclic heteroarene ethers as PDE10A inhibitors: Part II

Design, synthesis and pharmacological evaluation of novel polycyclic heteroarene ethers as PDE10A inhibitors: Part II

by Das, Sanjib, Shelke, Dnyaneshwar E., Harde, Rajendra L., Avhad, Vijayshree B., Khairatkar-Joshi, Neelima, Gullapalli, Srinivas, Gupta, Praveen K., Gandhi, Maulik N., Bhateja, Deepak K., Bajpai, Malini, Joshi, Ashwini A., Marathe, Megha Y., Gudi, Girish S., Jadhav, Satyawan B., Mahat, Mahamad Yunnus A., Thomas, Abraham
Published in Bioorganic & medicinal chemistry letters (01.08.2014)

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EFFECTS OF PROTEIN CALORIE MALNUTRITION ON THE PHARMACOKINETICS OF KETAMINE IN RATS

EFFECTS OF PROTEIN CALORIE MALNUTRITION ON THE PHARMACOKINETICS OF KETAMINE IN RATS

by WILLIAMS, Marion L, MAGER, Donald E, PARENTEAU, Heli, GUDI, Girish, TRACY, Timothy S, MULHERAN, Mike, WAINER, Irving W
Published in Drug metabolism and disposition (01.08.2004)

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