Food intake inhibition and reduction in body weight gain in lean and obese rodents treated with GW438014A, a potent and selective NPY-Y5 receptor antagonist
Daniels, A.J., Grizzle, M.K., Wiard, R.P., Matthews, J.E., Heyer, D.
Published in Regulatory peptides (15.06.2002)
Published in Regulatory peptides (15.06.2002)
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Optimization of 3-(1H-Indazol-3-ylmethyl)-1,5-benzodiazepines as Potent, Orally Active CCK-A Agonists
Henke, Brad R, Aquino, Christopher J, Birkemo, Larry S, Croom, Dallas K, Dougherty, Robert W, Ervin, Gregory N, Grizzle, Mary K, Hirst, Gavin C, James, Michael K, Johnson, Michael F, Queen, Kennedy L, Sherrill, Ronald G, Sugg, Elizabeth E, Suh, Edward M, Szewczyk, Jerzy W, Unwalla, Rayomand J, Yingling, Jeff, Willson, Timothy M
Published in Journal of medicinal chemistry (15.08.1997)
Published in Journal of medicinal chemistry (15.08.1997)
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The inotropic and beta blocking effects of a chimeric molecule that putatively inhibits both type III phosphodiesterase and beta adrenoceptors in anesthetized dogs
SHAFFER, J. E, GRIZZLE, M. K, ANDERSON, D. K, WHEELER, T. N
Published in The Journal of pharmacology and experimental therapeutics (01.06.1993)
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Published in The Journal of pharmacology and experimental therapeutics (01.06.1993)
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Effect of polyethylene glycol-superoxide dismutase and catalase on endotoxemia in pigs
Olson, N C, Grizzle, M K, Anderson, D L
Published in Journal of applied physiology (1985) (01.10.1987)
Published in Journal of applied physiology (1985) (01.10.1987)
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Dimethylthiourea attenuates endotoxin-induced acute respiratory failure in pigs
Olson, N C, Anderson, D L, Grizzle, M K
Published in Journal of applied physiology (1985) (01.12.1987)
Published in Journal of applied physiology (1985) (01.12.1987)
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3-[2-(N-Phenylacetamide)]-1,5-benzodiazepines: Orally Active, Binding Selective CCK-A Agonists
Willson, Timothy M, Henke, Brad R, Momtahen, Tanya M, Myers, Peter L, Sugg, Elizabeth E, Unwalla, Rayomand J, Croom, Dallas K, Dougherty, Robert W, Grizzle, Mary K, Johnson, Michael F, Queen, Kennedy L, Rimele, Thomas J, Yingling, Jeffrey D, James, Michael K
Published in Journal of medicinal chemistry (19.07.1996)
Published in Journal of medicinal chemistry (19.07.1996)
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Modification of Receptor Selectivity and Functional Activity in Cholecystokinin Peptoid Ligands
Dezube, Milana, Sugg, Elizabeth E, Birkemo, Larry S, Croom, Dallas K, Dougherty, Robert W, Ervin, Gregory N, Grizzle, Mary K, James, Michael K, Johnson, Michael F
Published in Journal of medicinal chemistry (01.08.1995)
Published in Journal of medicinal chemistry (01.08.1995)
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Discovery of 1,5-Benzodiazepines with Peripheral Cholecystokinin (CCK-A) Receptor Agonist Activity (II): Optimization of the C3 Amino Substituent
Hirst, Gavin C., Aquino, Christopher, Birkemo, Lawrence, Croom, Dallas K., Dezube, Milana, Dougherty, Robert W., Ervin, Gregory N., Grizzle, Mary K., Henke, Brad, James, Michael K., Johnson, Michael F., Momtahen, Tanya, Queen, Kennedy L., Sherrill, Ronald G., Szewczyk, Jerzy, Willson, Timothy M., Sugg, Elizabeth E.
