Rational Design of Potent Non-Nucleoside Inhibitors of HIV‑1 Reverse Transcriptase
Chong, Pek, Sebahar, Paul, Youngman, Michael, Garrido, Dulce, Zhang, Huichang, Stewart, Eugene L., Nolte, Robert T., Wang, Liping, Ferris, Robert G., Edelstein, Mark, Weaver, Kurt, Mathis, Amanda, Peat, Andrew
Published in Journal of medicinal chemistry (13.12.2012)
Published in Journal of medicinal chemistry (13.12.2012)
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Synthesis and activity of small molecule GPR40 agonists
Garrido, Dulce M., Corbett, David F., Dwornik, Kate A., Goetz, Aaron S., Littleton, Thomas R., McKeown, Steve C., Mills, Wendy Y., Smalley, Terrence L., Briscoe, Celia P., Peat, Andrew J.
Published in Bioorganic & medicinal chemistry letters (01.04.2006)
Published in Bioorganic & medicinal chemistry letters (01.04.2006)
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Anthranilimide based glycogen phosphorylase inhibitors for the treatment of type 2 diabetes. Part 3: X-ray crystallographic characterization, core and urea optimization and in vivo efficacy
Thomson, Stephen A., Banker, Pierette, Bickett, D. Mark, Boucheron, Joyce A., Carter, H. Luke, Clancy, Daphne C., Cooper, Joel P., Dickerson, Scott H., Garrido, Dulce M., Nolte, Robert T., Peat, Andrew J., Sheckler, Lauren R., Sparks, Steven M., Tavares, Francis X., Wang, Liping, Wang, Tony Y., Weiel, James E.
Published in Bioorganic & medicinal chemistry letters (15.02.2009)
Published in Bioorganic & medicinal chemistry letters (15.02.2009)
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The discovery and optimization of pyrimidinone-containing MCH R1 antagonists
Hertzog, Donald L., Al-Barazanji, Kamal A., Bigham, Eric C., Bishop, Michael J., Britt, Christy S., Carlton, David L., Cooper, Joel P., Daniels, Alex J., Garrido, Dulce M., Goetz, Aaron S., Grizzle, Mary K., Guo, Yu C., Handlon, Anthony L., Ignar, Diane M., Morgan, Ronda O., Peat, Andrew J., Tavares, Francis X., Zhou, Huiqiang
Published in Bioorganic & medicinal chemistry letters (15.09.2006)
Published in Bioorganic & medicinal chemistry letters (15.09.2006)
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Synthesis and evaluation of novel heterocyclic inhibitors of GSK-3
Smalley, Terrence L., Peat, Andrew J., Boucheron, Joyce A., Dickerson, Scott, Garrido, Dulce, Preugschat, Frank, Schweiker, Stephanie L., Thomson, Stephen A., Wang, Tony Y.
Published in Bioorganic & medicinal chemistry letters (15.04.2006)
Published in Bioorganic & medicinal chemistry letters (15.04.2006)
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Anthranilimide-based glycogen phosphorylase inhibitors for the treatment of Type 2 diabetes: 2. Optimization of serine and threonine ether amino acid residues
Sparks, Steven M., Banker, Pierette, Bickett, David M., Clancy, Daphne C., Dickerson, Scott H., Garrido, Dulce M., Golden, Pamela L., Peat, Andrew J., Sheckler, Lauren R., Tavares, Francis X., Thomson, Stephen A., Weiel, James E.
Published in Bioorganic & medicinal chemistry letters (01.02.2009)
Published in Bioorganic & medicinal chemistry letters (01.02.2009)
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6-(4-Chlorophenyl)-3-substituted-thieno[3,2-d]pyrimidin-4(3H)-one-Based Melanin-Concentrating Hormone Receptor 1 Antagonist
Tavares, Francis X, Al-Barazanji, Kamal A, Bishop, Michael J, Britt, Christy S, Carlton, David L, Cooper, Joel P, Feldman, Paul L, Garrido, Dulce M, Goetz, Aaron S, Grizzle, Mary K, Hertzog, Donald L, Ignar, Diane M, Lang, Daniel G, McIntyre, Maggie S, Ott, Ronda J, Peat, Andrew J, Zhou, Hui-Qiang
Published in Journal of medicinal chemistry (30.11.2006)
Published in Journal of medicinal chemistry (30.11.2006)
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Anthranilimide-based glycogen phosphorylase inhibitors for the treatment of type 2 diabetes: 1. Identification of 1-amino-1-cycloalkyl carboxylic acid headgroups
Sparks, Steven M., Banker, Pierette, Bickett, David M., Carter, H. Luke, Clancy, Daphne C., Dickerson, Scott H., Dwornik, Kate A., Garrido, Dulce M., Golden, Pamela L., Nolte, Robert T., Peat, Andrew J., Sheckler, Lauren R., Tavares, Francis X., Thomson, Stephen A., Wang, Liping, Weiel, James E.
