Discovery of Potent and Selective Dipeptidyl Peptidase IV Inhibitors Derived from [beta]-Aminoamides Bearing Subsituted Triazolopiperazines
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Published in Journal of medicinal chemistry (30.06.2008)
Published in Journal of medicinal chemistry (30.06.2008)
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Crystals of anti-human PD-1 monoclonal antibodies
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Year of Publication 01.08.2024
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Year of Publication 01.08.2024
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Discovery of Potent and Selective Dipeptidyl Peptidase IV Inhibitors Derived from β-Aminoaimdes Bearing Subsituted Triazolopiperazines
KIM, Dooseop, KOWALCHICK, Jennifer E, PATEL, Sangita B, PETROV, Aleksandr, PRYOR, Kellyann D, ROY, Ranabir Sinha, WU, Joseph K, XIAOPING ZHANG, WYVRATT, Matthew J, ZHANG, Bei B, LAN ZHU, THOMBERRY, Nancy A, BROCKUNIER, Linda L, WEBER, Ann E, PARMEE, Emma R, EIERMANN, George J, FISHER, Michael H, HUAIBING HE, LEITING, Barbara, LYONS, Kathryn, SCAPIN, Giovanna
Published in Journal of medicinal chemistry (2008)
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Published in Journal of medicinal chemistry (2008)
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Hybrid-Designed Inhibitors of p38 MAP Kinase Utilizing N-Arylpyridazinones
Colletti, Steven L, Frie, Jessica L, Dixon, Elizabeth C, Singh, Suresh B, Choi, Bernard K, Scapin, Giovanna, Fitzgerald, Catherine E, Kumar, Sanjeev, Nichols, Elizabeth A, O'Keefe, Stephen J, O'Neill, Edward A, Porter, Gene, Samuel, Koppara, Schmatz, Dennis M, Schwartz, Cheryl D, Shoop, Wesley L, Thompson, Chris M, Thompson, James E, Wang, Ruixiu, Woods, Andrea, Zaller, Dennis M, Doherty, James B
Published in Journal of medicinal chemistry (30.01.2003)
Published in Journal of medicinal chemistry (30.01.2003)
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Novel tetrahydropyran analogs as dipeptidyl peptidase IV inhibitors: Profile of clinical candidate (2R,3S,5R)-2- (2,5-difluorophenyl)-5-(4,6-dihydropyrrolo [3,4-c]pyrazol-5-(1H)-yl)tetrahydro-2H-pyran-3-amine (23) [corrected]
Biftu, Tesfaye, Qian, Xiaoxia, Chen, Ping, Feng, Dennis, Scapin, Giovanna, Gao, Ying-Duo, Cox, Jason, Roy, Ranabir Sinha, Eiermann, George, He, Huabing, Lyons, Kathy, Salituro, Gino, Patel, Sangita, Petrov, Alexander, Xu, Feng, Xu, Shiyao Sherrie, Zhang, Bei, Caldwell, Charles, Wu, Joseph K, Weber, Ann E
Published in Bioorganic & medicinal chemistry letters (01.10.2013)
Published in Bioorganic & medicinal chemistry letters (01.10.2013)
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Design, synthesis, and biological evaluation of triazolopiperazine-based SS-amino amides as potent, orally active dipeptidyl peptidase IV (DPP-4) inhibitors
KOWALCHICK, Jennifer E, LEITING, Barbara, PATEL, Reshma A, THORNBERRY, Nancy A, WEBER, Ann E, KIM, Dooseop, PRYOR, Kellyann D, MARSILIO, Frank, WU, Joseph K, HUAIBING HE, LYONS, Kathryn A, EIERMANN, George J, PETROV, Aleksandr, SCAPIN, Giovanna
Published in Bioorganic & medicinal chemistry letters (2007)
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Published in Bioorganic & medicinal chemistry letters (2007)
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'es_ES': 'CONSUMO DE ALCOHOL Y DESEMPEÑO ACADÉMICO DE ESTUDIANTES DE LOS PRIMEROS AÑOS DE ENFERMERÍA', 'pt_BR': 'CONSUMO DE ÁLCOOL E DESEMPENHO ACADÊMICO DE ALUNOS DOS ANOS INICIAIS DA GRADUAÇÃO EM ENFERMAGEM'
Giovanna Cardoso Scapin, Jamila Souza Gonçalves, Fabio Scorsolini-Comin, Janaína Cristina Pasquini de Almeida, Jaqueline Lemos de Oliveira, Jacqueline de Souza
