Virtual discovery of melatonin receptor ligands to modulate circadian rhythms
Stein, Reed M., Kang, Hye Jin, McCorvy, John D., Glatfelter, Grant C., Jones, Anthony J., Che, Tao, Slocum, Samuel, Huang, Xi-Ping, Savych, Olena, Moroz, Yurii S., Stauch, Benjamin, Johansson, Linda C., Cherezov, Vadim, Kenakin, Terry, Irwin, John J., Shoichet, Brian K., Roth, Bryan L., Dubocovich, Margarita L.
Published in Nature (London) (01.03.2020)
Published in Nature (London) (01.03.2020)
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Journal Article
Automated Computer Software Assessment of 5‑Hydroxytryptamine 2A Receptor-Mediated Head Twitch Responses from Video Recordings of Mice
Glatfelter, Grant C., Chojnacki, Michael R., McGriff, Shelby A., Wang, Tianpeng, Baumann, Michael H.
Published in ACS pharmacology & translational science (13.05.2022)
Published in ACS pharmacology & translational science (13.05.2022)
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Journal Article
Pharmacological evaluation and forensic case series of N-pyrrolidino etonitazene (etonitazepyne), a newly emerging 2-benzylbenzimidazole ‘nitazene’ synthetic opioid
Vandeputte, Marthe M., Krotulski, Alex J., Walther, Donna, Glatfelter, Grant C., Papsun, Donna, Walton, Sara E., Logan, Barry K., Baumann, Michael H., Stove, Christophe P.
Published in Archives of toxicology (01.06.2022)
Published in Archives of toxicology (01.06.2022)
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Journal Article
Plasma pharmacokinetics and pharmacodynamic effects of the 2-benzylbenzimidazole synthetic opioid, isotonitazene, in male rats
Walton, Sara E., Krotulski, Alex J., Glatfelter, Grant C., Walther, Donna, Logan, Barry K., Baumann, Michael H.
Published in Psychopharmacology (2023)
Published in Psychopharmacology (2023)
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Journal Article
Reinforcing effects of fentanyl analogs found in illicit drug markets
Maitland, Alexander D, McGriff, Shelby A, Glatfelter, Grant C, Schindler, Charles W, Baumann, Michael H
Published in Psychopharmacology (05.07.2024)
Published in Psychopharmacology (05.07.2024)
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Journal Article
Receptor binding profiles and behavioral effects of psilocybin analogs
Glatfelter, Grant C, Manke, David R, Chadayne, Andrew R, Baumann, Michael H
Published in The FASEB journal (01.05.2022)
Published in The FASEB journal (01.05.2022)
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Journal Article
First identification, chemical analysis and pharmacological characterization of N-piperidinyl etonitazene (etonitazepipne), a recent addition to the 2-benzylbenzimidazole opioid subclass
Vandeputte, Marthe M., Verougstraete, Nick, Walther, Donna, Glatfelter, Grant C., Malfliet, Jeroen, Baumann, Michael H., Verstraete, Alain G., Stove, Christophe P.
Published in Archives of toxicology (01.06.2022)
Published in Archives of toxicology (01.06.2022)
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Journal Article
Comparative neuropharmacology of structurally distinct non-fentanyl opioids that are appearing on recreational drug markets worldwide
Vandeputte, Marthe M., Tsai, Meng-Hua M., Chen, Li, Glatfelter, Grant C., Walther, Donna, Stove, Christophe P., Shi, Lei, Baumann, Michael H.
Published in Drug and alcohol dependence (01.08.2023)
Published in Drug and alcohol dependence (01.08.2023)
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Journal Article
Alkoxy chain length governs the potency of 2-benzylbenzimidazole ‘nitazene’ opioids associated with human overdose
Glatfelter, Grant C., Vandeputte, Marthe M., Chen, Li, Walther, Donna, Tsai, Meng-Hua M., Shi, Lei, Stove, Christophe P., Baumann, Michael H.
Published in Psychopharmacology (01.12.2023)
Published in Psychopharmacology (01.12.2023)
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Journal Article
(2-Aminopropyl)benzo[β]thiophenes (APBTs) are novel monoamine transporter ligands that lack stimulant effects but display psychedelic-like activity in mice
Rudin, Deborah, McCorvy, John D, Glatfelter, Grant C, Luethi, Dino, Szöllősi, Dániel, Ljubišić, Tea, Kavanagh, Pierce V, Dowling, Geraldine, Holy, Marion, Jaentsch, Kathrin, Walther, Donna, Brandt, Simon D, Stockner, Thomas, Baumann, Michael H, Halberstadt, Adam L, Sitte, Harald H
Published in Neuropsychopharmacology (New York, N.Y.) (01.03.2022)
Published in Neuropsychopharmacology (New York, N.Y.) (01.03.2022)
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Journal Article
Unique pharmacodynamic properties and low abuse liability of the µ-opioid receptor ligand (S)-methadone
Levinstein, Marjorie R., De Oliveira, Paulo A., Casajuana-Martin, Nil, Quiroz, Cesar, Budinich, Reece C., Rais, Rana, Rea, William, Ventriglia, Emilya N., Llopart, Natàlia, Casadó-Anguera, Verònica, Moreno, Estefanía, Walther, Donna, Glatfelter, Grant C., Weinshenker, David, Zarate, Carlos A., Casadó, Vicent, Baumann, Michael H., Pardo, Leonardo, Ferré, Sergi, Michaelides, Michael
Published in Molecular psychiatry (01.03.2024)
Published in Molecular psychiatry (01.03.2024)
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Journal Article
Psychedelic-like Activity of Norpsilocin Analogues
Sherwood, Alexander M., Burkhartzmeyer, Elise K., Williamson, Samuel E., Baumann, Michael H., Glatfelter, Grant C.
Published in ACS chemical neuroscience (17.01.2024)
Published in ACS chemical neuroscience (17.01.2024)
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Journal Article
Structure–Activity Relationships for Psilocybin, Baeocystin, Aeruginascin, and Related Analogues to Produce Pharmacological Effects in Mice
Glatfelter, Grant C., Pottie, Eline, Partilla, John S., Sherwood, Alexander M., Kaylo, Kristi, Pham, Duyen N. K., Naeem, Marilyn, Sammeta, Vamshikrishna Reddy, DeBoer, Stacie, Golen, James A., Hulley, Elliott B., Stove, Christophe P., Chadeayne, Andrew R., Manke, David R., Baumann, Michael H.
Published in ACS pharmacology & translational science (11.11.2022)
Published in ACS pharmacology & translational science (11.11.2022)
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Journal Article
Synthesis, Structural Characterization, and Pharmacological Activity of Novel Quaternary Salts of 4‑Substituted Tryptamines
Glatfelter, Grant C., Pham, Duyen N. K., Walther, Donna, Golen, James A., Chadeayne, Andrew R., Baumann, Michael H., Manke, David R.
Published in ACS omega (19.07.2022)
Published in ACS omega (19.07.2022)
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