Targeting the eIF4F translation initiation complex: a critical nexus for cancer development
Pelletier, Jerry, Graff, Jeremy, Ruggero, Davide, Sonenberg, Nahum
Published in Cancer research (Chicago, Ill.) (15.01.2015)
Published in Cancer research (Chicago, Ill.) (15.01.2015)
Get full text
Journal Article
Pharmacogenetic inhibition of eIF4E-dependent Mmp9 mRNA translation reverses fragile X syndrome-like phenotypes
Gkogkas, Christos G, Khoutorsky, Arkady, Cao, Ruifeng, Jafarnejad, Seyed Mehdi, Prager-Khoutorsky, Masha, Giannakas, Nikolaos, Kaminari, Archontia, Fragkouli, Apostolia, Nader, Karim, Price, Theodore J, Konicek, Bruce W, Graff, Jeremy R, Tzinia, Athina K, Lacaille, Jean-Claude, Sonenberg, Nahum
Published in Cell reports (Cambridge) (11.12.2014)
Published in Cell reports (Cambridge) (11.12.2014)
Get full text
Journal Article
Targeting the Eukaryotic Translation Initiation Factor 4E for Cancer Therapy
GRAFF, Jeremy R, KONICEK, Bruce W, CARTER, Julia H, MARCUSSON, Eric G
Published in Cancer research (Chicago, Ill.) (01.02.2008)
Published in Cancer research (Chicago, Ill.) (01.02.2008)
Get full text
Journal Article
Therapeutic suppression of translation initiation factor eIF4E expression reduces tumor growth without toxicity
Graff, Jeremy R, Konicek, Bruce W, Vincent, Thomas M, Lynch, Rebecca L, Monteith, David, Weir, Spring N, Schwier, Phil, Capen, Andrew, Goode, Robin L, Dowless, Michele S, Chen, Yuefeng, Zhang, Hong, Sissons, Sean, Cox, Karen, McNulty, Ann M, Parsons, Stephen H, Wang, Tao, Sams, Lillian, Geeganage, Sandaruwan, Douglass, Larry E, Neubauer, Blake Lee, Dean, Nicholas M, Blanchard, Kerry, Shou, Jianyong, Stancato, Louis F, Carter, Julia H, Marcusson, Eric G
Published in The Journal of clinical investigation (01.09.2007)
Published in The Journal of clinical investigation (01.09.2007)
Get full text
Journal Article
Inhibition of Mnk kinase activity by cercosporamide and suppressive effects on acute myeloid leukemia precursors
Altman, Jessica K., Szilard, Amy, Konicek, Bruce W., Iversen, Philip W., Kroczynska, Barbara, Glaser, Heather, Sassano, Antonella, Vakana, Eliza, Graff, Jeremy R., Platanias, Leonidas C.
