New Antibacterial Agents Derived from the DNA Gyrase Inhibitor Cyclothialidine
Angehrn, Peter, Buchmann, Stefan, Funk, Christoph, Goetschi, Erwin, Gmuender, Hans, Hebeisen, Paul, Kostrewa, Dirk, Link, Helmut, Luebbers, Thomas, Masciadri, Raffaello, Nielsen, Joergen, Reindl, Peter, Ricklin, Fabienne, Schmitt-Hoffmann, Anne, Theil, Frank-Peter
Published in Journal of medicinal chemistry (11.03.2004)
Published in Journal of medicinal chemistry (11.03.2004)
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Journal Article
Discovery of Balovaptan, a Vasopressin la Receptor Antagonist for the Treatment of Autism Spectrum Disorder
Schnider, Patrick, Bissantz, Caterina, Bruns, Andreas, Dolente, Cosimo, Goetschi, Erwin, Jakob-Roetne, Roland, Kuennecke, Basil, Mueggler, Thomas, Muster, Wolfgang, Parrott, Neil, Pinard, Emmanuel, Ratni, Hasane, Risterucci, Celine, Rogers-Evans, Mark, von Kienlin, Markus, Grundschober, Christophe
Published in Journal of medicinal chemistry (27.02.2020)
Published in Journal of medicinal chemistry (27.02.2020)
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Journal Article
Discovery of Balovaptan, a Vasopressin 1a Receptor Antagonist for the Treatment of Autism Spectrum Disorder
Schnider, Patrick, Bissantz, Caterina, Bruns, Andreas, Dolente, Cosimo, Goetschi, Erwin, Jakob-Roetne, Roland, Künnecke, Basil, Mueggler, Thomas, Muster, Wolfgang, Parrott, Neil, Pinard, Emmanuel, Ratni, Hasane, Risterucci, Céline, Rogers-Evans, Mark, von Kienlin, Markus, Grundschober, Christophe
Published in Journal of medicinal chemistry (27.02.2020)
Published in Journal of medicinal chemistry (27.02.2020)
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Journal Article
A New DNA Gyrase Inhibitor Subclass of the Cyclothialidine Family Based on a Bicyclic Dilactam−Lactone Scaffold. Synthesis and Antibacterial Properties
Angehrn, Peter, Goetschi, Erwin, Gmuender, Hans, Hebeisen, Paul, Hennig, Michael, Kuhn, Bernd, Luebbers, Thomas, Reindl, Peter, Ricklin, Fabienne, Schmitt-Hoffmann, Anne
Published in Journal of medicinal chemistry (14.04.2011)
Published in Journal of medicinal chemistry (14.04.2011)
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Journal Article
New Anti-MRSA and Anti-VRE Carbapenems; Synthesis and Structure-activity Relationships of 1.BETA.-Metyl-2-(thiazol-2-ylthio)carbapenems
SUNAGAWA, MAKOTO, ITOH, MASANORI, KUBOTA, KATSUMI, SASAKI, AKIRA, UEDA, YUTAKA, ANGEHRN, PETER, BOURSON, ANNE, GOETSCHI, ERWIN, HEBEISEN, PAUL, THEN, RUDOLF L.
Published in Journal of antibiotics (2002)
Published in Journal of antibiotics (2002)
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Synthesis and characterization of 1,3-dihydro-benzo[ b][1,4]diazepin-2-one derivatives: Part 4. In vivo active potent and selective non-competitive metabotropic glutamate receptor 2/3 antagonists
Woltering, Thomas J., Wichmann, Jürgen, Goetschi, Erwin, Knoflach, Frédéric, Ballard, Theresa M., Huwyler, Jörg, Gatti, Silvia
Published in Bioorganic & medicinal chemistry letters (01.12.2010)
Published in Bioorganic & medicinal chemistry letters (01.12.2010)
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Journal Article
From the DNA Gyrase Inhibitor Cyclothialidine to a New Class of Antibacterial Agents
Erwin Goetschi, Fabienne Ricklin, Peter Reindl, Raffaello Masciadri, Thomas Luebbers, Helmut Link, Dirk Kostrewa, Paul Hebeisen, Hans Gmuender, Peter Angehrn, Frank-Peter Theil
Published in Chimia (01.01.2003)
Published in Chimia (01.01.2003)
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Journal Article
P1‐246: N‐heteroaryl‐piperidinyl‐4‐amines as selective GAMMA secretase modulators for the potential treatment of Alzheimer's disease
Luebbers, Thomas, Limberg, Anja, Jolidon, Synese, Goetschi, Erwin, Jacobsen, Helmut, Green, Luke, Flohr, Alexander, Thomas, Andrew, Knust, Henner, David‐Pierson, Pascale, Baumann, Karlheinz
Published in Alzheimer's & dementia (01.07.2012)
Published in Alzheimer's & dementia (01.07.2012)
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Journal Article
N-heteroaryl-piperidinyl-4-amines as selective GAMMA secretase modulators for the potential treatment of Alzheimer's disease
