Discovery of an inhibitor of the production of the Pseudomonas aeruginosa virulence factor pyocyanin in wild-type cells
Morkunas, Bernardas, Gal, Balint, Galloway, Warren R J D, Hodgkinson, James T, Ibbeson, Brett M, Tan, Yaw Sing, Welch, Martin, Spring, David R
Published in Beilstein journal of organic chemistry (11.07.2016)
Published in Beilstein journal of organic chemistry (11.07.2016)
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Journal Article
583 Novel, potent, and selective inhibitors of hypoxia-inducible factor (HIF)-2α reverse pro-tumorigenic transcriptional programming in cancer, stromal, and immune cells
Gauthier, Kelsey Sivick, Piovesan, Dana, Lawson, Kenneth, Cho, Soonweng, Udyavar, Akshata, Chan, Jean, Chen, Ada, Au, Jennie, Meleza, Cesar, Zhao, Xiaoning, Tran, Anh, Drew, Samuel, Gal, Balint, Rosen, Brandon, Leleti, Manmohan, Ginn, Elaine, Jin, Lixia, Young, Stephen, Powers, Jay, Walters, Matthew
Published in Journal for immunotherapy of cancer (01.11.2020)
Published in Journal for immunotherapy of cancer (01.11.2020)
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Abstract 1206: Discovery and characterization of AB521, a novel, potent, and selective hypoxia-inducible factor (HIF)-2α inhibitor
Lawson, Kenneth V., Gauthier, Kelsey E. Sivick, Mailyan, Artur K., Fournier, Jeremy T., Beatty, Joel W., Drew, Samuel L., Kalisiak, Jarek, Gal, Balint, Mata, Guillaume, Wang, Zhang, Yan, Xuelei, Jin, Lixia, Ginn, Elaine, Piovesan, Dana, Au, Jennifer, Meleza, Cesar A., Young, Stephen W., Walters, Matthew J., Leleti, Manmohan, Powers, Jay P.
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
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Abstract P206: AB521 potently and selectively inhibits pro-tumorigenic gene transcription by Hypoxia-Inducible Factor (HIF)-2α in vitro and in vivo
Gauthier, Kelsey E. Sivick, Piovesan, Dana, Cho, Soonweng, Lawson, Kenneth V., Schweickert, Patrick G., Lopez, Alejandra, Liu, Suan, Park, Timothy, Mailyan, Artur, Fournier, Jeremy T. A., Beatty, Joel W., Drew, Samuel L., Kalisiak, Jarek, Gal, Balint, Mata, Guillaume, Wang, Zhang, Rosen, Brandon R., Hardman, Clayton, Epplin, Matthaw P., Yu, Kai, Haelsig, Karl T., Jin, Lixia, Ginn, Elaine, Au, Jennie, Meleza, Cesar A., Tencer, Joel, Pham, Amber, Kwon, Hyock J., Young, Stephen W., Leleti, Manmohan, Powers, Jay P., Walters, Matthew J.
Published in Molecular cancer therapeutics (01.12.2021)
Published in Molecular cancer therapeutics (01.12.2021)
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Enantiospecific Solvolytic Functionalization of Bromochlorides
Burckle, Alexander J, Gál, Bálint, Seidl, Frederick J, Vasilev, Vasil H, Burns, Noah Z
Published in Journal of the American Chemical Society (27.09.2017)
Published in Journal of the American Chemical Society (27.09.2017)
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Journal Article
HIF-2알파의 저해제 및 이의 사용 방법
EPPLIN MATTHEW, LAWSON KENNETH VICTOR, ROSEN BRANDON REID, MATA GUILLAUME, HARDMAN CLAYTON, BEATTY JOEL WORLEY, LIU DONGDONG, FOURNIER JEREMY, POWERS JAY PATRICK, DREW SAMUEL LAWRIE, YU KAI, GAL BALINT, PODUNAVAC MASA, MAILYAN ARTUR KARENOVICH, LELETI MANMOHAN REDDY
Year of Publication 16.07.2024
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Year of Publication 16.07.2024
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Enantioselective Total Synthesis of the Archaeal Lipid Parallel GDGT‐0 (Isocaldarchaeol)
Falk, Isaac D., Gál, Bálint, Bhattacharya, Ahanjit, Wei, Jeremy H., Welander, Paula V., Boxer, Steven G., Burns, Noah Z.
