One-Step, Catalyst-Free Continuous-Flow Method for the Rapid and Safe Synthesis of 1‑Substituted 1H‑Tetrazoles
Fülöp, Zsolt, Bana, Péter, Temesvári, Márton, Barabás, Júlia, Kazsu, Zoltán, Béni, Zoltán, Greiner, István, Éles, János
Published in Organic process research & development (20.09.2024)
Published in Organic process research & development (20.09.2024)
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Journal Article
Continuous Synthesis and Purification by Coupling a Multistep Flow Reaction with Centrifugal Partition Chromatography
Örkényi, Róbert, Éles, János, Faigl, Ferenc, Vincze, Péter, Prechl, Anita, Szakács, Zoltán, Kóti, János, Greiner, István
Published in Angewandte Chemie International Edition (17.07.2017)
Published in Angewandte Chemie International Edition (17.07.2017)
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Journal Article
Synthesis and Characterization of New V 1A Antagonist Compounds: The Separation of Four Atropisomeric Stereoisomers
Szeleczky, Zsolt, Szakács, Zoltán, Bozó, Éva, Baska, Ferenc, Vukics, Krisztina, Lévai, Sándor, Temesvári, Krisztina, Vass, Elemér, Béni, Zoltán, Krámos, Balázs, Magdó, Ildikó, Szántay, Csaba, Kóti, János, Domány-Kovács, Katalin, Greiner, István, Bata, Imre
Published in Journal of medicinal chemistry (22.07.2021)
Published in Journal of medicinal chemistry (22.07.2021)
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Journal Article
Biomimetic Synthesis of Drug Metabolites in Batch and Continuous‐Flow Reactors
Fődi, Tamás, Ignácz, Gergő, Decsi, Balázs, Béni, Zoltán, Túrós, György I., Kupai, József, Weiser, Diána Balogh, Greiner, István, Huszthy, Péter, Balogh, György T.
Published in Chemistry : a European journal (02.07.2018)
Published in Chemistry : a European journal (02.07.2018)
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Journal Article
Discovery of novel steroidal histamine H-3 receptor antagonists/inverse agonists. Part 2. Versatile steroidal carboxamide derivatives
Ledneczki, Istvan, Nemethy, Zsolt, Tapolcsanyi, Pal, Eles, Janos, Greiner, Istvan, Gabor, Eszter, Varga, Balazs, Balazs, Ottilia, Roman, Viktor, Levay, Gyorgy, Maho, Sandor
Published in Bioorganic & medicinal chemistry letters (15.10.2019)
Published in Bioorganic & medicinal chemistry letters (15.10.2019)
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Journal Article
“Greener” synthesis of bisphosphonic/dronic acid derivatives
Kovács, Rita, Grün, Alajos, Garadnay, Sándor, Greiner, István, Keglevich, György
Published in Green processing and synthesis (01.04.2014)
Published in Green processing and synthesis (01.04.2014)
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Journal Article
The route from problem to solution in multistep continuous flow synthesis of pharmaceutical compounds
Bana, Péter, Örkényi, Róbert, Lövei, Klára, Lakó, Ágnes, Túrós, György István, Éles, János, Faigl, Ferenc, Greiner, István
Published in Bioorganic & medicinal chemistry (01.12.2017)
Published in Bioorganic & medicinal chemistry (01.12.2017)
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Journal Article
A Mechanistic Study on the Formation of Dronic Acids
Ábrányi-Balogh, Péter, Greiner, István, Keglevich, György
Published in Molecules (Basel, Switzerland) (14.12.2021)
Published in Molecules (Basel, Switzerland) (14.12.2021)
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Journal Article
Selective NR1/2B N-Methyl-d-aspartate Receptor Antagonists among Indole-2-carboxamides and Benzimidazole-2-carboxamides
Borza, István, Bozó, Éva, Barta-Szalai, Gizella, Kiss, Csilla, Tárkányi, Gábor, Demeter, Ádám, Gáti, Tamás, Háda, Viktor, Kolok, Sándor, Gere, Anikó, Fodor, László, Nagy, József, Galgóczy, Kornél, Magdó, Ildikó, Ágai, Béla, Fetter, József, Bertha, Ferenc, Keserü, György M, Horváth, Csilla, Farkas, Sándor, Greiner, István, Domány, György
Published in Journal of medicinal chemistry (08.03.2007)
Published in Journal of medicinal chemistry (08.03.2007)
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Journal Article
Discovery and Characterization of RGH-122, a Potent, Selective, and Orally Bioavailable V1a Receptor Antagonist
