Inhibition of Hypoxia-Induced Gene Transcription by Substituted Pyrazolyl Oxadiazoles: Initial Lead Generation and Structure-Activity Relationships
Härter, Michael, Thierauch, Karl-Heinz, Boyer, Stephen, Bhargava, Ajay, Ellinghaus, Peter, Beck, Hartmut, Greschat-Schade, Susanne, Hess-Stumpp, Holger, Unterschemmann, Kerstin
Published in ChemMedChem (01.01.2014)
Published in ChemMedChem (01.01.2014)
Get full text
Journal Article
SUBSTITUTED HETEROCYCLYL BENZYL PYRAZOLES, AND USE THEREOF
ELLINGHAUS PETER, GRESCHAT SCHADE SUSANNE, UNTERSMAN KERSTIN, SCHUHMACHER JOACHIM, BECK HARTMUT, HAERTER MICHAEL
Year of Publication 07.10.2013
Get full text
Year of Publication 07.10.2013
Patent
HYDROXYALKYL BENZYL PYRAZOLES, AND USE THEREOF FOR THE TREATMENT OF HYPERPROLIFERATIVE AND ANGIOGENIC DISEASES
ELLINGHAUS PETER, GRESCHAT SCHADE SUSANNE, SUESSMEIER FRANK, SCHUHMACHER JOACHIM, THIERAUCH KARL HEINZ, BECK HARTMUT, UNTERSMANN KERSTIN, HAERTER MICHAEL
Year of Publication 07.10.2013
Get full text
Year of Publication 07.10.2013
Patent
IMI – oral biopharmaceutics tools project – evaluation of bottom-up PBPK prediction success part 1: Characterisation of the OrBiTo database of compounds
Margolskee, Alison, Darwich, Adam S., Pepin, Xavier, Pathak, Shriram M., Bolger, Michael B., Aarons, Leon, Rostami-Hodjegan, Amin, Angstenberger, Jonas, Graf, Franziska, Laplanche, Loic, Müller, Thomas, Carlert, Sara, Daga, Pankaj, Murphy, Dónal, Tannergren, Christer, Yasin, Mohammed, Greschat-Schade, Susanne, Mück, Wolfgang, Muenster, Uwe, van der Mey, Dorina, Frank, Kerstin Julia, Lloyd, Richard, Adriaenssen, Lieve, Bevernage, Jan, De Zwart, Loeckie, Swerts, Dominique, Tistaert, Christophe, Van Den Bergh, An, Van Peer, Achiel, Beato, Stefania, Nguyen-Trung, Anh-Thu, Bennett, Joanne, McAllister, Mark, Wong, Mei, Zane, Patricia, Ollier, Céline, Vicat, Pascale, Kolhmann, Markus, Marker, Alexander, Brun, Priscilla, Mazuir, Florent, Beilles, Stéphane, Venczel, Marta, Boulenc, Xavier, Loos, Petra, Lennernäs, Hans, Abrahamsson, Bertil
Published in European journal of pharmaceutical sciences (01.01.2017)
Published in European journal of pharmaceutical sciences (01.01.2017)
Get full text
Journal Article
Predicting biopharmaceutical performance of oral drug candidates – Extending the volume to dissolve applied dose concept
Muenster, Uwe, Mueck, Wolfgang, van der Mey, Dorina, Schlemmer, Karl-Heinz, Greschat-Schade, Susanne, Haerter, Michael, Pelzetter, Christian, Pruemper, Christian, Verlage, Joerg, Göller, Andreas H., Ohm, Andreas
Published in European journal of pharmaceutics and biopharmaceutics (01.05.2016)
Published in European journal of pharmaceutics and biopharmaceutics (01.05.2016)
Get full text
Journal Article
3-(FLUORVINYL)PYRAZOLES AND THE USE THEREOF
THIERAUCH, KARL-HEINZ, GRESCHAT-SCHADE, SUSANNE, ELLINGHAUS, PETER, SCHUHMACHER, JOACHIM, HÄRTER, MICHAEL, BECK, HARTMUT
Year of Publication 28.05.2014
Get full text
Year of Publication 28.05.2014
Patent
SUBSTITUTED HETEROCYCLYL BENZYL PYRAZOLES, AND USE THEREOF
GRESCHAT-SCHADE, Susanne, SCHUHMACHER, Joachim, ELLINGHAUS, Peter, HÄRTER, Michael, BECK, Hartmut, UNTERSMAN, Kerstin
Year of Publication 01.04.2014
Get full text
Year of Publication 01.04.2014
Patent
SUBSTITUTED HETEROCYCLYL BENZYL PYRAZOLES, AND USE THEREOF
GRESCHAT-SCHADE, SUSANNE, ELLINGHAUS, PETER, SCHUHMACHER, JOACHIM, HAERTER, MICHAEL, BECK, HARTMUT, UNTERSMANN, KERSTIN
Year of Publication 26.03.2014
Get full text
Year of Publication 26.03.2014
