High-Resolution Cryo-Electron Microscopy Structure Determination of IHaemophilus influenzae/I Tellurite-Resistance Protein A via 200 kV Transmission Electron Microscopy
Tran, Nhi L, Senko, Skerdi, Lucier, Kyle W, Farwell, Ashlyn C, Silva, Sabrina M, Dip, Phat V, Poweleit, Nicole, Scapin, Giovanna, Catalano, Claudio
Published in International journal of molecular sciences (01.04.2024)
Published in International journal of molecular sciences (01.04.2024)
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Serendipitous discovery of aryl boronic acids as β-lactamase inhibitors
Yang, Shu-Wei, Pan, Jianping, Root, Yuriko, Scapin, Giovanna, Xiao, Li, Su, Jing
Published in Bioorganic & medicinal chemistry letters (15.01.2020)
Published in Bioorganic & medicinal chemistry letters (15.01.2020)
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Discovery of MK-7655, a β-lactamase inhibitor for combination with Primaxin
Blizzard, Timothy A., Chen, Helen, Kim, Seongkon, Wu, Jane, Bodner, Rena, Gude, Candido, Imbriglio, Jason, Young, Katherine, Park, Young-Whan, Ogawa, Aimie, Raghoobar, Susan, Hairston, Nichelle, Painter, Ronald E., Wisniewski, Doug, Scapin, Giovanna, Fitzgerald, Paula, Sharma, Nandini, Lu, Jun, Ha, Sookhee, Hermes, Jeff, Hammond, Milton L.
Published in Bioorganic & medicinal chemistry letters (01.02.2014)
Published in Bioorganic & medicinal chemistry letters (01.02.2014)
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The CryoEM structure of human serum albumin in complex with ligands
Catalano, Claudio, Lucier, Kyle W., To, Dennis, Senko, Skerdi, Tran, Nhi L., Farwell, Ashlyn C., Silva, Sabrina M., Dip, Phat V., Poweleit, Nicole, Scapin, Giovanna
Published in Journal of structural biology (01.09.2024)
Published in Journal of structural biology (01.09.2024)
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Discovery of MK-4688: an Efficient Inhibitor of the HDM2–p53 Protein–Protein Interaction
Reutershan, Michael H, Machacek, Michelle R, Altman, Michael D, Bogen, Stephane, Cai, Mingmei, Cammarano, Carolyn, Chen, Dapeng, Christopher, Matthew, Cryan, John, Daublain, Pierre, Fradera, Xavier, Geda, Prasanthi, Goldenblatt, Peter, Hill, Armetta D, Kemper, Raymond A, Kutilek, Victoria, Li, Chaomin, Martinez, Michelle, McCoy, Mark, Nair, Latha, Pan, Weidong, Thompson, Christopher F, Scapin, Giovanna, Shizuka, Manami, Spatz, Marianne L, Steinhuebel, Dietrich, Sun, Binyuan, Voss, Matthew E, Wang, Xiao, Yang, Liping, Yeh, Tammie C, Dussault, Isabelle, Marshall, C. Gary, Trotter, B. Wesley
Published in Journal of medicinal chemistry (11.11.2021)
Published in Journal of medicinal chemistry (11.11.2021)
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Small-molecule microcrystal electron diffraction (MicroED) for the pharmaceutical industry
Bruhn, Jessica, Cheng, Anchi, Nieusma, Travis, Dallakyan, Sargis, Speir, Jeff, Schneemann, Anette, Potter, Clint, Carragher, Bridget, Scapin, Giovanna
Published in Acta crystallographica. Section A, Foundations and advances (02.08.2020)
Published in Acta crystallographica. Section A, Foundations and advances (02.08.2020)
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Small-molecule microcrystal electron diffraction (MicroED) for the pharmaceutical industry – lessons learned from examining over fifty samples
