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Ghosh, Rajarshi, Wang, Likun, Wang, Eric S., Perera, B. Gayani K., Igbaria, Aeid, Morita, Shuhei, Prado, Kris, Thamsen, Maike, Caswell, Deborah, Macias, Hector, Weiberth, Kurt F., Gliedt, Micah J., Alavi, Marcel V., Hari, Sanjay B., Mitra, Arinjay K., Bhhatarai, Barun, Schürer, Stephan C., Snapp, Erik L., Gould, Douglas B., German, Michael S., Backes, Bradley J., Maly, Dustin J., Oakes, Scott A., Papa, Feroz R.
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Discovery of RMC-5552, a Selective Bi-Steric Inhibitor of mTORC1, for the Treatment of mTORC1-Activated Tumors
Burnett, G. Leslie, Yang, Yu C., Aggen, James B., Pitzen, Jennifer, Gliedt, Micah K., Semko, Chris M., Marquez, Abby, Evans, James W., Wang, Gang, Won, Walter S., Tomlinson, Aidan C. A., Kiss, Gert, Tzitzilonis, Christos, Thottumkara, Arun P., Cregg, James, Mellem, Kevin T., Choi, Jong S., Lee, Julie C., Zhao, Yongyuan, Lee, Bianca J., Meyerowitz, Justin G., Knox, John E., Jiang, Jingjing, Wang, Zhican, Wildes, David, Wang, Zhengping, Singh, Mallika, Smith, Jacqueline A. M., Gill, Adrian L.
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Parallel Signaling through IRE1α and PERK Regulates Pancreatic Neuroendocrine Tumor Growth and Survival
Moore, Paul C, Qi, Jenny Y, Thamsen, Maike, Ghosh, Rajarshi, Peng, Justin, Gliedt, Micah J, Meza-Acevedo, Rosa, Warren, Rachel E, Hiniker, Annie, Kim, Grace E, Maly, Dustin J, Backes, Bradley J, Papa, Feroz R, Oakes, Scott A
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Structural and Functional Analysis of the Allosteric Inhibition of IRE1α with ATP-Competitive Ligands
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Published in ACS chemical biology (19.08.2016)
Published in ACS chemical biology (19.08.2016)
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Toxicity Modulation, Resistance Enzyme Evasion, and A‑Site X‑ray Structure of Broad-Spectrum Antibacterial Neomycin Analogs
Maianti, Juan Pablo, Kanazawa, Hiroki, Dozzo, Paola, Matias, Rowena D, Feeney, Lee Ann, Armstrong, Eliana S, Hildebrandt, Darin J, Kane, Timothy R, Gliedt, Micah J, Goldblum, Adam A, Linsell, Martin S, Aggen, James B, Kondo, Jiro, Hanessian, Stephen
Published in ACS chemical biology (19.09.2014)
Published in ACS chemical biology (19.09.2014)
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Toward Overcoming Staphylococcus aureus Aminoglycoside Resistance Mechanisms with a Functionally Designed Neomycin Analogue
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Published in ACS medicinal chemistry letters (08.12.2011)
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Abstract 1273: Discovery of a potent, selective, and orally bioavailable SOS1 inhibitor, RMC-023, an in vivo tool compound that blocks RAS activation via disruption of the RAS-SOS1 interaction
Buckl, Andreas, Quintana, Elsa, Lee, Grace J., Shifrin, Nataliya, Zhong, Mengqi, Garrenton, Lindsay S., Montgomery, David C., Stahlhut, Carlos, Zhao, Frances, Whalen, Dan M., Thompson, Severin K., Tambo-ong, Arlyn, Gliedt, Micah, Knox, John E., Cregg, James J., Aay, Naing, Choi, Jong, Nguyen, Bao, Tripathi, Atti, Zhao, Ruiping, Saldajeno-Concar, Mae, Marquez, Abby, Hsieh, Daphne, McDowell, Laura L., Koltun, Elena S., Bermingham, Alun, Wildes, David, Singh, Mallika, Wang, Zhengping, Hansen, Richard, Smith, Jan A., Gill, Adrian L.
Published in Cancer research (Chicago, Ill.) (01.07.2021)
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Abstract PR04: 4EBP1 reactivation by potent and selective bi-steric inhibitors of mTORC1
Tibrewal, Nidhi, Aggen, James B., Bassan, Abraham I., Burnett, G. Leslie, Evans, Jim, Gliedt, Micah J., Hsieh, Daphne, Kiss, Gert, Lee, Bianca J., Lee, Dong, Lorenzana, Ed, Marquez, Abby, Thottumkara, Arun, Wang, Zhengping, Wilson, Stacy, Zhao, Frances, Goldsmith, Mark, Singh, Mallika, Wildes, Pete, Gill, Adrian L., Smith, Jacqueline A.M.
Published in Molecular cancer research (01.10.2020)
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Abstract 2862: The balance of divergent IRE1α signaling regulates pancreatic neuroendocrine tumor growth
Qi, Jenny Y., Moore, Paul C., Thamsen, Maike, Ghosh, Rajarshi, Gliedt, Micah J., Maly, Dustin J., Backes, Bradley J., Papa, Feroz R., Oakes, Scott A.
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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