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Highly Efficient Asymmetric Synthesis of Sitagliptin

Highly Efficient Asymmetric Synthesis of Sitagliptin

by Hansen, Karl B, Hsiao, Yi, Xu, Feng, Rivera, Nelo, Clausen, Andrew, Kubryk, Michele, Krska, Shane, Rosner, Thorsten, Simmons, Bryon, Balsells, Jaume, Ikemoto, Nori, Sun, Yongkui, Spindler, Felix, Malan, Christophe, Grabowski, Edward J. J, Armstrong, Joseph D
Published in Journal of the American Chemical Society (01.07.2009)

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Correction to “Highly Efficient Asymmetric Synthesis of Sitagliptin”

Correction to “Highly Efficient Asymmetric Synthesis of Sitagliptin”

by Hansen, Karl B, Hsiao, Yi, Xu, Feng, Rivera, Nelo, Clausen, Andrew, Kubryk, Michele, Krska, Shane, Rosner, Thorsten, Simmons, Bryon, Balsells, Jaume, Ikemoto, Nori, Sun, Yongkui, Spindler, Felix, Malan, Christophe, Grabowski, Edward J. J
Published in Journal of the American Chemical Society (05.08.2020)

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Synthesis of Substituted Imidazoles via Organocatalysis

Synthesis of Substituted Imidazoles via Organocatalysis

by Frantz, Doug E, Morency, Louis, Soheili, Arash, Murry, Jerry A, Grabowski, Edward J. J, Tillyer, Richard D
Published in Organic letters (04.03.2004)

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Highly Efficient Synthesis of β-Amino Acid Derivatives via Asymmetric Hydrogenation of Unprotected Enamines

Highly Efficient Synthesis of β-Amino Acid Derivatives via Asymmetric Hydrogenation of Unprotected Enamines

by Hsiao, Yi, Rivera, Nelo R, Rosner, Thorsten, Krska, Shane W, Njolito, Eugenia, Wang, Fang, Sun, Yongkui, Armstrong, Joseph D, Grabowski, Edward J. J, Tillyer, Richard D, Spindler, Felix, Malan, Christophe
Published in Journal of the American Chemical Society (18.08.2004)

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Stereoselective Formation of Carbon−Carbon Bonds via SN2-Displacement: Synthesis of Substituted Cycloalkyl[b]indoles

Stereoselective Formation of Carbon−Carbon Bonds via SN2-Displacement: Synthesis of Substituted Cycloalkyl[b]indoles

by Hillier, Michael C, Marcoux, Jean-François, Zhao, Dalian, Grabowski, Edward J. J, McKeown, Arlene E, Tillyer, Richard D
Published in Journal of organic chemistry (14.10.2005)

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Asymmetric Synthesis of a Prostaglandin D2 Receptor Antagonist

Asymmetric Synthesis of a Prostaglandin D2 Receptor Antagonist

by Campos, Kevin R, Journet, Michel, Lee, Sandra, Grabowski, Edward J. J, Tillyer, Richard D
Published in Journal of organic chemistry (07.01.2005)

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Mechanistic Evidence for an α-Oxoketene Pathway in the Formation of β-Ketoamides/Esters via Meldrum's Acid Adducts

Mechanistic Evidence for an α-Oxoketene Pathway in the Formation of β-Ketoamides/Esters via Meldrum's Acid Adducts

by Xu, Feng, Armstrong, Joseph D, Zhou, George X, Simmons, Bryon, Hughes, David, Ge, Zhihong, Grabowski, Edward J. J
Published in Journal of the American Chemical Society (13.10.2004)

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Stereoselective Carbon−Carbon Bond Formation via the Mitsunobu Displacement of Chiral Secondary Benzylic Alcohols

Stereoselective Carbon−Carbon Bond Formation via the Mitsunobu Displacement of Chiral Secondary Benzylic Alcohols

by Hillier, Michael C, Desrosiers, Jean-Nicolas, Marcoux, Jean-François, Grabowski, Edward J. J
Published in Organic letters (19.02.2004)

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Asymmetric Hydrogenation of N-Sulfonylated-α-dehydroamino Acids: Toward the Synthesis of an Anthrax Lethal Factor Inhibitor

Asymmetric Hydrogenation of N-Sulfonylated-α-dehydroamino Acids: Toward the Synthesis of an Anthrax Lethal Factor Inhibitor

by Shultz, C. Scott, Dreher, Spencer D, Ikemoto, Norihiro, Williams, J. Michael, Grabowski, Edward J. J, Krska, Shane W, Sun, Yongkui, Dormer, Peter G, DiMichele, Lisa
Published in Organic letters (04.08.2005)

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First Generation Process for the Preparation of the DPP-IV Inhibitor Sitagliptin

First Generation Process for the Preparation of the DPP-IV Inhibitor Sitagliptin

by Hansen, Karl B, Balsells, Jaume, Dreher, Spencer, Hsiao, Yi, Kubryk, Michele, Palucki, Michael, Rivera, Nelo, Steinhuebel, Dietrich, Armstrong, Joseph D, Askin, David, Grabowski, Edward J. J
Published in Organic process research & development (01.09.2005)

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Practical Asymmetric Synthesis of a Potent PDE4 Inhibitor via Stereoselective Enolate Alkylation of a Chiral Aryl−Heteroaryl Secondary Tosylate

Practical Asymmetric Synthesis of a Potent PDE4 Inhibitor via Stereoselective Enolate Alkylation of a Chiral Aryl−Heteroaryl Secondary Tosylate

by O'Shea, Paul D, Chen, Cheng-yi, Chen, Weirong, Dagneau, Philippe, Frey, Lisa F, Grabowski, Edward J. J, Marcantonio, Karen M, Reamer, Robert A, Tan, Lushi, Tillyer, Richard D, Roy, Amélie, Wang, Xin, Zhao, Dalian
Published in Journal of organic chemistry (15.04.2005)