Patent
Substituted heterocyclyl benzyl pyrazoles, and use thereof
ELLINGHAUS PETER, SCHUHMACHER JOACHIM, BECK HARTMUT, UNTERSMANN KERSTIN, HAERTER MICHAEL, GRESCHAT-SCHADE SUSANNE
Year of Publication 04.07.2013
Get full text
Year of Publication 04.07.2013
Patent
HYDROXYALKYL BENZYL PYRAZOLES,AND USE THEREOF FOR THE TREATMENT OF HYPERPROLIFERATIVE AND ANGIOGENIC DISEASES
SUBMEIER FRANK, ELLINGHAUS PETER, SCHUHMACHER JOACHIM, THIERAUCH KARL-HEINZ, BECK HARTMUT, HARTER MICHAEL, BERHORSTER KERSTIN, GRESCHAT-SCHADE SUSANNE
Year of Publication 28.05.2014
Get full text
Year of Publication 28.05.2014
Patent
SUBSTITUTED HETEROCYCLYL BENZYL PYRAZOLES, AND USE THEREOF
GRESCHAT-SCHADE, SUSANNE, ELLINGHAUS, PETER, SCHUHMACHER, JOACHIM, HAERTER, MICHAEL, BECK, HARTMUT, UNTERSMANN, KERSTIN
Year of Publication 20.03.2013
Get full text
Year of Publication 20.03.2013
Patent
3-(FLUORVINYL)PYRAZOLES AND THE USE THEREOF
THIERAUCH, KARL-HEINZ, GRESCHAT-SCHADE, SUSANNE, ELLINGHAUS, PETER, SCHUHMACHER, JOACHIM, HARTER, MICHAEL, BECK, HARTMUT
Year of Publication 24.01.2013
Get full text
Year of Publication 24.01.2013
Patent
SUBSTITUTED HETEROCYCLYL BENZYL PYRAZOLES, AND USE THEREOF
UNTERSMAN, KERSTIN, GRESCHAT-SCHADE, SUSANNE, ELLINGHAUS, PETER, SCHUHMACHER, JOACHIM, HAERTER, MICHAEL, BECK, HARTMUT
Year of Publication 28.12.2012
Get full text
Year of Publication 28.12.2012
Patent
HYDROXYALKYL BENZYL PYRAZOLES, AND USE THEREOF FOR THE TREATMENT OF HYPERPROLIFERATIVE AND ANGIOGENIC DISEASES
THIERAUCH, KARL-HEINZ, GRESCHAT-SCHADE, SUSANNE, ELLINGHAUS, PETER, SCHUHMACHER, JOACHIM, SUESMEIER, FRANK, HAERTER, MICHAEL, BECK, HARTMUT, UNTERSMANN, KERSTIN
Year of Publication 20.03.2013
Get full text
Year of Publication 20.03.2013
Patent
SUBSTITUTED HETEROCYCLYL BENZYL PYRAZOLES, AND USE THEREOF
UNTERSMAN, KERSTIN, GRESCHAT-SCHADE, SUSANNE, ELLINGHAUS, PETER, SCHUHMACHER, JOACHIM, HAERTER, MICHAEL, BECK, HARTMUT
Year of Publication 17.11.2011
Get full text
Year of Publication 17.11.2011
Patent
Hydroxyalkyl benzyl pyrazoles, and use thereof for the treatment of hyperproliferative and angiogenic diseases
THIERAUCH, KARL-HEINZ, GRESCHAT-SCHADE, SUSANNE, ELLINGHAUS, PETER, SCHUHMACHER, JOACHIM, SUSSMEIER, FRANK, HARTER, MICHAEL, BECK, HARTMUT, UNTERSMANN, KERSTIN
Year of Publication 06.12.2012
Get full text
Year of Publication 06.12.2012
Patent
HYDROXYALKYL BENZYL PYRAZOLES, AND USE THEREOF FOR THE TREATMENT OF HYPERPROLIFERATIVE AND ANGIOGENIC DISEASES
THIERAUCH, KARL-HEINZ, GRESCHAT-SCHADE, SUSANNE, ELLINGHAUS, PETER, SCHUHMACHER, JOACHIM, HAERTER, MICHAEL, SUESSMEIER, FRANK, BECK, HARTMUT, UNTERSMANN, KERSTIN
Year of Publication 17.11.2011
Get full text
Year of Publication 17.11.2011
Patent
heterociclilbenzilpirazóis substituídos e uso do mesmo
HARTMUT BECK, PETER ELLINGHAUS, KERSTIN UNTERSMANN, SUSANNE GRESCHAT-SCHADE, JOACHIM SCHUHMACHER, MICHAEL HÄRTER
Year of Publication 09.08.2016
Get full text
Year of Publication 09.08.2016
Patent
hidroxialquilbenzilpirazois e seu uso
HARTMUT BECK, PETER ELLINGHAUS, KARL-HEINZ THIERAUCH, FRANK SÜSSMEIER, KERSTIN UNTERSMANN, SUSANNE GRESCHAT-SCHADE, JOACHIM SCHUHMACHER, MICHAEL HÄRTER
Year of Publication 09.08.2016
Get full text
Year of Publication 09.08.2016
Patent
Heterociclilbencilpirazoles sustituidos y uso de los mismos
GRESCHAT-SCHADE, SUSANNE, ELLINGHAUS, PETER, SCHUHMACHER, JOACHIM, HÄRTER, MICHAEL, BECK, HARTMUT, UNTERSMANN, KERSTIN
Year of Publication 23.05.2014
Get full text
Year of Publication 23.05.2014
Patent