Published in Bioorganic & medicinal chemistry letters (01.02.2009)
Published in Bioorganic & medicinal chemistry letters (01.02.2009)
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3-(αR)-α-((2S,5R)-4-Allyl-2,5-dimethyl-1-piperazinyl)-3-hydroxybenzyl)- N-alkyl-N-arylbenzamides: Potent, Non-Peptidic Agonists of Both the μ and δ Opioid Receptors
Bishop, Michael J, Garrido, Dulce M, Boswell, G. Evan, Collins, Mark A, Harris, Philip A, McNutt, Robert W, O'Neill, Scott J, Wei, Ke, Chang, Kwen-Jen
Published in Journal of medicinal chemistry (13.02.2003)
Published in Journal of medicinal chemistry (13.02.2003)
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A novel one-pot synthesis of N-substituted thieno[3,2-d]pyrimidin-4(3H)-ones
Peat, Andrew J., Feldman, Paul L., Garrido, Dulce, Guo, Yu C., Hertzog, Donald L.
Published in Heterocycles (31.12.2006)
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Design and synthesis of spirocyclic compounds as HCV replication inhibitors by targeting viral NS4B protein
Tai, Vincent W.-F., Garrido, Dulce, Price, Daniel J., Maynard, Andrew, Pouliot, Jeffrey J., Xiong, Zhiping, Seal, John W., Creech, Katrina L., Kryn, Luz H., Baughman, Todd M., Peat, Andrew J.
Published in Bioorganic & medicinal chemistry letters (15.05.2014)
Published in Bioorganic & medicinal chemistry letters (15.05.2014)
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Imidazo[1,2-a]pyridines That Directly Interact with Hepatitis C NS4B: Initial Preclinical Characterization
Shotwell, J. Brad, Baskaran, Subramanian, Chong, Pek, Creech, Katrina L, Crosby, Renae M, Dickson, Hamilton, Fang, Jing, Garrido, Dulce, Mathis, Amanda, Maung, Jack, Parks, Derek J, Pouliot, Jeffrey J, Price, Daniel J, Rai, Roopa, Seal, John W, Schmitz, Uli, Tai, Vincent W. F, Thomson, Michael, Xie, Mi, Xiong, Zhiping Z, Peat, Andrew J
Published in ACS medicinal chemistry letters (12.07.2012)
Published in ACS medicinal chemistry letters (12.07.2012)
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Novel pyrazolopyrimidine derivatives as GSK-3 inhibitors
PEAT, Andrew J, BOUCHERON, Joyce A, WANG, Tony Y, ZHOU, Huiqiang Q, THOMSON, Stephen A, DICKERSON, Scott H, GARRIDO, Dulce, MILLS, Wendy, PECKHAM, Jennifer, PREUGSCHAT, Frank, SMALLEY, Terrence, SCHWEIKER, Stephanie L, WILSON, Jayme R
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
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3-Trifluoromethyl-4-nitro-5-arylpyrazoles are novel K ATP channel agonists
Peat, Andrew J., Townsend, Claire, Craig McKay, M., Garrido, Dulce, Terry, Christopher M., Wilson, Jayme L.R., Thomson, Stephen A.
Published in Bioorganic & medicinal chemistry letters (09.02.2004)
Published in Bioorganic & medicinal chemistry letters (09.02.2004)
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3-(alphaR)-alpha-((2S,5R)-4-allyl-2,5-dimethyl-1-piperazinyl)-3-hydroxybenzyl)-N-alkyl-N-arylbenzamides: potent, non-peptidic agonists of both the micro and delta opioid receptors
Bishop, Michael J, Garrido, Dulce M, Boswell, G Evan, Collins, Mark A, Harris, Philip A, McNutt, Robert W, O'Neill, Scott J, Wei, Ke, Chang, Kwen-Jen
Published in Journal of medicinal chemistry (13.02.2003)
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Published in Journal of medicinal chemistry (13.02.2003)
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3-(αR) -α-((2S, 5R)-4-allyl-2,5-dimethyl-1-piperazinyl)-3-hydroxybenzyl-N-alkyl-N-arylb enzamides: Potent, non-peptidic agonists of both the μ and δ opioid receptors
BISHOP, Michael J, GARRIDO, Dulce M, BOSWELL, G. Evan, COLLINS, Mark A, HARRIS, Philip A, MCNUTT, Robert W, O'NEILL, Scott J, KE WEI, CHANG, Kwen-Jen
Published in Journal of medicinal chemistry (2003)
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Published in Journal of medicinal chemistry (2003)
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Synthesis and evaluation of 7-substituted-3-cyclobutylamino-4H-1,2,4-benzothiadiazine-1,1-dioxide derivatives as KATP channel agonists
PEAT, Andrew J, TOWNSEND, Claire, THOMSON, Stephen A, WORLEY, Jennings F, ALLEN, Scott H, GARRIDO, Dulce, MERTZ, Robert J, PFOHL, Jeffrey L, TERRY, Christopher M, TRUAX, Jim F, VEASEY, Robert L
Published in Bioorganic & medicinal chemistry letters (21.10.2002)
Published in Bioorganic & medicinal chemistry letters (21.10.2002)
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