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Glaser, K.B., Li, J., Pease, L.J., Staver, M.J., Marcotte, P.A., Guo, J., Frey, R.R., Garland, R.B., Heyman, H.R., Wada, C.K., Vasudevan, A., Michaelides, M.R., Davidsen, S.K., Curtin, M.L.
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Potent in vitro and in vivo inhibitors of platelet aggregation based upon the Arg-Gly-Asp-Phe sequence of fibrinogen. A proposal on the nature of the binding interaction between the Arg-guanidine of RGDX mimetics and the platelet GP IIb-IIIa receptor
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Published in Journal of medicinal chemistry (01.06.1993)
Published in Journal of medicinal chemistry (01.06.1993)
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The design, synthesis, and structure-activity relationships of a series of macrocyclic MMP inhibitors
Steinman, Douglas H., Curtin, Michael L., Garland, Robert B., Davidsen, Steven K., Heyman, H.Robin, Holms, James H., Albert, Daniel H., Magoc, Terry J., Nagy, Ildiko B., Marcotte, Patrick A., Li, Junling, Morgan, Douglas W., Hutchins, Charles, Summers, James B.
Published in Bioorganic & medicinal chemistry letters (18.08.1998)
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Phenoxyphenyl Sulfone N-Formylhydroxylamines (Retrohydroxamates) as Potent, Selective, Orally Bioavailable Matrix Metalloproteinase Inhibitors
Wada, Carol K, Holms, James H, Curtin, Michael L, Dai, Yujia, Florjancic, Alan S, Garland, Robert B, Guo, Yan, Heyman, H. Robin, Stacey, Jamie R, Steinman, Douglas H, Albert, Daniel H, Bouska, Jennifer J, Elmore, Ildiko N, Goodfellow, Carole L, Marcotte, Patrick A, Tapang, Paul, Morgan, Douglas W, Michaelides, Michael R, Davidsen, Steven K
Published in Journal of medicinal chemistry (03.01.2002)
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Discovery and characterization of the potent, selective and orally bioavailable MMP inhibitor ABT-770
Curtin, Michael L., Florjancic, Alan S., Heyman, H.Robin, Michaelides, Michael R., Garland, Robert B., Holms, James H., Steinman, Douglas H., Dellaria, Joseph F., Gong, Jane, Wada, Carol K., Guo, Yan, Elmore, Ildiko B., Tapang, Paul, Albert, Daniel H., Magoc, Terrance J., Marcotte, Patrick A., Bouska, Jennifer J., Goodfellow, Carole L., Bauch, Joy L., Marsh, Kennan C., Morgan, Douglas W., Davidsen, Steven K.
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
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Broad spectrum matrix metalloproteinase inhibitors : An examination of succinamide hydroxamate inhibitors with p1 Cα gem-disubstitution
CURTIN, M. L, GARLAND, R. B, DAVIDSEN, S. K, MARCOTTE, P. A, ALBERT, D. H, MAGOC, T. J, HUTCHINS, C
Published in Bioorganic & medicinal chemistry letters (16.06.1998)
Published in Bioorganic & medicinal chemistry letters (16.06.1998)
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Design of orally active, non-peptide fibrinogen receptor antagonists. An evolutionary process from the RGD sequence to novel anti-platelet aggregation agents
Bovy, P.R., Tjoeng, F.S., Rico, J.G., Rogers, T.E., Lindmark, R.J., Zablocki, J.A., Garland, R.B., McMackins, D.E., Dayringer, H., Tóth, M.V., Zupec, M.E., Rao, S., Panzer-Knodle, S.G., Nicholson, N.S., Salyers, A., Taite, B.B., Herin, M., Miyano, M., Feigen, L.P., Adams, S.P.
Published in Bioorganic & medicinal chemistry (01.09.1994)
Published in Bioorganic & medicinal chemistry (01.09.1994)
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A novel series of orally active antiplatelet agents
Zablocki, Jeffery A., Tjoeng, Foe S., Bovy, Philippe R., Miyano, Masateru, Garland, Robert B., Williams, Kenneth, Schretzman, Lori, Zupec, Mark E., Rico, Joseph G., Lindmark, Richard J., Toth, Mihaly V., McMackins, Dudley E., Adams, Steven P., Panzer-Knodle, Susan G., Nicholson, Nancy S., Taite, Beatrice B., Salyers, Anita K., King, Lucy W., Campion, James G., Feigen, Larry P.