Bruhn, Jessica, Scapin, Giovanna, Cheng, Anchi, Mercado, Brandon, Waterman, David, Ganesh, Thejusvi, Dallakyan, Sargis, Read, Brandon, Nieusma, Travis, Lucier, Kyle, Mayer, Megan, Chiang, Nicole, Poweleit, Nicole
Published in Acta crystallographica. Section A, Foundations and advances (30.07.2021)
Published in Acta crystallographica. Section A, Foundations and advances (30.07.2021)
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Structure Guided Discovery of Novel Pan Metallo-β-Lactamase Inhibitors with Improved Gram-Negative Bacterial Cell Penetration
Dong, Shuzhi, Zhao, Zhiqiang, Tang, Haiqun, Li, Guoqing, Pan, Jianping, Gu, Xin, Jiang, Jinlong, Xiao, Li, Scapin, Giovanna, Hunter, David N., Yang, Dexi, Huang, Yuhua, Bennett, Frank, Yang, Shu-Wei, Mandal, Mihirbaran, Tang, Haifeng, Su, Jing, Tudge, Clare, deJesus, Reynalda Keh, Ding, Fa-Xiang, Lombardo, Matthew, Hicks, Jacqueline D., Fischmann, Thierry, Mirza, Asra, Dayananth, Priya, Painter, Ronald E., Villafania, Artjohn, Garlisi, Charles G., Zhang, Rumin, Mayhood, Todd W., Si, Qian, Li, Nianyu, Amin, Rupesh P., Bhatt, Bhavana, Chen, Feifei, Regan, Christopher P., Regan, Hillary, Lin, Xinjie, Wu, Jin, Leithead, Andrew, Pollack, Scott R., Scott, Jack D., Nargund, Ravi P., Therien, Alex G., Black, Todd, Young, Katherine, Pasternak, Alexander
Published in Journal of medicinal chemistry (14.03.2024)
Published in Journal of medicinal chemistry (14.03.2024)
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A novel storage system for cryoEM samples
Scapin, Giovanna, Prosise, Winifred W., Wismer, Michael K., Strickland, Corey
Published in Journal of structural biology (01.07.2017)
Published in Journal of structural biology (01.07.2017)
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Rapid Evolution of a Fragment-like Molecule to Pan-Metallo-Beta-Lactamase Inhibitors: Initial Leads toward Clinical Candidates
Mandal, Mihirbaran, Xiao, Li, Pan, Weidong, Scapin, Giovanna, Li, Guoqing, Tang, Haiqun, Yang, Shu-Wei, Pan, Jianping, Root, Yuriko, de Jesus, Reynalda Keh, Yang, Christine, Prosise, Winnie, Dayananth, Priya, Mirza, Asra, Therien, Alex G., Young, Katherine, Flattery, Amy, Garlisi, Charles, Zhang, Rumin, Chu, Donald, Sheth, Payal, Chu, Inhou, Wu, Jin, Markgraf, Carrie, Kim, Hai-Young, Painter, Ronald, Mayhood, Todd W., DiNunzio, Edward, Wyss, Daniel F., Buevich, Alexei V., Fischmann, Thierry, Pasternak, Alexander, Dong, Shuzhi, Hicks, Jacqueline D., Villafania, Artjohn, Liang, Lianzhu, Murgolo, Nicholas, Black, Todd, Hagmann, William K., Tata, Jim, Parmee, Emma R., Weber, Ann E., Su, Jing, Tang, Haifeng
Published in Journal of medicinal chemistry (22.12.2022)
Published in Journal of medicinal chemistry (22.12.2022)
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Cerastecin Inhibition of the Lipooligosaccharide Transporter MsbA to Combat Acinetobacter baumannii : From Screening Impurity to In Vivo Efficacy
