Search Results - "GENEVOIS-BORELLA, Arielle" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Synthesis and pharmacological properties of 5H,10H-imidazo[1,2-a]indeno[1,2-e]pyrazine-4-one, a new competitive AMPA/KA receptor antagonist

Synthesis and pharmacological properties of 5H,10H-imidazo[1,2-a]indeno[1,2-e]pyrazine-4-one, a new competitive AMPA/KA receptor antagonist

by Mignani, Serge, Aloup, Jean-Claude, Barreau, Michel, Blanchard, Jean Charles, Böhme, Georg Andrees, Boireau, Alain, Damour, Dominique, Debono, Marc-Williams, Dubroeucq, Marie-Christine, Genevois-Borella, Arielle, Imperato, Assunta, Jimonet, Patrick, Pratt, Jeremy, Randle, John C.R., Reibaud, Michel, Ribeill, Yves, Stutzmann, Jean-Marie
Published in Drug development research (01.11.1999)

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Journal Article

In vitro and in vivo characterization of TC-1827, a novel brain α4β2 nicotinic receptor agonist with pro-cognitive activity

In vitro and in vivo characterization of TC-1827, a novel brain α4β2 nicotinic receptor agonist with pro-cognitive activity

by Bohme, Georg Andrees, Letchworth, Sharon R., Piot-Grosjean, Odile, Gatto, Gregory J., Obinu, Marie-Carmen, Caldwell, William S., Laville, Michel, Brunel, Pascale, Pellerin, Rachel, Leconte, Jean-Pierre, Genevois-Borella, Arielle, Dubedat, Pierre, Mazadier, Martine, Pradier, Laurent, Bencherif, Merouane, Benavides, Jesus
Published in Drug development research (01.05.2004)

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Journal Article

A preparative route to fused 4-hydroxy-3-phenylindeno(benzothieno)pyridin-2-ones

A preparative route to fused 4-hydroxy-3-phenylindeno(benzothieno)pyridin-2-ones

by Genevois-Borella, A, Vuilhorgne, M, Mignani, S
Published in Heterocycles (01.02.2002)

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Journal Article

DERIVATIVES OF 1-OXO-1,2-DIHYDROISOQUINOLINE-5-CARBOXAMIDES AND OF 4-OXO-3,4-DIHYDROQUINAZOLINE-8-CARBOXAMIDES, PREPARATION THEREOF AND APPLICATION THEREOF IN THERAPEUTICS

DERIVATIVES OF 1-OXO-1,2-DIHYDROISOQUINOLINE-5-CARBOXAMIDES AND OF 4-OXO-3,4-DIHYDROQUINAZOLINE-8-CARBOXAMIDES, PREPARATION THEREOF AND APPLICATION THEREOF IN THERAPEUTICS

by GENEVOIS BORELLA ARIELLE, MALLERON JEAN LUC, EVERS MICHEL, KARLSSON ANDREAS
Year of Publication 07.05.2010

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Patent

ARYLVINYLAZACYCLOALKANE COMPOUNDS AND METHODS OF PREPARATION AND USE THEREOF

ARYLVINYLAZACYCLOALKANE COMPOUNDS AND METHODS OF PREPARATION AND USE THEREOF

by SCHMITT JEFFREY DANIEL, GENEVOIS BORELLA ARIELLE, CAPET MARC, CHEVE MICHEL, DULL GARY MAURICE
Year of Publication 16.02.2012

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Patent

1-OXO-ISOINDOLINE-4-CARBOXAMIDE AND 1-OXO-1,2,3,4-TETRAHYDROISOQUINOLINE-5-CARBOXAMIDE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF

1-OXO-ISOINDOLINE-4-CARBOXAMIDE AND 1-OXO-1,2,3,4-TETRAHYDROISOQUINOLINE-5-CARBOXAMIDE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF

by BAUDOIN BERNARD, GENEVOIS BORELLA ARIELLE, MALLERON JEAN LUC, MATHIEU MAGALI, EVERS MICHEL, KARLSSON ANDREAS
Year of Publication 18.05.2010

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Patent

1,2,3,4-TETRAHYDROPYRROLO[1,2-A]PYRAZINE-6-CARBOXAMIDE AND 2,3,4,5-TETRAHYDROPYRROLO[1,2-A][1,4]-DIAZEPINE-7-CARBOXAMIDE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF

