Discovery of a novel series of selective MMP inhibitors: Identification of the γ-sulfone-thiols
Freskos, John N., Mischke, Brent V., DeCrescenzo, Gary A., Heintz, Robert, Getman, Daniel P., Howard, Susan C., Kishore, Nandini N., McDonald, Joseph J., Munie, Grace E., Rangwala, Shaukat, Swearingen, Craig A., Voliva, Charles, Welsch, Dean J.
Published in Bioorganic & medicinal chemistry letters (05.04.1999)
Published in Bioorganic & medicinal chemistry letters (05.04.1999)
Get full text
Journal Article
Kinetic and structural evidence for a sequential ordered Bi Bi mechanism of catalysis by Saccharomyces cerevisiae myristoyl-CoA:protein N-myristoyltransferase
RUDNICK, D. A, MCWHERTER, C. A, ROCQUE, W. J, LENNON, P. J, GETMAN, D. P, GORDON, J. I
Published in The Journal of biological chemistry (25.05.1991)
Published in The Journal of biological chemistry (25.05.1991)
Get full text
Journal Article
Scanning alanine mutagenesis and de-peptidization of a Candida albicans myristoyl-CoA:protein N-myristoyltransferase octapeptide substrate reveals three elements critical for molecular recognition
McWherter, C A, Rocque, W J, Zupec, M E, Freeman, S K, Brown, D L, Devadas, B, Getman, D P, Sikorski, J A, Gordon, J I
Published in The Journal of biological chemistry (02.05.1997)
Published in The Journal of biological chemistry (02.05.1997)
Get full text
Journal Article
Structural determinants of haloenol lactone-mediated suicide inhibition of canine myocardial calcium-independent phospholipase A2
Zupan, Lori A., Weiss, Randy H., Hazen, Stanley L., Parnas, Barry L., Aston, Karl W., Lennon, Patrick J., Getman, Daniel P., Gross, Richard W.
Published in Journal of medicinal chemistry (1993)
Published in Journal of medicinal chemistry (1993)
Get full text
Journal Article
A CONVENIENT ASYMMETRIC-SYNTHESIS OF THE UNNATURAL AMINO-ACID 2,6-DIMETHYL-L-TYROSINE
DYGOS, JH, YONAN, EE, SCAROS, MG, GOODMONSON, OJ, GETMAN, DP, PERIANA, RA, BECK, GR
Published in Synthesis (Stuttgart) (1992)
Published in Synthesis (Stuttgart) (1992)
Get more information
Journal Article
Inhibitors of HIV-1 Protease Containing the Novel and Potent (R)-(Hydroxyethyl)sulfonamide Isostere
Vazquez, Michael L, Bryant, Martin L, Clare, Michael, DeCrescenzo, Gary A, Doherty, Elizabeth M, Freskos, John N, Getman, Daniel P, Houseman, Kathryn A, Julien, Janet A, Kocan, Geralyn P, Mueller, Richard A, Shieh, Huey-Sheng, Stallings, William C, Stegeman, Roderick A, Tilley, John J
Published in Journal of medicinal chemistry (01.02.1995)
Published in Journal of medicinal chemistry (01.02.1995)
Get full text
Journal Article
Replacements for lysine in l-seryl- l-lysyl dipeptide amide inhibitors of candida albicans myristoyl-CoA:protein N-myristoyltransferase
Brown, David L., Devadas, Balekudru, Lu, Hwang-Fun, Nagarajan, Srinivasan, Zupec, Mark E., Freeman, Sandra K., McWherter, Charles A., Getman, Daniel P., Sikorski, James A.
Published in Bioorganic & medicinal chemistry letters (04.02.1997)
Published in Bioorganic & medicinal chemistry letters (04.02.1997)
Get full text
Journal Article
(Hydroxyethyl) sulfonamide HIV-1 Protease inhibitors: Identification of the 2-methylbenzoyl moiety at P-2
Freskos, John N., Bertenshaw, Deborah E., Getman, Daniel P., Heintz, Robert M., Mischke, Brent V., Blystone, Lisa W., Bryant, Martin L., Funckes-Shippy, Christine, Houseman, Kathyrn A., Kishore, Nandini N., Kocan, Geralyn P., Mehta, Pramod P.
Published in Bioorganic & medicinal chemistry letters (20.02.1996)
Published in Bioorganic & medicinal chemistry letters (20.02.1996)
Get full text
Journal Article
BROADSPECTRUM 2-AMINO-BENZOTHIAZOLE SULFONAMIDE HIV PROTEASE INHIBITORS
GETMAN, DANIEL P, SURLERAUX, DOMINIQUE LOUIS NESTOR GHISLAIN, WIGERINCK, PIET TOM BERT PAUL
Year of Publication 22.05.2012
Get full text
Year of Publication 22.05.2012
Patent