Crystal structure and functional domains of the Mambaquaretin-1, a vasopressin type 2 receptor peptide inhibitor for kidney cysts treatment
Droctové, Laura, Ciolek, Justyna, Lancien, Manon, Stura, Enrico A., Vera, Laura, Floquet, Nicolas, Witzgall, Ralph, Mouillac, Bernard, Mendre, Christiane, Mourier, Gilles, Servent, Denis, Gilles, Nicolas
Published in Toxicon (Oxford) (01.07.2018)
Published in Toxicon (Oxford) (01.07.2018)
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Journal Article
Discovery and characterization of EII B, a new α-conotoxin from Conus ermineus venom by nAChRs affinity capture monitored by MALDI-TOF/TOF mass spectrometry
Echterbille, Julien, Gilles, Nicolas, Araóz, Romulo, Mourier, Gilles, Amar, Muriel, Servent, Denis, De Pauw, Edwin, Quinton, Loic
Published in Toxicon (Oxford) (01.05.2017)
Published in Toxicon (Oxford) (01.05.2017)
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Journal Article
New α-adrenergic property for synthetic MTβ and CM-3 three-finger fold toxins from black mamba
Blanchet, Guillaume, Upert, Gregory, Mourier, Gilles, Gilquin, Bernard, Gilles, Nicolas, Servent, Denis
Published in Toxicon (Oxford) (01.12.2013)
Published in Toxicon (Oxford) (01.12.2013)
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Journal Article
Ion Mobility-Mass Spectrometry as a Tool for the Structural Characterization of Peptides Bearing Intramolecular Disulfide Bond(s)
Massonnet, Philippe, Haler, Jean R. N., Upert, Gregory, Degueldre, Michel, Morsa, Denis, Smargiasso, Nicolas, Mourier, Gilles, Gilles, Nicolas, Quinton, Loïc, De Pauw, Edwin
Published in Journal of the American Society for Mass Spectrometry (01.10.2016)
Published in Journal of the American Society for Mass Spectrometry (01.10.2016)
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Structural model of ligand-G protein-coupled receptor (GPCR) complex based on experimental double mutant cycle data: MT7 snake toxin bound to dimeric hM1 muscarinic receptor
Marquer, Catherine, Fruchart-Gaillard, Carole, Letellier, Guillaume, Marcon, Elodie, Mourier, Gilles, Zinn-Justin, Sophie, Ménez, André, Servent, Denis, Gilquin, Bernard
Published in The Journal of biological chemistry (09.09.2011)
Published in The Journal of biological chemistry (09.09.2011)
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Journal Article
Natural agents targeting the α7‐nicotinic‐receptor in NSCLC: A promising prospective in anti‐cancer drug development
Grozio, Alessia, Paleari, Laura, Catassi, Alessia, Servent, Denis, Cilli, Michele, Piccardi, Federica, Paganuzzi, Michela, Cesario, Alfredo, Granone, Pierluigi, Mourier, Gilles, Russo, Patrizia
Published in International journal of cancer (15.04.2008)
Published in International journal of cancer (15.04.2008)
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Journal Article
High-throughput production of two disulphide-bridge toxinsElectronic supplementary information (ESI) available. See DOI: 10.1039/c4cc02679a
Upert, Grégory, Mourier, Gilles, Pastor, Alexandra, Verdenaud, Marion, Alili, Doria, Servent, Denis, Gilles, Nicolas
Year of Publication 03.07.2014
Year of Publication 03.07.2014
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Journal Article
Natural agents targeting the alpha 7-nicotinic-receptor in NSCLC: A promising prospective in anti-cancer drug development
Grozio, Alessia, Paleari, Laura, Catassi, Alessia, Servent, Denis, Cilli, Michele, Piccardi, Federica, Paganuzzi, Michela, Cesario, Alfredo, Granone, Pierluigi, Mourier, Gilles, Russo, Patrizia
Published in International journal of cancer (15.04.2008)
Published in International journal of cancer (15.04.2008)
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Journal Article
Mambalgins, snake peptides against inflammatory and neuropathic pain through inhibition of ASIC channels
Baron, Anne, Diochot, Sylvie, Salinas, Miguel, Alloui, Abdelkrim, Douguet, Dominique, Mourier, Gilles, Kessler, Pascal, Stura, Enrico A., Besson, Thomas, Friend, Valérie, Servent, Denis, Eschalier, Alain, Lingueglia, Eric
Published in Toxicon (Oxford) (01.07.2018)
Published in Toxicon (Oxford) (01.07.2018)
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Journal Article
A snake toxin as a theranostic agent for the type 2 vasopressin receptor
Droctové, Laura, Lancien, Manon, Tran, Vu Long, Susset, Michaël, Jego, Benoit, Theodoro, Frederic, Kessler, Pascal, Mourier, Gilles, Robin, Philippe, Diarra, Sékou Siramakan, Palea, Stefano, Flahault, Adrien, Chorfa, Amélia, Corbani, Maithé, Llorens-Cortes, Catherine, Mouillac, Bernard, Mendre, Christiane, Pruvost, Alain, Servent, Denis, Truillet, Charles, Gilles, Nicolas
Published in Theranostics (01.01.2020)
Published in Theranostics (01.01.2020)
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Journal Article
A snake toxin as a theranostic agent for the type 2 vasopressin receptor