1,2,3,4-TETRAHYDROPYRROLO[1,2-A]PYRAZINE-6-CARBOXAMIDE AND 2,3,4,5-TETRAHYDROPYRROLO[1,2-A][1,4]-DIAZEPINE-7-CARBOXAMIDE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF

by BAUDOIN BERNARD, GENEVOIS BORELLA ARIELLE, MALLERON JEAN LUC, MATHIEU MAGALI, EVERS MICHEL, KARLSSON ANDREAS
Year of Publication 13.05.2010

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Patent

Abstract 130: Pharmacological effects of selective xCT inhibition in ARID1A mutated cancer models

Abstract 130: Pharmacological effects of selective xCT inhibition in ARID1A mutated cancer models

by Henry, Christophe, Péron, Philippe, Blanchet, Anne-Marie, Genevois-Borella, Arielle, Trellu, Marc, Bourges, Dorothée, Lienard, Philippe, Basset, Alexandra, Jouannot, Erwan, Philippo, Christophe, Debussche, Laurent, Moll, Jürgen
Published in Cancer research (Chicago, Ill.) (15.06.2022)

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Journal Article

A preparative route to fused indeno[1,2-e][1,2,4]-triazolo[4,3-a]pyrazin-4-ones

A preparative route to fused indeno[1,2-e][1,2,4]-triazolo[4,3-a]pyrazin-4-ones

by Ribeill, Y, Genevois-Borella, A, Vuilhorgne, M, Mignani, S
Published in Heterocycles (01.12.1999)

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Journal Article

PYRAZOLOPYRAZINONE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND THERAPEUTIC USES THEREOF

PYRAZOLOPYRAZINONE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND THERAPEUTIC USES THEREOF

by GENEVOIS-BORELLA, Arielle, OBINU-REIBAUD, Maria-Carmen
Year of Publication 05.10.2023

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Patent

A convenient one-pot synthesis of phosphino-dipeptide analogs

A convenient one-pot synthesis of phosphino-dipeptide analogs

by Cristau, Henri-Jean, Coulombeau, Agnès, Genevois-Borella, Arielle, Pirat, Jean-Luc
Published in Tetrahedron letters (02.07.2001)

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Journal Article

PYRAZOLOPYRAZINE COMPOUNDS AS SHP2 INHIBITORS

PYRAZOLOPYRAZINE COMPOUNDS AS SHP2 INHIBITORS

by KARLSSON, Andreas, DEVILLERS, Ingrid, GENEVOIS-BORELLA, Arielle, BEGIS, Guillaume, FORICHER, Yann, GILL, Adrian L, BIANCIOTTO, Marc, KOLTUN, Elena S
Year of Publication 23.10.2024

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Patent

Preparation of phosphinodipeptide analogs as building blocks for pseudopeptides synthesis

Preparation of phosphinodipeptide analogs as building blocks for pseudopeptides synthesis

by Cristau, Henri-Jean, Coulombeau, Agnès, Genevois-Borella, Arielle, Sanchez, Frédéric, Pirat, Jean-Luc
Published in Journal of organometallic chemistry (01.02.2002)

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Journal Article

9-Carboxymethyl-5H, 10H-imidazo[1,2-a]indeno[1,2-e]pyrazin-4-one-2-carbocylic acid (RPR117824): Selective anticonvulsive and neuroprotective AMPA antagonist

9-Carboxymethyl-5H, 10H-imidazo[1,2-a]indeno[1,2-e]pyrazin-4-one-2-carbocylic acid (RPR117824): Selective anticonvulsive and neuroprotective AMPA antagonist

by MIGNANI, Serge, BOHME, Georg Andrees, WAHL, Florence, STUTZMANN, Jean-Marie, BIRRAUX, Guillaume, BOIREAU, T. Alain, JIMONET, Patrick, DAMOUR, Dominique, GENEVOIS-BORELLA, Arielle, DEBONO, Marc-Williams, PRATT, Jeremy, VUILHORGNE, Marc
Published in Bioorganic & medicinal chemistry (01.05.2002)

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Journal Article

PYRAZOLOPYRAZINE COMPOUNDS AS SHP2 INHIBITORS

PYRAZOLOPYRAZINE COMPOUNDS AS SHP2 INHIBITORS

by KARLSSON, Andreas, DEVILLERS, Ingrid, GENEVOIS-BORELLA, Arielle, BEGIS, Guillaume, FORICHER, Yann, GILL, Adrian L, BIANCIOTTO, Marc, KOLTUN, Elena S
Year of Publication 22.06.2023