Published in Bioorganic & medicinal chemistry (01.05.1995)
Published in Bioorganic & medicinal chemistry (01.05.1995)
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Evaluation of the Inhibition of other Metalloproteinases by Matrix Metalloproteinase Inhibitors
Marcotte, Patrick A., Elmore, Ildiko N., Guan, Zhiwen, Magoc, Terrance J., Albert, Daniel H., Morgan, Douglas W., Curtin, Michael L., Garland, Robert B., Guo, Yan, Heyman, H. Robin, Holms, James H., Sheppard, George S., Steinman, Douglas H., Wada, Carol K., Davidsen, Steven K.
Published in Journal of enzyme inhibition (01.01.1999)
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Synthesis of 5-fluoroprostacyclin
Djuric, Stevan W, Garland, Robert B, Nysted, Leonard N, Pappo, Raphael, Plume, Gatis, Swenton, Lydia
Published in Journal of organic chemistry (01.03.1987)
Published in Journal of organic chemistry (01.03.1987)
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Trifluoromethyl ketones as inhibitors of histone deacetylase
Frey, Robin R., Wada, Carol K., Garland, Robert B., Curtin, Michael L., Michaelides, Michael R., Li, Junling, Pease, Lori J., Glaser, Keith B., Marcotte, Patrick A., Bouska, Jennifer J., Murphy, Shannon S., Davidsen, Steven K.
Published in Bioorganic & medicinal chemistry letters (02.12.2002)
Published in Bioorganic & medicinal chemistry letters (02.12.2002)
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Potent in Vitro and in Vivo Inhibitors of Platelet Aggregation Based Upon the Arg-Gly-Asp Sequence of Fibrinogen. (Aminobenzamidino)succinyl (ABAS) Series of Orally Active Fibrinogen Receptor Antagonists
Zablocki, Jeffery A, Rico, Joseph G, Garland, Robert B, Rogers, Thomas E, Williams, Kenneth, Schretzman, Lori A, Rao, Shashidhar A, Bovy, Philippe R, Tjoeng, Foe S
Published in Journal of medicinal chemistry (01.06.1995)
Published in Journal of medicinal chemistry (01.06.1995)
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Succinimide hydroxamic acids as potent inhibitors of histone deacetylase (HDAC)
CURTIN, Michael L, GARLAND, Robert B, HEYMAN, H. Robin, FREY, Robin R, MICHAELIDES, Michael R, JUNLING LI, PEASE, Lori J, GLASER, Keith B, MARCOTTE, Patrick A, DAVIDSEN, Steven K
Published in Bioorganic & medicinal chemistry letters (21.10.2002)
Published in Bioorganic & medicinal chemistry letters (21.10.2002)
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α-Keto amides as inhibitors of histone deacetylase
Wada, Carol K., Frey, Robin R., Ji, Zhiqin, Curtin, Michael L., Garland, Robert B., Holms, James H., Li, Junling, Pease, Lori J., Guo, Jun, Glaser, Keith B., Marcotte, Patrick A., Richardson, Paul L., Murphy, Shannon S., Bouska, Jennifer J., Tapang, Paul, Magoc, Terrance J., Albert, Daniel H., Davidsen, Steven K., Michaelides, Michael R.
Published in Bioorganic & medicinal chemistry letters (06.10.2003)
Published in Bioorganic & medicinal chemistry letters (06.10.2003)
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Potent in vitro and in vivo inhibitors of platelet aggregation based upon the Arg-Gly-Asp sequence of fibrinogen. (Aminobenzamidino)succinyl (ABAS) series of orally activ fibrinogen receptor antagonists
ZABLOCKI, J. A, RICO, J. G, TOTH, M. V, ZUPEC, M. E, MCMACKINS, D. E, ADAMS, S. P, MIYANO, M, MARKOS, C. S, MILTON, M. N, PAULSON, S, HERIN, M, JACQMIN, P, GARLAND, R. B, NICHOLSON, N. S, PANZER-KNODLE, S. G, HAAS, N. F, PAGE, J. D, SZALONY, J. A, TAITE, B. B, SALYERS, A. K, KING, L. W, CAMPION, J. G, FEIGEN, L. P, ROGERS, T. E, WILLIAMS, K, SCHRETZMAN, L. A, RAO, S. A, BOVY, P. R, TJOENG, F. S, LINDMARK, R. J
Published in Journal of medicinal chemistry (1995)
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Published in Journal of medicinal chemistry (1995)
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