Droctové, Laura, Lancien, Manon, Tran, Vu Long, Susset, Michaël, Jego, Benoit, Theodoro, Frederic, Kessler, Pascal, Mourier, Gilles, Robin, Philippe, Diarra, Sékou Siramakan, Palea, Stefano, Flahault, Adrien, Chorfa, Amélia, Corbani, Maithé, Llorens-Cortes, Catherine, Mouillac, Bernard, Mendre, Christiane, Pruvost, Alain, Servent, Denis, Truillet, Charles, Gilles, Nicolas
Published in Theranostics (18.09.2020)
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Published in Theranostics (18.09.2020)
Journal Article
Green mamba peptide targets type-2 vasopressin receptor against polycystic kidney disease
Ciolek, Justyna, Reinfrank, Helen, Quinton, Loïc, Viengchareun, Say, Stura, Enrico, Vera, Laura, Sigismeau, Sabrina, Mouillac, Bernard, Orcel, Hélène, Peigneur, Steve, Tytgat, Jan, Droctové, Laura, Beau, Fabrice, Nevoux, Jerome, Lombès, Marc, Mourier, Gilles, de Pauw, Edwin, Servent, Denis, Mendre, Christiane, Witzgall, Ralph, Gilles, Nicolas
Published in Proceedings of the National Academy of Sciences - PNAS (19.06.2017)
Published in Proceedings of the National Academy of Sciences - PNAS (19.06.2017)
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Journal Article
Identification of a novel snake peptide toxin displaying high affinity and antagonist behaviour for the α 2 ‐adrenoceptors
Rouget, Céline, Quinton, Loïc, Maïga, Arhamatoulaye, Gales, Céline, Masuyer, Geoffrey, Malosse, Christian, Chamot‐Rooke, Julia, Thai, Robert, Mourier, Gilles, De Pauw, Edwin, Gilles, Nicolas, Servent, Denis
Published in British journal of pharmacology (01.11.2010)
Published in British journal of pharmacology (01.11.2010)
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Journal Article
Identification of a novel snake peptide toxin displaying high affinity and antagonist behaviour for the α(2) -adrenoceptors
Rouget, Céline, Quinton, Loïc, Maïga, Arhamatoulaye, Gales, Céline, Masuyer, Geoffrey, Malosse, Christian, Chamot-Rooke, Julia, Thai, Robert, Mourier, Gilles, de Pauw, Edwin, Gilles, Nicolas, Servent, Denis
Published in British journal of pharmacology (01.11.2010)
Published in British journal of pharmacology (01.11.2010)
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Journal Article
Echocardiographic Evaluation of the Acute Cardiovascular Effects of an Endothelin-Like Peptide Extracted from the Venom of Atractaspis irregularis
Mahjoub, Yazine, Malaquin, Stéphanie, Abou Arab, Osama, Mourier, Gilles, Lorne, Emmanuel, Salomon, Alexis, Kamel, Saïd, Dupont, Hervé, Ducancel, Frédéric
Published in Cardiovascular toxicology (01.04.2017)
Published in Cardiovascular toxicology (01.04.2017)
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Journal Article
Pharmacological and structural characterization of long-sarafotoxins, a new family of endothelin-like peptides: Role of the C-terminus extension
Mourier, Gilles, Hajj, Mariana, Cordier, Florence, Zorba, Adelajda, Gao, XingHuang, Coskun, Tolga, Herbet, Amaury, Marcon, Elodie, Beau, Fabrice, Delepierre, Muriel, Ducancel, Frédéric, Servent, Denis
Published in Biochimie (01.02.2012)
Published in Biochimie (01.02.2012)
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Journal Article
G protein-coupled receptors, an unexploited animal toxin targets: Exploration of green mamba venom for novel drug candidates active against adrenoceptors
Maïga, Arhamatoulaye, Mourier, Gilles, Quinton, Loïc, Rouget, Céline, Gales, Céline, Denis, Colette, Lluel, Philippe, Sénard, Jean-Michel, Palea, Stefano, Servent, Denis, Gilles, Nicolas
Published in Toxicon (Oxford) (15.03.2012)
Published in Toxicon (Oxford) (15.03.2012)
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Different Interactions between MT7 Toxin and the Human Muscarinic M 1 Receptor in Its Free and N -Methylscopolamine-Occupied States
Fruchart-Gaillard, Carole, Mourier, Gilles, Marquer, Catherine, Stura, Enrico, Birdsall, Nigel J. M., Servent, Denis
Published in Molecular pharmacology (01.12.2008)
Published in Molecular pharmacology (01.12.2008)
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Journal Article
Isolation and pharmacological characterization of AdTx1, a natural peptide displaying specific insurmountable antagonism of the alpha(1A)-adrenoceptor
Quinton, L., Girard, Emmanuelle, Maiga, A., Rekik, M., Lluel, P., Masuyer, G., Larregola, M., Marquer, C., Ciolek, J., Magnin, T., Wagner, R., Molgó, Jordi, Thai, Robert, Fruchart-Gaillard, C., Mourier, Gilles, Chamot-Rooke, J., Ménez, André, Palea, S., Servent, Denis, Gilles, Nicolas
Published in British journal of pharmacology (01.01.2010)
Published in British journal of pharmacology (01.01.2010)
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Journal Article
140. Identification, Pharmacological and Structural characterization and Engineering of Three-finger Toxins interacting with GPCRs
Blanchet, Guillaume, Mourier, Gilles, Marcon, Elodie, Gilquin, Bernard, Gilles, Nicolas, Servent, Denis
Published in Toxicon (Oxford) (01.08.2012)
Published in Toxicon (Oxford) (01.08.2012)
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