Exploration of the HDAC2 foot pocket: Synthesis and SAR of substituted N-(2-aminophenyl)benzamides
Bressi, Jerome C., Jennings, Andy J., Skene, Robert, Wu, Yiqin, Melkus, Robert, Jong, Ron De, O’Connell, Shawn, Grimshaw, Charles E., Navre, Marc, Gangloff, Anthony R.
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
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Journal Article
Discovery of novel benzo[b][1,4]oxazin-3(4H)-ones as poly(ADP-ribose)polymerase inhibitors
Gangloff, Anthony R., Brown, Jason, de Jong, Ron, Dougan, Douglas R., Grimshaw, Charles E., Hixon, Mark, Jennings, Andy, Kamran, Ruhi, Kiryanov, Andre, O’Connell, Shawn, Taylor, Ewan, Vu, Phong
Published in Bioorganic & medicinal chemistry letters (15.08.2013)
Published in Bioorganic & medicinal chemistry letters (15.08.2013)
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Journal Article
Benzimidazole and imidazole inhibitors of histone deacetylases: Synthesis and biological activity
Bressi, Jerome C., Jong, Ron de, Wu, Yiqin, Jennings, Andy J., Brown, Jason W., O’Connell, Shawn, Tari, Leslie W., Skene, Robert J., Vu, Phong, Navre, Marc, Cao, Xiaodong, Gangloff, Anthony R.
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
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Journal Article
Highly potent non-peptidic inhibitors of the HCV NS3/NS4A serine protease
Sperandio, David, Gangloff, Anthony R., Litvak, Joane, Goldsmith, Richard, Hataye, Jason M., Wang, Vivian R., Shelton, Emma J., Elrod, Kyle, Janc, James W., Clark, James M., Rice, Ken, Weinheimer, Steve, Yeung, Kap-Sun, Meanwell, Nicholas A., Hernandez, Dennis, Staab, Andrew J., Venables, Brian L., Spencer, Jeffrey R.
Published in Bioorganic & medicinal chemistry letters (04.11.2002)
Published in Bioorganic & medicinal chemistry letters (04.11.2002)
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Journal Article
Light-induced, iodine-catalyzed aerobic oxidation of unsaturated tertiary amines
Gangloff, Anthony R, Judge, Thomas M, Helquist, Paul
Published in Journal of organic chemistry (01.05.1990)
Published in Journal of organic chemistry (01.05.1990)
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Journal Article
Dibasic inhibitors of human mast cell tryptase. Part 2: Structure–activity relationships and requirements for potent activity
Rice, Kenneth D, Wang, Vivian R, Gangloff, Anthony R, Kuo, Elaine Y.-L, Dener, Jeffrey M, Newcomb, William S, Young, Wendy B, Putnam, Daun, Cregar, Lynne, Wong, Martin, Simpson, Paul J
Published in Bioorganic & medicinal chemistry letters (16.10.2000)
Published in Bioorganic & medicinal chemistry letters (16.10.2000)
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Journal Article
Dibasic inhibitors of human mast cell tryptase. Part 1: Synthesis and optimization of a novel class of inhibitors
Rice, Kenneth D, Gangloff, Anthony R, Kuo, Elaine Y.-L, Dener, Jeffrey M, Wang, Vivian R, Lum, Robert, Newcomb, William S, Havel, Chris, Putnam, Daun, Cregar, Lynne, Wong, Martin, Warne, Robert L
Published in Bioorganic & medicinal chemistry letters (16.10.2000)
Published in Bioorganic & medicinal chemistry letters (16.10.2000)
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Journal Article
Dibasic Inhibitors of Human Mast Cell Tryptase. Part 3: Identification of a Series of Potent and Selective Inhibitors Containing the Benzamidine Functionality
Dener, Jeffrey M., Rice, Kenneth D., Newcomb, William S., Wang, Vivian R., Young, Wendy B., Gangloff, Anthony R., Kuo, Elaine Y.-L., Cregar, Lynne, Putnam, Daun, Wong, Martin
Published in Bioorganic & medicinal chemistry letters (09.07.2001)
Published in Bioorganic & medicinal chemistry letters (09.07.2001)
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Journal Article
Monocharged inhibitors of mast cell tryptase derived from potent and selective dibasic inhibitors
Dener, Jeffrey M, Wang, Vivian R, Rice, Kenneth D, Gangloff, Anthony R, Kuo, Elaine Y.-L, Newcomb, William S, Putnam, Daun, Wong, Martin
Published in Bioorganic & medicinal chemistry letters (03.09.2001)
Published in Bioorganic & medicinal chemistry letters (03.09.2001)
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Journal Article
POLY(ADP-RIBOSE)POLYMERASE(PARP) INHIBITORS
KIRYANOV ANDRE A, GANGLOFF ANTHONY R, JONES BENJAMIN, JENNINGS ANDREW JOHN
Year of Publication 30.09.2011
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Year of Publication 30.09.2011
Patent
Abstract 5676: Discovery of novel benzo[b][1,4]oxazin-3(4H)-ones as poly(ADP-Ribose)polymerase inhibitors
Gangloff, Anthony R., Brown, Jason, De Jong, Ron, Erickson, Philip, Grimshaw, Charles, Hixon, Mark, Jennings, Andy, Kamran, Ruhi, Kiryanov, Andre, O'Connell, Shawn, Taylor, Ewan, Vu, Phong
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Published in Cancer research (Chicago, Ill.) (15.04.2013)
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Journal Article
FORMATION, ISOLATION, AND IDENTIFICATION OF PRODUCTS FROM THE INACTIVATION OF VIRGINIAMYCIN M1 BY Actinoplanes utahensis
GIAMBATTISTA, MARIO DI, VANNUFFEL, PASCAL, COCITO, CARLO, FRIEBEE, TIMOTHY L., GANGLOFF, ANTHONY R., HELQUIST, PUAL
Published in Journal of antibiotics (01.01.1994)
Published in Journal of antibiotics (01.01.1994)
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Journal Article
Heteroarylamide inhibitors of TBK1
Keung, Walter, Vu, Phong H, Bigi, Simone, Gangloff, Anthony R, Woodhead, Steven John, Swann, Steve
Year of Publication 12.06.2018
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Year of Publication 12.06.2018
Patent
inibidores de poli (adp-ribose) polimerase (parp)
Benjamin Jones, Andre A. Kiryanov, Andrew John Jennings, Anthony R. Gangloff
Year of Publication 06.03.2018
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Year of Publication 06.03.2018
Patent
HETEROARYLAMIDE INHIBITORS OF TBK1
Vu Phong H, Gangloff Anthony R, Swann Steve, Bigi Simone, Woodhead Steven John, Keung Walter
Year of Publication 02.11.2017
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Year of Publication 02.11.2017
Patent
Heteroarylamide inhibitors of TBK1
Gangloff Anthony R, Scorah Nicholas, Kwok Lily, Wang Haixia, Sabat Mark, Woodhead Steven John, Keung Walter
Year of Publication 21.03.2017
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Year of Publication 21.03.2017
Patent