Discovery of 4-amino-3-arylsulfoquinolines, a novel non-acetylenic chemotype of metabotropic glutamate 5 (mGlu5) receptor negative allosteric modulators
Galambos, János, Bielik, Attila, Wágner, Gábor, Domány, György, Kóti, János, Béni, Zoltán, Szigetvári, Áron, Sánta, Zsuzsanna, Orgován, Zoltán, Bobok, Amrita, Kiss, Béla, Mikó-Bakk, Mónika L., Vastag, Mónika, Sághy, Katalin, Krasavin, Mikhail, Gál, Krisztina, Greiner, István, Szombathelyi, Zsolt, Keserű, György M.
Published in European journal of medicinal chemistry (16.06.2017)
Published in European journal of medicinal chemistry (16.06.2017)
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Journal Article
4-Aryl-3-arylsulfonyl-quinolines as negative allosteric modulators of metabotropic GluR5 receptors: From HTS hit to development candidate
Galambos, János, Domány, György, Nógrádi, Katalin, Wágner, Gábor, Keserű, György M., Bobok, Amrita, Kolok, Sándor, Mikó-Bakk, Mónika L., Vastag, Mónika, Sághy, Katalin, Kóti, János, Szakács, Zoltán, Béni, Zoltán, Gál, Krisztina, Szombathelyi, Zsolt, Greiner, István
Published in Bioorganic & medicinal chemistry letters (15.02.2016)
Published in Bioorganic & medicinal chemistry letters (15.02.2016)
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Journal Article
NMR and mass spectrometric characterization of vinblastine, vincristine and some new related impurities—Part II
Háda, Viktor, Dubrovay, Zsófia, Lakó-Futó, Ágnes, Galambos, János, Gulyás, Zoltán, Aranyi, Antal, Szántay, Csaba
Published in Journal of pharmaceutical and biomedical analysis (01.10.2013)
Published in Journal of pharmaceutical and biomedical analysis (01.10.2013)
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Journal Article
Carbamoyloximes as novel non-competitive mGlu5 receptor antagonists
Galambos, János, Wágner, Gábor, Nógrádi, Katalin, Bielik, Attila, Molnár, László, Bobok, Amrita, Horváth, Attila, Kiss, Béla, Kolok, Sándor, Nagy, József, Kurkó, Dalma, Bakk, Mónika L., Vastag, Mónika, Sághy, Katalin, Gyertyán, István, Gál, Krisztina, Greiner, István, Szombathelyi, Zsolt, Keserű, György M., Domány, György
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
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Journal Article
Novel sulfonamides having dual dopamine D2 and D3 receptor affinity show in vivo antipsychotic efficacy with beneficial cognitive and EPS profile
Ágai-Csongor, Éva, Nógrádi, Katalin, Galambos, János, Vágó, István, Bielik, Attila, Magdó, Ildikó, Ignácz-Szendrei, Györgyi, Keserű, György Miklós, Greiner, István, Laszlovszky, István, Béla Kiss, Éva Schmidt, Judit Laszy, Katalin Sághy, Gyertyán, István, Zájer-Balázs, Mária, Gémesi, Larisza, Domány, György
Published in Bioorganic & medicinal chemistry letters (01.10.2007)
Published in Bioorganic & medicinal chemistry letters (01.10.2007)
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Journal Article
Discovery and Preclinical Characterization of 3‑((4-(4-Chlorophenyl)-7-fluoroquinoline-3-yl)sulfonyl)benzonitrile, a Novel Non-acetylenic Metabotropic Glutamate Receptor 5 (mGluR5) Negative Allosteric Modulator for Psychiatric Indications
Galambos, János, Bielik, Attila, Krasavin, Mikhail, Orgován, Zoltán, Domány, György, Nógrádi, Katalin, Wágner, Gábor, Balogh, György T, Béni, Zoltán, Kóti, János, Szakács, Zoltán, Bobok, Amrita, Kolok, Sándor, Mikó-Bakk, Mónika L, Vastag, Mónika, Sághy, Katalin, Laszy, Judit, Halász, Attila Sándor, Balázs, Ottilia, Gál, Krisztina, Greiner, István, Szombathelyi, Zsolt, Keserű, György M
Published in Journal of medicinal chemistry (23.03.2017)
Published in Journal of medicinal chemistry (23.03.2017)
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Journal Article
On Characterizations of Gamma Distribution
Lee, Min-Young, Galambos, Janos
Published in Bulletin of the Malaysian Mathematical Sciences Society (2015)
Published in Bulletin of the Malaysian Mathematical Sciences Society (2015)
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Journal Article
Classical Extreme Value Model and Prediction of Extreme Winds
Galambos, Janos, Macri, Nicholas
Published in Journal of structural engineering (New York, N.Y.) (01.07.1999)
Published in Journal of structural engineering (New York, N.Y.) (01.07.1999)
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Journal Article
Substituted (aza)indole derivatives
Ledneczki Istvan dr, Eles Janos dr, Horvath Anita dr, Galambos Janos dr, Nemethy Zsolt dr, Levay Gyoergy Istvan dr, Tapolcsanyi Pal dr
Year of Publication 28.02.2024
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Year of Publication 28.02.2024
Patent
Substituted (aza)indole derivatives
Ledneczki Istvan dr, Eles Janos dr, Horvath Anita dr, Galambos Janos dr, Nemethy Zsolt dr, Levay Gyoergy Istvan dr, Tapolcsanyi Pal dr
Year of Publication 28.01.2020
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Year of Publication 28.01.2020
Patent
PIPERAZINE SALT AND A PROCESS FOR THE PREPARATION THEREOF
AGAINE CSONGOR, Eva, JUHASZ, Balint, SEBOEK, Ferenc, NOGRADI, Katalin, CZIBULA, Laszlo, VAGO, Istvan, GALAMBOS, Janos
Year of Publication 28.04.2017
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Year of Publication 28.04.2017
Patent