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Published in REME (01.09.2021)
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The three-dimensional structure of MAP kinase p38[beta]: different features of the ATP-binding site in p38[beta] compared with p38[alpha]
Patel, Sangita B., Cameron, Patricia M., O'Keefe, Stephen J., Frantz-Wattley, Betsy, Thompson, Jed, O'Neill, Edward A., Tennis, Trevor, Liu, Luping, Becker, Joseph W., Scapin, Giovanna, Merck
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Published in Acta crystallographica. Section D, Biological crystallography. (18.10.2010)
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Three-dimensional structure of recombinant human muscle fatty acid-binding protein
ZANOTTI, G, SCAPIN, G, SPADON, P, VEERKAMP, J. H, SACCHETTINI, J. C
Published in The Journal of biological chemistry (15.09.1992)
Published in The Journal of biological chemistry (15.09.1992)
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Refinement of the structure of recombinant rat intestinal fatty acid-binding apoprotein at 1.2-A resolution
SCAPIN, G, GORDON, J. I, SACCHETTIN, J. C
Published in The Journal of biological chemistry (25.02.1992)
Published in The Journal of biological chemistry (25.02.1992)
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Structural studies on human muscle fatty acid binding protein at 1.4 å resolution: binding interactions with three C18 fatty acids
Young, Aideen CM, Scapin, Giovanna, Kromminga, Arno, Patel, Sangita B, Veerkamp, Jacques H, Sacchettini, James C
Published in Structure (London) (15.06.1994)
Published in Structure (London) (15.06.1994)
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ARGINASE 1 BINDERS FOR INHIBITING ARGINASE 1 ACTIVITY
Chakravarthy, Kalyan, Taremi, Shahriar Shane, Scapin, Giovanna, Fayad, Ghassan Najib, Bailly, Marc Andre, Fayadat-Dilman, Laurence, Kofman, Esther, O'Neil, Jennifer E, Palte, Rachel Lynn, Handa, Masahisa
Year of Publication 04.01.2024
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Year of Publication 04.01.2024
Patent
ARGINASE 1 BINDERS FOR INHIBITING ARGINASE 1 ACTIVITY
Chakravarthy, Kalyan, Taremi, Shahriar Shane, Scapin, Giovanna, Fayad, Ghassan Najib, Bailly, Marc Andre, Fayadat-Dilman, Laurence, Kofman, Esther, O'Neil, Jennifer E, Palte, Rachel Lynn, Juan, Veronica, Handa, Masahisa
Year of Publication 04.01.2024
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Year of Publication 04.01.2024
Patent
Crystals of anti-human PD-1 monoclonal antibodies
KASHI, Ramesh, STRICKLAND, Corey, PROSISE, Winifred W, REICHERT, Paul, YANG, Xiaoyu, SCAPIN, Giovanna
Year of Publication 10.02.2022
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Year of Publication 10.02.2022
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Structural basis for p38[alpha] MAP kinase quinazolinone and pyridol-pyrimidine inhibitor specificity
Fitzgerald, Catherine E, Patel, Sangita B, Becker, Joseph W, Cameron, Patricia M, Zaller, Dennis, Pikounis, Vasilis Bill, O'Keefe, Stephen J, Scapin, Giovanna
Published in Nature structural & molecular biology (01.09.2003)
Published in Nature structural & molecular biology (01.09.2003)
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ARGINASE 1 BINDERS FOR INHIBITING ARGINASE 1 ACTIVITY
FAYADAT-DILMAN, Laurence, BAILLY, Marc Andre, CHAKRAVARTHY, Kalyan, KOFMAN, Esther, O'NEIL, Jennifer, E, FAYAD, Ghassan Najib, SCAPIN, Giovanna, JUAN, Veronica, HANDA, Masahisa, PALTE, Rachel Lynn, TAREMI, Shahriar Shane
Year of Publication 04.10.2023
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Year of Publication 04.10.2023
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