Luebbers, Thomas, Limberg, Anja, Jolidon, Synese, Goetschi, Erwin, Jacobsen, Helmut, Green, Luke, Flohr, Alexander, Thomas, Andrew, Knust, Henner, David-Pierson, Pascale, Baumann, Karlheinz
Published in Alzheimer's & dementia (01.07.2012)
Published in Alzheimer's & dementia (01.07.2012)
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Journal Article
P2‐477: Aminopyrimidines as selective γ‐secretase modulators for the potential treatment of AD
Limberg, Anja, Luebbers, Thomas, Goetschi, Erwin, Jolidon, Synese, Laurence, Ozmen, Jacobsen, Helmut, David‐Pierson, Pascale, Flohr, Alexander, Baumann, Karlheinz
Published in Alzheimer's & dementia (01.07.2011)
Published in Alzheimer's & dementia (01.07.2011)
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Journal Article
Aminopyrimidines as selective γ-secretase modulators for the potential treatment of AD
Limberg, Anja, Luebbers, Thomas, Goetschi, Erwin, Jolidon, Synese, Laurence, Ozmen, Jacobsen, Helmut, David-Pierson, Pascale, Flohr, Alexander, Baumann, Karlheinz
Published in Alzheimer's & dementia (01.07.2011)
Published in Alzheimer's & dementia (01.07.2011)
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Journal Article
Synthesis and characterization of 8-ethynyl-1,3-dihydro-benzo[ b][1,4]diazepin-2-one derivatives: Part 2. New potent non-competitive metabotropic glutamate receptor 2/3 antagonists
Woltering, Thomas J., Adam, Geo, Wichmann, Jürgen, Goetschi, Erwin, Kew, James N.C., Knoflach, Frédéric, Mutel, Vincent, Gatti, Silvia
Published in Bioorganic & medicinal chemistry (01.02.2008)
Published in Bioorganic & medicinal chemistry (01.02.2008)
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Journal Article
PYRIDINE AND PYRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS
GATTI MCARTHUR SILVIA, WOLTERING THOMAS JOHANNES, GOETSCHI ERWIN, WICHMANN JUERGEN
Year of Publication 12.04.2012
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Year of Publication 12.04.2012
Patent
Synthesis and characterization of 1,3-dihydro-benzo[ b][1,4]diazepin-2-one derivatives: Part 3. New potent non-competitive metabotropic glutamate receptor 2/3 antagonists
Woltering, Thomas J., Wichmann, Jürgen, Goetschi, Erwin, Adam, Geo, Kew, James N.C., Knoflach, Frédéric, Ballard, Theresa M., Huwyler, Jörg, Mutel, Vincent, Gatti, Silvia
Published in Bioorganic & medicinal chemistry (15.04.2008)
Published in Bioorganic & medicinal chemistry (15.04.2008)
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Journal Article
HETEROCYCLIC GAMMA SECRETASE MODULATORS
GOETSCHI ERWIN, LUEBBERS THOMAS, BAUMANN KARLHEINZ, JOLIDON SYNESE, LIMBERG ANJA
Year of Publication 20.07.2011
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Year of Publication 20.07.2011
Patent
Synthesis and characterization of 8-ethynyl-1,3-dihydrobenzo[b][1,4]diazepin-2-one derivatives: Part 2. New potent non-competitive metabotropic glutamate receptor 2/3 antagonists
WELTERING, Thomas J, ADAM, Geo, WICHMANN, Jürgen, GOETSCHI, Erwin, KEW, James N. C, KNOFLACH, Frédéric, MUTEL, Vincent, GATTI, Silvia
Published in Bioorganic & medicinal chemistry letters (2008)
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Published in Bioorganic & medicinal chemistry letters (2008)
Journal Article
MODULATORS FOR AMYLOID BETA
JACOBSEN HELMUT, FLOHR ALEXANDER, GOETSCHI ERWIN, LUEBBERS THOMAS, BAUMANN KARLHEINZ, JOLIDON SYNESE
Year of Publication 04.11.2010
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Year of Publication 04.11.2010
Patent
MODULATORS FOR AMYLOID BETA
JACOBSEN HELMUT, FLOHR ALEXANDER, GOETSCHI ERWIN, LUEBBERS THOMAS, BAUMANN KARLHEINZ, JOLIDON SYNESE
Year of Publication 17.08.2010
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Year of Publication 17.08.2010
Patent
SPIRO-5,6-DIHYDRO-4H-2,3,5,10B-TETRAAZA-BENZO[E]AZULENES
MASCIADRI RAFFAELLO, SCHNIDER PATRICK, JAKOB ROETNE ROLAND, ROGERS EVANS MARK, PINARD EMMANUEL, BISSANTZ CATERINA, GOETSCHI ERWIN, RATNI HASANE
Year of Publication 30.06.2011
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Year of Publication 30.06.2011
Patent