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A Novel, Highly Enantioselective Ketone Alkynylation Reaction Mediated by Chiral Zinc Aminoalkoxides

A Novel, Highly Enantioselective Ketone Alkynylation Reaction Mediated by Chiral Zinc Aminoalkoxides

by Tan, Lushi, Chen, Cheng-yi, Tillyer, Richard D., Grabowski, Edward J. J., Reider, Paul J.
Published in Angewandte Chemie (International ed.) (01.03.1999)

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Practical Asymmetric Synthesis of a Potent Cathepsin K Inhibitor. Efficient Palladium Removal Following Suzuki Coupling

Practical Asymmetric Synthesis of a Potent Cathepsin K Inhibitor. Efficient Palladium Removal Following Suzuki Coupling

by Chen, Cheng-yi, Dagneau, Philippe, Grabowski, Edward J. J, Oballa, Renata, O'Shea, Paul, Prasit, Peppi, Robichaud, Joël, Tillyer, Rich, Wang, Xin
Published in Journal of organic chemistry (04.04.2003)

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Highly Diastereoselective Heterogeneously Catalyzed Hydrogenation of Enamines for the Synthesis of Chiral β-Amino Acid Derivatives

Highly Diastereoselective Heterogeneously Catalyzed Hydrogenation of Enamines for the Synthesis of Chiral β-Amino Acid Derivatives

by Ikemoto, Norihiro, Tellers, David M, Dreher, Spencer D, Liu, Jinchu, Huang, Angie, Rivera, Nelo R, Njolito, Eugenia, Hsiao, Yi, McWilliams, J. Christopher, Williams, J. Michael, Armstrong, Joseph D, Sun, Yongkui, Mathre, David J, Grabowski, Edward J. J, Tillyer, Richard D
Published in Journal of the American Chemical Society (17.03.2004)

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Practical Synthesis of a Potent Hepatitis C Virus RNA Replication Inhibitor

Practical Synthesis of a Potent Hepatitis C Virus RNA Replication Inhibitor

by Bio, Matthew M, Xu, Feng, Waters, Marjorie, Williams, J. Michael, Savary, Kimberly A, Cowden, Cameron J, Yang, Chunhua, Buck, Elizabeth, Song, Zhiguo J, Tschaen, David M, Volante, R. P, Reamer, Robert A, Grabowski, Edward J. J
Published in Journal of organic chemistry (17.09.2004)

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Practical Asymmetric Synthesis of Aprepitant, a Potent Human NK-1 Receptor Antagonist, via a Stereoselective Lewis Acid-Catalyzed Trans Acetalization Reaction

Practical Asymmetric Synthesis of Aprepitant, a Potent Human NK-1 Receptor Antagonist, via a Stereoselective Lewis Acid-Catalyzed Trans Acetalization Reaction

by Zhao, Matthew M, McNamara, James M, Ho, Guo-Jie, Emerson, Khateeta M, Song, Zhiguo J, Tschaen, David M, Brands, Karel M. J, Dolling, Ulf-H, Grabowski, Edward J. J, Reider, Paul J, Cottrell, Ian F, Ashwood, Michael S, Bishop, Brian C
Published in Journal of organic chemistry (20.09.2002)

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Lithium Ephedrate-Mediated Addition of a Lithium Acetylide to a Ketone: Solution Structures and Relative Reactivities of Mixed Aggregates Underlying the High Enantioselectivities

Lithium Ephedrate-Mediated Addition of a Lithium Acetylide to a Ketone: Solution Structures and Relative Reactivities of Mixed Aggregates Underlying the High Enantioselectivities

by Thompson, Andrew, Corley, Edward G, Huntington, Martha F, Grabowski, Edward J. J, Remenar, Julius F, Collum, David B
Published in Journal of the American Chemical Society (11.03.1998)

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Lithium Alkoxides of Cinchona Alkaloids as Chiral Controllers for Enantioselective Acetylide Addition to Cyclic N-Acyl Ketimines

Lithium Alkoxides of Cinchona Alkaloids as Chiral Controllers for Enantioselective Acetylide Addition to Cyclic N-Acyl Ketimines

by Huffman, Mark A, Yasuda, Nobuyoshi, DeCamp, Ann E, Grabowski, Edward J. J
Published in Journal of organic chemistry (01.03.1995)

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Highly Enantioselective 1,2-Addition of Lithium Acetylide-Ephedrate Complexes: Spectroscopic Evidence for Reaction Proceeding via a 2:2 Tetramer, and X-ray Characterization of Related Complexes

Highly Enantioselective 1,2-Addition of Lithium Acetylide-Ephedrate Complexes: Spectroscopic Evidence for Reaction Proceeding via a 2:2 Tetramer, and X-ray Characterization of Related Complexes

by Xu, Feng, Reamer, Robert A, Tillyer, Richard, Cummins, Jordan M, Grabowski, Edward J. J, Reider, Paul J, Collum, David B, Huffman, John C
Published in Journal of the American Chemical Society (15.11.2000)

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Highly regioselective synthesis of 1-aryl-3,4,5-substituted pyrazoles

Highly regioselective synthesis of 1-aryl-3,4,5-substituted pyrazoles

by Gosselin, Francis, O'Shea, Paul D., Webster, Robert A., Reamer, Robert A., Tillyer, Richard D., Grabowski, Edward J. J.
Published in Synlett (01.12.2006)

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