Published in Journal of medicinal chemistry (20.12.1996)
Published in Journal of medicinal chemistry (20.12.1996)
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3-(1H-indazol-3-ylmethyl)-1,5-benzo-diazepines : CCK-A agonists that demonstrate oral activity as satiety agents
HENKE, B. R, WILLSON, T. M, JAMES, M. K, SUGG, E. E, CROOM, D. K, DOUGHERTY, R. W, QUEEN, K. L, BIRKEMO, L. S, ERVIN, G. N, GRIZZLE, M. K, JOHNSON, M. T
Published in Journal of medicinal chemistry (1996)
Published in Journal of medicinal chemistry (1996)
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Discovery of 1,5-Benzodiazepines with Peripheral Cholecystokinin (CCK-A) Receptor Agonist Activity. 1. Optimization of the Agonist “Trigger”
Aquino, Christopher J, Armour, Duncan R, Berman, Judd M, Birkemo, Larry S, Carr, Robin A. E, Croom, Dallas K, Dezube, Milana, Dougherty, Robert W, Ervin, Gregory N, Grizzle, Mary K, Head, Julie E, Hirst, Gavin C, James, Michael K, Johnson, Michael F, Miller, Laurence J, Queen, Kennedy L, Rimele, Thomas J, Smith, David N, Sugg, Elizabeth E
Published in Journal of medicinal chemistry (19.01.1996)
Published in Journal of medicinal chemistry (19.01.1996)
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1,4-Benzodiazepine Peripheral Cholecystokinin (CCK-A) Receptor Agonists
Sherrill, Ronald G, Berman, Judd M, Birkemo, Lawrence, Croom, Dallas K, Dezube, Milana, Ervin, Gregory N, Grizzle, Mary K, James, Michael K, Johnson, Michael F, Queen, Kennedy L, Rimele, Thomas J, Vanmiddlesworth, Frank, Sugg, Elizabeth E
Published in Bioorganic & medicinal chemistry letters (07.05.2001)
Published in Bioorganic & medicinal chemistry letters (07.05.2001)
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6-AZASTEROIDS - POTENT DUAL INHIBITORS OF HUMAN TYPE-1 AND 2 STEROID 5-ALPHA-REDUCTASE
FRYE, SV, HAFFNER, CD, MALONEY, PR, MOOK, RA, HINER, RN, BATCHELOR, KW, BRAMSON, HN, STUART, JD, SCHWEIKER, SL, VANARNOLD, J, BICKETT, DM, MOSS, ML, TIAN, GC, UNWALLA, RJ, LEE, FW, TIPPIN, TK, JAMES, MK, GRIZZLE, MK, LONG, JE, SCHUSTER, SV, DORSEY, GF
Published in Journal of medicinal chemistry (24.12.1993)
Published in Journal of medicinal chemistry (24.12.1993)
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Journal Article
3-(1H-Indazol-3-ylmethyl)-1,5-benzodiazepines: CCK-A Agonists That Demonstrate Oral Activity as Satiety Agents
Henke, Brad R, Willson, Timothy M, Sugg, Elizabeth E, Croom, Dallas K, Dougherty, Robert W, Queen, Kennedy L, Birkemo, Larry S, Ervin, Gregory N, Grizzle, Mary K, Johnson, Michael F, James, Michael K
Published in Journal of medicinal chemistry (05.07.1996)
Published in Journal of medicinal chemistry (05.07.1996)
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Characterisation of olanzapine-induced weight gain and effect of aripiprazole vs olanzapine on body weight and prolactin secretion in female rats
KALINICHEV, Mikhail, ROURKE, Claire, DANIELS, Alex J, GRIZZLE, Mary K, BRITT, Christy S, IGNAR, Diane M, JONES, Declan N. C
Published in Psychopharmacologia (01.10.2005)
Published in Psychopharmacologia (01.10.2005)
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Discovery of 1,5-benzodiazepines with peripheral cholecystokinin (CCK-A) receptor agonist activity. I: Optimization of the agonist trigger
AQUINO, C. J, ARMOUR, D. R, HEAD, J. E, HIRST, G. C, JAMES, M. K, JOHNSON, M. F, MILLER, L. J, QUEEN, K. L, RIMELE, T. J, SMITH, D. N, SUGG, E. E, BERMAN, J. M, BIRKEMA, L. S, CARR, R. A. E, CROOM, D. K, DEZUBE, M, DOUGHERTY, R. W, ERVIN, G. N, GRIZZLE, M. K
Published in Journal of medicinal chemistry (1996)
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Published in Journal of medicinal chemistry (1996)
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Structure-activity relationships for inhibition of type 1 and 2 human 5α-reductase and human adrenal 3β-hydroxy-Δ5-steroid dehydrogenase/3-keto-Δ5-steroid isomerase by 6-azaandrost-4-en-3-ones : optimization of the C17 substituent
FRYE, S. V, HAFFNER, C. D, SCHWEIKER, S. L, VAN ARNOLD, J, BICKETT, D. M, MOSS, M. L, GAOCHOA TIAN, LEE, F. W, TIPPIN, T. K, JAMES, M. K, GRIZZLE, M. K, LONG, J. E, MALONEY, P. R, CROOM, D. K, HINER, R. N, DORSEY, G. F, NOE, R. A, UNWALLA, R. J, BATCHELOR, K. W, BRAMSON, H. N, STUART, J. D
Published in Journal of medicinal chemistry (1995)
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Published in Journal of medicinal chemistry (1995)
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