Published in Blood (02.05.2013)
Published in Blood (02.05.2013)
Get full text
Journal Article
Imprime PGG-Mediated Anti-Cancer Immune Activation Requires Immune Complex Formation
Chan, Anissa S H, Jonas, Adria Bykowski, Qiu, Xiaohong, Ottoson, Nadine R, Walsh, Richard M, Gorden, Keith B, Harrison, Ben, Maimonis, Peter J, Leonardo, Steven M, Ertelt, Kathleen E, Danielson, Michael E, Michel, Kyle S, Nelson, Mariana, Graff, Jeremy R, Patchen, Myra L, Bose, Nandita
Published in PloS one (03.11.2016)
Published in PloS one (03.11.2016)
Get full text
Journal Article
Therapeutic Inhibition of MAP Kinase Interacting Kinase Blocks Eukaryotic Initiation Factor 4E Phosphorylation and Suppresses Outgrowth of Experimental Lung Metastases
KONICEK, Bruce W, STEPHENS, Jennifer R, MCCANN, Denis J, PELLETIER, Jerry, FURIC, Luc, YINGLING, Jonathan M, STANCATO, Louis F, SONENBERG, Nahum, GRAFF, Jeremy R, MCNULTY, Ann M, ROBICHAUD, Nathaniel, PEERY, Robert B, DUMSTORF, Chad A, DOWLESS, Michele S, IVERSEN, Philip W, PARSONS, Stephen, ELLIS, Karen E
Published in Cancer research (Chicago, Ill.) (01.03.2011)
Published in Cancer research (Chicago, Ill.) (01.03.2011)
Get full text
Journal Article
Targeting eukaryotic translation in mesothelioma cells with an eIF4E-specific antisense oligonucleotide
Jacobson, Blake A, Thumma, Saritha C, Jay-Dixon, Joseph, Patel, Manish R, Dubear Kroening, K, Kratzke, Marian G, Etchison, Ryan G, Konicek, Bruce W, Graff, Jeremy R, Kratzke, Robert A
Published in PloS one (18.11.2013)
Published in PloS one (18.11.2013)
Get full text
Journal Article
Cotargeting MNK and MEK kinases induces the regression of NF1-mutant cancers
Lock, Rebecca, Ingraham, Rachel, Maertens, Ophélia, Miller, Abigail L, Weledji, Nelly, Legius, Eric, Konicek, Bruce M, Yan, Sau-Chi B, Graff, Jeremy R, Cichowski, Karen
Published in The Journal of clinical investigation (01.06.2016)
Published in The Journal of clinical investigation (01.06.2016)
Get full text
Journal Article
Phosphorylation of eIF4E serine 209 is associated with tumour progression and reduced survival in malignant melanoma
Carter, Julia H, Deddens, James A, Spaulding IV, Nelson Reed, Lucas, Denise, Colligan, Bruce M, Lewis, Thomas Grant, Hawkins, Elyse, Jones, Jordan, Pemberton, Jackson O, Douglass, Larry E, Graff, Jeremy R
Published in British journal of cancer (16.02.2016)
Published in British journal of cancer (16.02.2016)
Get full text
Journal Article
Imprime PGG Enhances Anti-Tumor Effects of Tumor-Targeting, Anti-Angiogenic, and Immune Checkpoint Inhibitor Antibodies
Chan, Anissa S H, Kangas, Takashi O, Qiu, Xiaohong, Uhlik, Mark T, Fulton, Ross B, Ottoson, Nadine R, Gorden, Keith B, Yokoyama, Yumi, Danielson, Michael E, Jevne, Trinda M, Michel, Kyle S, Graff, Jeremy R, Bose, Nandita
Published in Frontiers in oncology (26.05.2022)
Published in Frontiers in oncology (26.05.2022)
Get full text
Journal Article
LY2801653 is an orally bioavailable multi-kinase inhibitor with potent activity against MET, MST1R, and other oncoproteins, and displays anti-tumor activities in mouse xenograft models
Yan, S. Betty, Peek, Victoria L., Ajamie, Rose, Buchanan, Sean G., Graff, Jeremy R., Heidler, Steven A., Hui, Yu-Hua, Huss, Karen L., Konicek, Bruce W., Manro, Jason R., Shih, Chuan, Stewart, Julie A., Stewart, Trent R., Stout, Stephanie L., Uhlik, Mark T., Um, Suzane L., Wang, Yong, Wu, Wenjuan, Yan, Lei, Yang, Wei J., Zhong, Boyu, Walgren, Richard A.
