Scalable Synthesis and Isolation of the Four Stereoisomers of Methyl 1-Amino-3-(4-bromophenyl)cyclopentanecarboxylate, Useful Intermediates for the Synthesis of S1P1 Receptor Agonists
Wallace, Grier A, Gordon, Thomas D, Hayes, Martin E, Konopacki, Donald B, Fix-Stenzel, Shannon R, Zhang, Xiaolei, Grongsaard, Pintipa, Cusack, Kevin P, Schaffter, Lisa M, Henry, Rodger F, Stoffel, Robert H
Published in Journal of organic chemistry (03.07.2009)
Published in Journal of organic chemistry (03.07.2009)
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A stereoselective and scalable synthesis of a conformationally constrained S1P1 agonist
Fix-Stenzel, Shannon R., Hayes, Martin E., Zhang, Xiaolei, Wallace, Grier A., Grongsaard, Pintipa, Schaffter, Lisa M., Hannick, Steven M., Franczyk, Thaddeus S., Stoffel, Robert H., Cusack, Kevin P.
Published in Tetrahedron letters (01.07.2009)
Published in Tetrahedron letters (01.07.2009)
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Convergent, Kilogram Scale Synthesis of an Akt Kinase Inhibitor
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Published in Organic process research & development (18.05.2012)
Published in Organic process research & development (18.05.2012)
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Identification of a selective thieno[2,3-c]pyridine inhibitor of COT kinase and TNF-alpha production
Cusack, Kevin, Allen, Hamish, Bischoff, Agnieszka, Clabbers, Anca, Dixon, Richard, Fix-Stenzel, Shannon, Friedman, Michael, Gaumont, Yvette, George, Dawn, Gordon, Thomas, Grongsaard, Pintipa, Janssen, Bernd, Jia, Yong, Moskey, Maria, Quinn, Christopher, Salmeron, Andres, Thomas, Christine, Wallace, Grier, Wishart, Neil, Yu, Zhengtian
Published in Bioorganic & medicinal chemistry letters (15.03.2009)
Published in Bioorganic & medicinal chemistry letters (15.03.2009)
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Discovery of small molecule benzimidazole antagonists of the chemokine receptor CXCR3
Hayes, Martin E., Wallace, Grier A., Grongsaard, Pintipa, Bischoff, Agnieszka, George, Dawn M., Miao, Wenyan, McPherson, Michael J., Stoffel, Robert H., Green, David W., Roth, Gregory P.
Published in Bioorganic & medicinal chemistry (01.03.2008)
Published in Bioorganic & medicinal chemistry (01.03.2008)
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A stereoselective and scalable synthesis of a conformationally constrained S1P(1) agonist
Fix-Stenzel, Shannon R., Hayes, Martin E., Zhang, Xiaolei, Wallace, Grier A., Grongsaard, Pintipa, Schaffter, Lisa M., Hannick, Steven M., Franczyk, Thaddeus S., Stoffel, Robert H., Cusack, Kevin P.
Published in Tetrahedron letters (15.07.2009)
Published in Tetrahedron letters (15.07.2009)
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Journal Article
Lead identification of 2-iminobenzimidazole antagonists of the chemokine receptor CXCR3
Hayes, Martin E., Breinlinger, Eric C., Wallace, Grier A., Grongsaard, Pintipa, Miao, Wenyan, McPherson, Michael J., Stoffel, Robert H., Green, David W., Roth, Gregory P.
Published in Bioorganic & medicinal chemistry (01.04.2008)
Published in Bioorganic & medicinal chemistry (01.04.2008)
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Journal Article
A stereoselective and scalable synthesis of a conformationally constrained S1P 1 agonist
Fix-Stenzel, Shannon R., Hayes, Martin E., Zhang, Xiaolei, Wallace, Grier A., Grongsaard, Pintipa, Schaffter, Lisa M., Hannick, Steven M., Franczyk, Thaddeus S., Stoffel, Robert H., Cusack, Kevin P.
Published in Tetrahedron letters (2009)
Published in Tetrahedron letters (2009)
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Journal Article
Identification of a selective thieno[2,3-c]pyridine inhibitor of COT kinase and TNF-a production
CUSACK, Kevin, ALLEN, Hamish, GRONGSAARD, Pintipa, JANSSEN, Bernd, YONG JIA, MOSKEY, Maria, QUINN, Christopher, SALMERON, Andres, THOMAS, Christine, WALLACE, Grier, WISHART, Neil, ZHENGTIAN YU, BISCHOFF, Agnieszka, CLABBERS, Anca, DIXON, Richard, FIX-STENZEL, Shannon, FRIEDMAN, Michael, GAUMONT, Yvette, GEORGE, Dawn, GORDON, Thomas
Published in Bioorganic & medicinal chemistry letters (2009)
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Published in Bioorganic & medicinal chemistry letters (2009)
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NOVEL OXADIAZOLE COMPOUNDS
FIX STENZEL SHANNON, WOLLER KEVIN R, GRONGSAARD PINTIPA, BREINLINGER ERIC C, ANSELL GRAHAM K, HOBSON ADRIAN D, CUSACK KEVIN P, STOFFEL ROBERT H
Year of Publication 09.09.2009
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Year of Publication 09.09.2009
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2-IMINO-BENZIMIDAZOLES
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Year of Publication 18.08.2010
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Year of Publication 18.08.2010
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NOVEL OXADIAZOLE COMPOUNDS
HOBSON, ADRIAN D, CUSACK, KEVIN P, ANSELL, GRAHAM K, FIX-STENZEL, SHANNON, STOFFEL, ROBERT H, BREINLINGER, ERIC C, GRONGSAARD, PINTIPA, WOLLER, KEVIN R
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Year of Publication 30.01.2012
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Novel Oxadiazole Compounds
WOLLER KEVIN R, GRONGSAARD PINTIPA, BREINLINGER ERIC C, CUSACK KEVIN P, STOFFEL ROBERT H, HOBSON ADRIAN D, FIX-STENZEL SHANNON R
Year of Publication 25.08.2011
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Year of Publication 25.08.2011
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