Baska, Ferenc, Bozó, Éva, Szeleczky, Zsolt, Szántó, Gábor, Vukics, Krisztina, Szakács, Zoltán, Domány-Kovács, Katalin, Kurkó, Dalma, Vass, Elemér, Thán, Márta, Vastag, Mónika, Temesvári, Krisztina, Lévai, Sándor, Halász, Attila Sándor, Szondiné Kordás, Krisztina, Román, Viktor, Greiner, István, Bata, Imre
Published in Journal of medicinal chemistry (11.01.2024)
Published in Journal of medicinal chemistry (11.01.2024)
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Journal Article
Discovery of Novel Steroid-Based Histamine H3 Receptor Antagonists/Inverse Agonists
Ledneczki, István, Tapolcsányi, Pál, Gábor, Eszter, Éles, János, Barabás, Júlia, Béni, Zoltán, Varga, Balázs, Balázs, Ottilia, Román, Viktor, Fodor, László, Szikra, Judit, Vastag, Mónika, Lévay, György, Schmidt, Éva, Lendvai, Balázs, Greiner, István, Kiss, Béla, Némethy, Zsolt, Mahó, Sándor
Published in Journal of medicinal chemistry (14.03.2024)
Published in Journal of medicinal chemistry (14.03.2024)
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Journal Article
Optimization of Novel α7 Nicotinic Acetylcholine Receptor Positive Allosteric Modulators and the Discovery of a Preclinical Development Candidate Molecule (RGH-560)
Ledneczki, István, Némethy, Zsolt, Molnár, Katalin Dudásné, Tapolcsányi, Pál, Ilkei, Viktor, Vágó, István, Kolok, Sándor, Thán, Márta, Laszy, Judit, Balázs, Ottilia, Krámos, Balázs, Szigetvári, Áron, Bata, Imre, Makó, Attila, Visegrády, András, Fodor, László, Vastag, Mónika, Lévay, György, Lendvai, Balázs, Greiner, István, Éles, János
Published in Journal of medicinal chemistry (14.12.2023)
Published in Journal of medicinal chemistry (14.12.2023)
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Journal Article
Design, synthesis and biological evaluation of novel cyclic malonamide derivatives as selective RIPK1 inhibitors
Petró, József Levente, Bényei, Gyula, Bana, Péter, Linke, Nikolett, Horti, Ferenc, Szabó, Judit Eszter, Szalai, Krisztina Katalin, Hornyánszky, Gábor, Greiner, István, Éles, János
Published in Bioorganic & medicinal chemistry letters (01.03.2024)
Published in Bioorganic & medicinal chemistry letters (01.03.2024)
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Journal Article
Fragment Based Optimization of Metabotropic Glutamate Receptor 2 (mGluR2) Positive Allosteric Modulators in the Absence of Structural Information
Szabó, György, Túrós, György I, Kolok, Sándor, Vastag, Mónika, Sánta, Zsuzsanna, Dékány, Miklós, Lévay, György I, Greiner, István, Natsumi, Minami, Tatsuya, Watanabe, Keserű, György M
Published in Journal of medicinal chemistry (10.01.2019)
Published in Journal of medicinal chemistry (10.01.2019)
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Journal Article
Fragment-Based Optimization of Dihydropyrazino-Benzimidazolones as Metabotropic Glutamate Receptor‑2 Positive Allosteric Modulators against Migraine
Szabó, György, Erdélyi, Péter, Kolok, Sándor, Vastag, Mónika, Halász, Attila S, Kis-Varga, Istvánné, Lévay, György I, Béni, Zoltán, Kóti, János, Greiner, István, Keserű, György M
Published in Journal of medicinal chemistry (24.06.2021)
Published in Journal of medicinal chemistry (24.06.2021)
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Journal Article
Novel-Type GABAB PAMs: Structure–Activity Relationship in Light of the Protein Structure
Krámos, Balázs, Hadady, Zsuzsa, Makó, Attila, Szántó, Gábor, Felföldi, Nóra, Magdó, Ildikó, Bobok, Amrita Ágnes, Bata, Imre, Román, Viktor, Visegrády, András, Keserű, György M., Greiner, István, Éles, János
Published in ACS medicinal chemistry letters (14.03.2024)
Published in ACS medicinal chemistry letters (14.03.2024)
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Journal Article
Synthesis of Hydroxymethylenebisphosphonic Acid Derivatives in Different Solvents
Nagy, Dávid Illés, Grün, Alajos, Garadnay, Sándor, Greiner, István, Keglevich, György
Published in Molecules (11.08.2016)
Published in Molecules (11.08.2016)
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Book Review