Skudlarek, Jason W, Cooke, Andrew J, Mitchell, Helen J, Babaoglu, Kerim, Shaw, Anthony W, Tong, Ling, Nomland, Ashley B, Labroli, Marc, Sha, Deyou, Mulhearn, James J, Wu, Chengwei, Li, Sarah W, Beshore, Douglas C, Hughes, Jonathan M E, Jouffroy, Matthieu, Wang, Hao, Balibar, Carl J, Painter, Ronald E, Shen, Pamela, Lange, Henry S, Ishchenko, Andrii, Chen, Yun-Ting, Klein, Daniel J, Tracy, Rodger W, Miller, Randy R, Cabalu, Tamara D, Wu, Zhe, Leithead, Andrew, Scapin, Giovanna, Hruza, Alan W, Dzhekieva, Liudmila, Bukhtiyarova, Marina, Homsher, Michelle F, Xu, Min, Bahnck-Teets, Carolyn, McKenney, David, Buevich, Alexei V, Liu, Jian, Zhang, Li-Kang, Meng, Tao, Kelly, Terri, DiNunzio, Edward, Soisson, Stephen, Cheng, Robert K Y, Hennig, Michael, Raheem, Izzat, Walker, Scott S
Published in Journal of medicinal chemistry (12.09.2024)
Published in Journal of medicinal chemistry (12.09.2024)
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Structure of the insulin receptorinsulin complex by single-particle cryo-EM analysis
Scapin, Giovanna, Dandey, Venkata P, Zhang, Zhening, Prosise, Winifred, Hruza, Alan, Kelly, Theresa, Mayhood, Todd, Strickland, Corey, Potter, Clinton S, Carragher, Bridget
Published in Nature (London) (05.04.2018)
Published in Nature (London) (05.04.2018)
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Journal Article
Structure of the Insulin Receptor-Insulin Complex by Single Particle CryoEM analysis
Scapin, Giovanna, Dandey, Venkata P., Zhang, Zhening, Prosise, Winifred, Hruza, Alan, Kelly, Theresa, Mayhood, Todd, Strickland, Corey, Potter, Clinton S., Carragher, Bridget
Published in Nature (London) (28.02.2018)
Published in Nature (London) (28.02.2018)
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For the record: The three‐dimensional structure of the ternary complex of Corynebacterium glutamicum diaminopimelate dehydrogenase‐NADPH‐L‐2‐amino‐6‐methylene‐pimelate
Cirilli, Maurizio, Scapin, Giovanna, Sutherland, Andrew, Vederas, John C., Blanchard, John S.
Published in Protein science (2000)
Published in Protein science (2000)
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Cryo-EM structures of inhibitory antibodies complexed with Arginase1 provide insight into mechanism of action
Palte, Rachel, Juan, Veronica, Gomez-Llorente, Yacob, Scapin, Giovanna, Bailly, Marc, Fayadat-Dilman, Laurence, Gathiaka, Symon, Hall, Brian, Handa, Mas, Kofman, Esther, Hsieh, Mark, Miller, J. Richard, Taremi, Shane
Published in Acta crystallographica. Section A, Foundations and advances (30.07.2021)
Published in Acta crystallographica. Section A, Foundations and advances (30.07.2021)
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Structure and Function of Salmonella typhimurium Orotate Phosphoribosyltransferase: Protein Complementation Reveals Shared Active Sites
Ozturk, Derya H, Dorfman, Ryan H, Scapin, Giovanna, Sacchettini, James C, Grubmeyer, Charles
Published in Biochemistry (Easton) (29.08.1995)
Published in Biochemistry (Easton) (29.08.1995)
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Cryoet of Single Particle CryoEM Grids Reveals Widespread, but Reducible, Particle Adsorption to the Air-Water Interface
Noble, Alex J., Dandey, Venkata P., Wei, Hui, Brasch, Julia, Chase, Jillian, Acharya, Priyamvada, Zi Tan, Yong, Zhang, Zhening, Kim, Laura Y., Scapin, Giovanna, Rapp, Micah, Eng, Edward T., Rice, William J., Cheng, Anchi, Negro, Carl J.
Published in Biophysical journal (01.02.2019)
Published in Biophysical journal (01.02.2019)
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