Orally active, nonpeptide oxytocin antagonists
Evans, Ben E, Leighton, James L, Rittle, Kenneth E, Gilbert, Kevin F, Lundell, George F, Gould, Norman P, Hobbs, Doug W, DiPardo, Robert M, Veber, Daniel F, Pettibone, Douglas J, Clineschmidt, Bradley V, Anderson, Paul S, Freidinger, Roger M
Published in Journal of medicinal chemistry (01.10.1992)
Published in Journal of medicinal chemistry (01.10.1992)
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Use of N-Fmoc amino acid chlorides and activated 2-(fluorenylmethoxy)-5(4H)-oxazolones in solid-phase peptide synthesis. Efficient syntheses of highly N-alkylated cyclic hexapeptide oxytocin antagonists related to L-365,209
Perlow, Debra S, Erb, Jill M, Gould, Norman P, Tung, Roger D, Freidinger, Roger M, Williams, Peter D, Veber, Daniel F
Published in Journal of organic chemistry (01.07.1992)
Published in Journal of organic chemistry (01.07.1992)
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Development of a novel class of cyclic hexapeptide oxytocin antagonists based on a natural product
Williams, Peter D, Bock, Mark G, Tung, Roger D, Garsky, Victor M, Perlow, Debra S, Erb, Jill M, Lundell, G. F, Gould, Norman P, Whitter, Willie L
Published in Journal of medicinal chemistry (01.10.1992)
Published in Journal of medicinal chemistry (01.10.1992)
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NANOMOLAR-AFFINITY, NONPEPTIDE OXYTOCIN RECEPTOR ANTAGONISTS
EVANS, BE, LUNDELL, GF, GILBERT, KF, BOCK, MG, RITTLE, KE, CARROLL, LA, WILLIAMS, PD, PAWLUCZYK, JM, LEIGHTON, JL, YOUNG, MB, ERB, JM, HOBBS, DW, GOULD, NP, DIPARDO, RM, HOFFMAN, JB, PERLOW, DS, WHITTER, WL, VEBER, DF, PETTIBONE, DJ, CLINESCHMIDT, BV, ANDERSON, PS, FREIDINGER, RM
Published in Journal of medicinal chemistry (10.12.1993)
Published in Journal of medicinal chemistry (10.12.1993)
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Design of nonpeptidal ligands for a peptide receptor: cholecystokinin antagonists
Evans, B. E, Rittle, K. E, Bock, M. G, DiPardo, R. M, Freidinger, R. M, Whitter, W. L, Gould, N. P, Lundell, G. F, Homnick, C. F
Published in Journal of medicinal chemistry (01.07.1987)
Published in Journal of medicinal chemistry (01.07.1987)
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Novel glutamic acid-derived cholecystokinin receptor ligands
Freidinger, R. M, Whitter, W. L, Gould, N. P, Holloway, M. K, Chang, R. S. L, Lotti, V. J
Published in Journal of medicinal chemistry (01.02.1990)
Published in Journal of medicinal chemistry (01.02.1990)
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Agents for the treatment of brain edema. 2. [(2,3,9,9a-Tetrahydro-3-oxo-9a-substituted-1H-fluoren-7-yl)oxy]alkanoic acids and some of their analogs
Cragoe, E. J, Woltersdorf, O. W, Gould, N. P, Pietruszkiewicz, A. M, Ziegler, C, Sakurai, Y, Stokker, G. E, Anderson, P. S, Bourke, R. S
Published in Journal of medicinal chemistry (01.05.1986)
Published in Journal of medicinal chemistry (01.05.1986)
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3-Hydroxy-3-methylglutaryl-coenzyme A reductase inhibitors. 2. Structural modification of 7-(substituted aryl)-3,5-dihydroxy-6-heptenoic acids and their lactone derivatives
Hoffman, William F, Alberts, A. W, Cragoe, E. J, Deana, A. A, Evans, B. E, Gilfillan, J. L, Gould, N. P, Huff, J. W, Novello, F. C
Published in Journal of medicinal chemistry (01.02.1986)
Published in Journal of medicinal chemistry (01.02.1986)
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Journal Article
Design and discovery in the development of long-acting renin inhibitors
Veber, D F, Payne, L S, Williams, P D, Perlow, D S, Lundell, G F, Gould, N P, Siegl, P K, Sweet, C S, Freidinger, R M
Published in Biochemical Society transactions (01.12.1990)
Published in Biochemical Society transactions (01.12.1990)
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Agents for the treatment of brain injury. 1. (Aryloxy)alkanoic acids
Cragoe, E. J, Gould, N. P, Woltersdorf, O. W, Ziegler, C, Bourke, R. S, Nelson, L. R, Kimelberg, H. K, Waldman, J. B, Popp, A. J, Sedransk, N
Published in Journal of medicinal chemistry (01.05.1982)
Published in Journal of medicinal chemistry (01.05.1982)
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Prostaglandin isosteres. 2. Chain-modified thiazolidinone prostaglandin analogs as renal vasodilators
Bicking, John B, Bock, Mark G, Cragoe, Edward J, DiPardo, Robert M, Gould, Norman, Holtz, Wilbur J, Lee, T. J, Robb, Charles M, Smith, Robert L
Published in Journal of medicinal chemistry (01.03.1983)
Published in Journal of medicinal chemistry (01.03.1983)
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11,12-Secoprostaglandins. 3. 8-Alkylthio(sulfinyl and sulfonyl)-12-hydroxyalkanoic acids and related compounds
Smith, Robert L, Bicking, John B, Gould, Norman P, Lee, Ta-Jyh, Robb, Charles M, Kuehl, Frederick A, Mandel, Lewis R, Cragoe, Edward J
Published in Journal of medicinal chemistry (01.04.1977)
Published in Journal of medicinal chemistry (01.04.1977)
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