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Patent

Enantioselective synthesis of (+)-3-isorauniticine via a catalytic tandem palladium-ene/carbonylation reaction

Enantioselective synthesis of (+)-3-isorauniticine via a catalytic tandem palladium-ene/carbonylation reaction

by Oppolzer, Wolfgang, Bienayme, Hugues, Genevois-Borella, Arielle
Published in Journal of the American Chemical Society (01.12.1991)

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Journal Article

MACROCYCLIC COMPOUNDS, COMPOSITIONS AND METHODS OF USING THEREOF

MACROCYCLIC COMPOUNDS, COMPOSITIONS AND METHODS OF USING THEREOF

by BORCHERDING, David, GUESSREGEN, Stefan, GAO, Zhongli, CAUSSANEL, Franck, GOOD, Andrew, BERNADELLI, Patrick, DEVILLERS, Ingrid, SCHWINK, Lothar, RACKELMANN, Nils, THURAIRATNAM, Sukanthini, HIRTH, Brad, LIU, Jinyu, HURLBUT, Greg, GENEVOIS-BORELLA, Arielle, TOPALOV, George, THOMPSON, Fabienne, RUF, Sven, MACOR, John, VAZ, Roy, LI, Yi, LIAO, Junkai, GLOMBIK, Heiner, NICOLAI, Eric, RUVINSKY, Anatoly, MUNSON, Mark, KOTHE, Michael, PODESCHWA, Michael, SLOWINSKI, Franck
Year of Publication 14.03.2024

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Patent

MACROCYCLIC COMPOUNDS, COMPOSITIONS, AND METHODS OF USING THEREOF

MACROCYCLIC COMPOUNDS, COMPOSITIONS, AND METHODS OF USING THEREOF

by BORCHERDING, David, GUESSREGEN, Stefan, GAO, Zhongli, CAUSSANEL, Franck, GOOD, Andrew, DEVILLERS, Ingrid, SCHWINK, Lothar, RACKELMANN, Nils, THURAIRATNAM, Sukanthini, HIRTH, Brad, LIU, Jinyu, HURLBUT, Greg, GENEVOIS-BORELLA, Arielle, TOPALOV, George, THOMPSON, Fabienne, RUF, Sven, MACOR, John, VAZ, Roy, LI, Yi, BERNARDELLI, Patrick, LIAO, Junkai, GLOMBIK, Heiner, NICOLAI, Eric, RUVINSKY, Anatoly, MUNSON, Mark, KOTHE, Michael, PODESCHWA, Michael, SLOWINSKI, Franck
Year of Publication 14.03.2024

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Patent

9-Carboxymethyl-5 H ,10 H -imidazo[1,2- a ]indeno[1,2- e ]pyrazin-4-one-2-carbocylic Acid (RPR117824): Selective Anticonvulsive and Neuroprotective AMPA Antagonist

9-Carboxymethyl-5 H ,10 H -imidazo[1,2- a ]indeno[1,2- e ]pyrazin-4-one-2-carbocylic Acid (RPR117824): Selective Anticonvulsive and Neuroprotective AMPA Antagonist

by Mignani, Serge, Bohme, Georg Andrees, Birraux, Guillaume, Boireau, Alain, Jimonet, Patrick, Damour, Dominique, Genevois-Borella, Arielle, Debono, Marc-Williams, Pratt, Jeremy, Vuilhorgne, Marc, Wahl, Florence, Stutzmann, Jean-Marie
Published in Bioorganic & medicinal chemistry (01.05.2002)

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Journal Article

Indeno[1,2-b]pyrazin-2,3-diones: A New Class of Antagonists at the Glycine Site of the NMDA Receptor with Potent in Vivo Activity

Indeno[1,2-b]pyrazin-2,3-diones: A New Class of Antagonists at the Glycine Site of the NMDA Receptor with Potent in Vivo Activity

by Jimonet, Patrick, Ribeill, Yves, Bohme, Georg Andrees, Boireau, Alain, Chevé, Michel, Damour, Dominique, Doble, Adam, Genevois-Borella, Arielle, Herman, Frédéric, Imperato, Assunta, Le Guern, Sylvain, Manfré, Franco, Pratt, Jeremy, Randle, John C. R, Stutzmann, Jean-Marie, Mignani, Serge
Published in Journal of medicinal chemistry (15.06.2000)

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