Eyes on Topical Ocular Disposition: The Considered Design of a Lead Janus Kinase (JAK) Inhibitor That Utilizes a Unique Azetidin-3-Amino Bridging Scaffold to Attenuate Off-Target Kinase Activity, While Driving Potency and Aqueous Solubility
Gordhan, Heeren M., Miller, Steven T., Clancy, Daphne C., Ina, Maria, McDougal, Alan V., Cutno, D’Quan K., Brown, Robert V., Lichorowic, Cynthia L., Sturdivant, Jill M., Vick, Kyle A., Williams, Stuart S., deLong, Mitchell A., White, Jeffrey C., Kopczynski, Casey C., Ellis, David A.
Published in Journal of medicinal chemistry (13.07.2023)
Published in Journal of medicinal chemistry (13.07.2023)
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Journal Article
Evaluation of substituted ebselen derivatives as potential trypanocidal agents
Gordhan, Heeren M., Patrick, Stephen L., Swasy, Maria I., Hackler, Amber L., Anayee, Mark, Golden, Jennifer E., Morris, James C., Whitehead, Daniel C.
Published in Bioorganic & medicinal chemistry letters (01.02.2017)
Published in Bioorganic & medicinal chemistry letters (01.02.2017)
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Journal Article
A targeted delivery strategy for the development of potent trypanocides
Gordhan, Heeren M., Milanes, Jillian E., Qiu, Yijian, Golden, Jennifer E., Christensen, Kenneth A., Morris, James C., Whitehead, Daniel C.
Published in Chemical communications (Cambridge, England) (11.08.2017)
Published in Chemical communications (Cambridge, England) (11.08.2017)
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Journal Article
아제티디닐 피리미딘 및 그의 용도
DELONG MITCHELL A, GORDHAN HEEREN M, SENCHYNA MICHELLE, WHITE JEFFREY C, LICHOROWIC CYNTHIA L, KOPCZYNSKI CASEY, HOLLANDER DAVID, ELLIS DAVID ARCHER, STURDIVANT JILL M
Year of Publication 07.03.2024
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Year of Publication 07.03.2024
Patent
A targeted delivery strategy for the development of potent trypanocidesElectronic supplementary information (ESI) available: Full experimental details and physical data for all new compounds. See DOI: 10.1039/c7cc03378h
Gordhan, Heeren M, Milanes, Jillian E, Qiu, Yijian, Golden, Jennifer E, Christensen, Kenneth A, Morris, James C, Whitehead, Daniel C
Year of Publication 01.08.2017
Year of Publication 01.08.2017
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Journal Article
N-SUBSTITUTED C6 CYCLYL CARBOXAMIDE COMPOUNDS AND USES THEREOF
deLong, Mitchell A, Ellis, David Archer, Lichorowic, Cynthia L, Gordhan, Heeren M, Sturdivant, Jill M
Year of Publication 31.10.2024
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Year of Publication 31.10.2024
Patent
N-SUBSTITUTED C6 CYCLYL CARBOXAMIDE COMPOUNDS AND USES THEREOF
GORDHAN, Heeren M, DELONG, Mitchell A, STURDIVANT, Jill M, LICHOROWIC, Cynthia L, ELLIS, David Archer
Year of Publication 24.10.2024
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Year of Publication 24.10.2024
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JANUS KINASE INHIBITING PYRAZOLE COMPOUNDS AND USES THEREOF
STURDIVANT, Jill, M, ELLIS, David, Archer, GORDHAN, Heeren, M, LICHOROWIC, Cynthia, L, DELONG, Mitchell, A
Year of Publication 14.08.2024
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Year of Publication 14.08.2024
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Azetidinyl Pyrimidines and Uses Thereof
deLong, Mitchell A, Ellis, David Archer, Lichorowic, Cynthia L, Gordhan, Heeren M, Sturdivant, Jill M
Year of Publication 04.01.2024