Published in Investigational new drugs (01.08.2013)
Published in Investigational new drugs (01.08.2013)
Get full text
Journal Article
Characterization of LY2228820 dimesylate, a potent and selective inhibitor of p38 MAPK with antitumor activity
Campbell, Robert M, Anderson, Bryan D, Brooks, Nathan A, Brooks, Harold B, Chan, Edward M, De Dios, Alfonso, Gilmour, Raymond, Graff, Jeremy R, Jambrina, Enrique, Mader, Mary, McCann, Denis, Na, Songqing, Parsons, Stephen H, Pratt, Susan E, Shih, Chuan, Stancato, Louis F, Starling, James J, Tate, Courtney, Velasco, Juan A, Wang, Yong, Ye, Xiang S
Published in Molecular cancer therapeutics (01.02.2014)
Published in Molecular cancer therapeutics (01.02.2014)
Get full text
Journal Article
eIF4E Activation Is Commonly Elevated in Advanced Human Prostate Cancers and Significantly Related to Reduced Patient Survival
GRAFF, Jeremy R, KONICEK, Bruce W, HURST, Bernadette M, DEDDENS, James A, NEUBAUER, Blake L, STANCATO, Louis F, CARTER, Harry W, DOUGLASS, Larry E, CARTER, Julia H, LYNCH, Rebecca L, DUMSTORF, Chad A, DOWLESS, Michele S, MCNULTY, Ann M, PARSONS, Stephen H, BRAIL, Leslie H, COLLIGAN, Bruce M, KOOP, Jonathan W
Published in Cancer research (Chicago, Ill.) (01.05.2009)
Published in Cancer research (Chicago, Ill.) (01.05.2009)
Get full text
Journal Article
Immune Pharmacodynamic Responses of the Novel Cancer Immunotherapeutic Imprime PGG in Healthy Volunteers
Bose, Nandita, Ottoson, Nadine R, Qiu, Xiaohong, Harrison, Ben, Lowe, Jamie R, Uhlik, Mark T, Rathmann, Blaine T, Kangas, Takashi O, Jordan, Lindsay R, Ertelt, Kathleen E, Jonas, Adria Bykowski, Walsh, Richard M, Chan, Anissa S H, Fulton, Ross B, Leonardo, Steven M, Fraser, Kathryn A, Gorden, Keith B, Matson, Mark A, Graff, Jeremy R, Huhn, Richard D
Published in The Journal of immunology (1950) (15.05.2019)
Published in The Journal of immunology (1950) (15.05.2019)
Get full text
Journal Article
The protein kinase Cβ-selective inhibitor, enzastaurin (LY317615.HCI), suppresses signaling through the AKT pathway, induces apoptosis, and suppresses growth of human colon cancer and glioblastoma xenografts
GRAFF, Jeremy R, MCNULTY, Ann M, SAMS, Lillian, HUSS, Karen L, CAMPBELL, Robert M, IVERSEN, Philip W, NEUBAUER, Blake Lee, BROWN, Thomas J, MUSIB, Luna, GEEGANAGE, Sandaruwan, THORNTON, Donald, ROSS HANNA, Kimberly, KONICEK, Bruce W, LYNCH, Rebecca L, BAILEY, Spring N, BANKS, Crystal, CAPEN, Andrew, GOODE, Robin, LEWIS, Jason E
Published in Cancer research (Chicago, Ill.) (15.08.2005)
Published in Cancer research (Chicago, Ill.) (15.08.2005)
Get full text
Journal Article
Targeting the eIF4F translation initiation complex for cancer therapy
Konicek, Bruce W., Dumstorf, Chad A., Graff, Jeremy R.
Published in Cell cycle (Georgetown, Tex.) (15.08.2008)
Published in Cell cycle (Georgetown, Tex.) (15.08.2008)
Get full text
Journal Article
Abstract LB-087: Imprime PGG drives adaptive immune resistance within the tumor microenvironment by modulating the myeloid compartment and enhances the efficacy of anti-PD1 antibody in vivo
Bykowski Jonas, Adria L., Chan, Anissa SH, Ottoson, Nadine R., Qiu, Xiaohong, Fraser, Kathryn, Kangas, Takashi O., Fulton, Ross, Rathmann, Blaine, Graff, Jeremy R., Bose, Nandita
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Get full text
Journal Article