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Year of Publication 04.01.2024
Patent
AZETIDINYL PYRIMIDINES AND USES THEREOF AS JAK INHIBITORS
GORDHAN, Heeren M, DELONG, Mitchell A, STURDIVANT, Jill M, LICHOROWIC, Cynthia L, ELLIS, David Archer
Year of Publication 04.01.2024
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Year of Publication 04.01.2024
Patent
JANUS KINASE INHIBITING PYRAZOLE COMPOUNDS AND USES THEREOF
GORDHAN, HEEREN M, DELONG, MITCHELL A, LICHOROWIC, CYNTHIA L, ELLIS, DAVID ARCHER, STURDIVANT, JILL M
Year of Publication 13.04.2023
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Year of Publication 13.04.2023
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HETEROBICYCLIC CARBOXAMIDES AND USES THEREOF
deLong, Mitchell A, Lichorowic, Cynthia L, Gordhan, Heeren M, Sturdivant, Jill M
Year of Publication 05.01.2023
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Year of Publication 05.01.2023
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POLYMORPHS OF A JAK1/TYK2 INHIBITOR AND USES THEREOF
MCCLURE, Michael S, GORDHAN, Heeren M, HAXELL, Thomas Francis Nelson, DELONG, Mitchell A, COOLEY, Bob E, ELLIS, David Archer, MCIVER, Andrew Louis
Year of Publication 11.07.2024
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Year of Publication 11.07.2024
Patent
AZETIDINYL PYRIMIDINES AND USES THEREOF
HOLLANDER, David, GORDHAN, Heeren M, DELONG, Mitchell A, STURDIVANT, Jill M, KOPCZYNSKI, Casey, LICHOROWIC, Cynthia L, ELLIS, David Archer, WHITE, Jeffrey C, SENCHYNA, Michelle
Year of Publication 08.05.2024
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Year of Publication 08.05.2024
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Azetidinyl pyrimidines and uses thereof
Jill M. STURDIVANT, Mitchell A. DELONG, David Archer ELLIS, Cynthia L. LICHOROWIC, Heeren M. GORDHAN, Michelle SENCHYNA, David HOLLANDER, Casey KOPCZYNSKI, Jeffrey C. WHITE
Year of Publication 01.03.2024
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Year of Publication 01.03.2024
Patent
AZETIDINYL PYRIMIDINES AND USES THEREOF
HOLLANDER, David, GORDHAN, Heeren M, DELONG, Mitchell A, STURDIVANT, Jill M, KOPCZYNSKI, Casey, LICHOROWIC, Cynthia L, ELLIS, David Archer, WHITE, Jeffrey C, SENCHYNA, Michelle
Year of Publication 04.01.2024
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Year of Publication 04.01.2024
Patent
AZETIDINYL PYRIMIDINES AND USES THEREOF
HOLLANDER, David, GORDHAN, Heeren M, DELONG, Mitchell A, STURDIVANT, Jill M, KOPCZYNSKI, Casey, LICHOROWIC, Cynthia L, ELLIS, David Archer, WHITE, Jeffrey C, SENCHYNA, Michelle
Year of Publication 05.01.2023
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Year of Publication 05.01.2023
Patent
AZETIDINYL PYRIMIDINES AND USES THEREOF
GORDHAN, HEEREN M, WHITE, JEFFREY C, DELONG, MITCHELL A, LICHOROWIC, CYNTHIA L, HOLLANDER, DAVID, ELLIS, DAVID ARCHER, SENCHYNA, MICHELLE, KOPCZYNSKI, CASEY, STURDIVANT, JILL M
Year of Publication 05.01.2023
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Year of Publication 05.01.2023
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AZETIDINYL PYRIMIDINES AND USES THEREOF
KOPCZYNSKI Casey, STURDIVANT Jill M, LICHOROWIC Cynthia L, SENCHYNA Michelle, DELONG Mitchell A, ELLIS David Archer, WHITE Jeffrey C, HOLLANDER David, GORDHAN Heeren M
Year of Publication 31.01.2024
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Year of Publication 31.01.2024
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