Published in Angewandte Chemie International Edition (02.08.2021)
Published in Angewandte Chemie International Edition (02.08.2021)
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HIF-2알파의 억제제로서의 테트랄린 및 테트라히드로퀴놀린 화합물
JACOB STEVEN DONALD, LAWSON KENNETH VICTOR, GUNEY TEZCAN, MATA GUILLAUME, WANG ZHANG, JEFFREY JENNA LEIGH, SU YONGLI, MANDAL DEBASHIS, MOON HYUNYOUNG, HAELSIG KARL T, GAL BALINT, MAILYAN ARTUR KARENOVICH, EPPLIN MATTHEW, ROSEN BRANDON REID, LINDSEY ERICK ALLEN, HARDMAN CLAYTON, BEATTY JOEL WORLEY, FOURNIER JEREMY THOMAS ANDRE, YAN XUELEI, POWERS JAY PATRICK, DREW SAMUEL LAWRIE, YU KAI, KALISIAK JAROSLAW, TRAN ANH THU, LELETI MANMOHAN REDDY
Year of Publication 23.11.2022
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Year of Publication 23.11.2022
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COMPOUNDS AS INHIBITORS OF AXL
LELETI, Manmohan Reddy, LAMANI, Manjunath, PALADUGU, Srinivas, POWERS, Jay Patrick, MILES, Dillon Harding, BEATTY, Joel Worley, GAL, Balint, FOLEY, Corinne Nicole, QU, Shiwei
Year of Publication 25.04.2024
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Year of Publication 25.04.2024
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COMPOUNDS AS INHIBITORS OF AXL
LELETI, Manmohan Reddy, LAMANI, Manjunath, PALADUGU, Srinivas, POWERS, Jay Patrick, MILES, Dillon Harding, BEATTY, Joel Worley, GAL, Balint, FOLEY, Corinne Nicole, QU, Shiwei
Year of Publication 04.01.2024
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Year of Publication 04.01.2024
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COMPOUNDS AS INHIBITORS OF AXL
LELETI, Manmohan Reddy, LAMANI, Manjunath, PALADUGU, Srinivas, POWERS, Jay Patrick, MILES, Dillon Harding, BEATTY, Joel Worley, GAL, Balint, FOLEY, Corinne Nicole, QU, Shiwei
Year of Publication 28.12.2023
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Year of Publication 28.12.2023
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INHIBITORS OF HIF-2ALPHA AND METHODS OF USE THEREOF
LELETI, Manmohan Reddy, DREW, Samuel Lawrie, EPPLIN, Matthew, PODUNAVAC, Masa, MATA, Guillaume, ROSEN, Brandon Reid, HARDMAN, Clayton, FOURNIER, Jeremy, LIU, Dongdong, LAWSON, Kenneth Victor, YU, Kai, POWERS, Jay Patrick, BEATTY, Joel Worley, GAL, Balint, MAILYAN, Artur Karenovich
Year of Publication 04.09.2024
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Year of Publication 04.09.2024
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Inhibitors of HIF-2α and methods of use thereof
Gal, Balint, Yu, Kai, Liu, Dongdong, Mata, Guillaume, Epplin, Matthew, Mailyan, Artur Karenovich, Hardman, Clayton, Lawson, Kenneth Victor, Rosen, Brandon Reid, Podunavac, Ma{hacek over (s)}a, Drew, Samuel Lawrie, Powers, Jay Patrick, Fournier, Jeremy, Leleti, Manmohan Reddy, Beatty, Joel Worley
Year of Publication 27.08.2024
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Year of Publication 27.08.2024
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Inhibitors of hif-2alpha and methods of use thereof
BEATTY Joel Worley, FOURNIER Jeremy, LIU Dongdong, YU Kai, LELETI Manmohan Reddy, HARDMAN Clayton, MATA Guillaume, GAL Balint, POWERS Jay Patrick, ROSEN Brandon Reid, MAILYAN Artur Karenovich, EPPLIN Matthew, LAWSON Kenneth Victor, DREW Samuel Lawrie, PODUNAVAC Ma?a
Year of Publication 01.06.2024
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Year of Publication 01.06.2024
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INHIBITORS OF HIF-2ALPHA AND METHODS OF USE THEREOF
LELETI, Manmohan Reddy, DREW, Samuel Lawrie, EPPLIN, Matthew, MATA, Guillaume, ROSEN, Brandon Reid, HARDMAN, Clayton, FOURNIER, Jeremy, LIU, Dongdong, PODUNAVAC, Maša, LAWSON, Kenneth Victor, YU, Kai, POWERS, Jay Patrick, BEATTY, Joel Worley, GAL, Balint, MAILYAN, Artur Karenovich
Year of Publication 16.05.2024
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Year of Publication 16.05.2024
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CBL-B INHIBITORS AND METHODS OF USE THEREOF
GANGAM, Srikanth Kumar, LAWSON, Kenneth Victor, YU, Kai, LELETI, Manmohan Reddy, YU, Tzu-Yu, YIN, Xianglin, BEATTY, Joel Worley, GAL, Balint, MAILYAN, Artur Karenovich, HARDMAN, Clayton, LIU, Dongdong, PODUNAVAC, Maša
Year of Publication 25.01.2024
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Year of Publication 25.01.2024
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INHIBITORS OF HIF-2ALPHA AND METHODS OF USE THEREOF
LELETI, Manmohan Reddy, DREW, Samuel Lawrie, EPPLIN, Matthew, PODUNAVAC, Masa, MATA, Guillaume, ROSEN, Brandon Reid, HARDMAN, Clayton, FOURNIER, Jeremy, LIU, Dongdong, LAWSON, Kenneth Victor, YU, Kai, POWERS, Jay Patrick, BEATTY, Joel Worley, GAL, Balint, MAILYAN, Artur Karenovich
Year of Publication 25.05.2023
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Year of Publication 25.05.2023
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INHIBITORS OF HIF-2ALPHA AND METHODS OF USE THEREOF
LELETI, Manmohan Reddy, DREW, Samuel Lawrie, EPPLIN, Matthew, PODUNAVAC, Masa, MATA, Guillaume, ROSEN, Brandon Reid, HARDMAN, Clayton, FOURNIER, Jeremy, LIU, Dongdong, LAWSON, Kenneth Victor, YU, Kai, POWERS, Jay Patrick, BEATTY, Joel Worley, GAL, Balint, MAILYAN, Artur Karenovich
Year of Publication 04.05.2023
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Year of Publication 04.05.2023
Patent
TETRALIN AND TETRAHYDROQUINOLINE COMPOUNDS AS INHIBITORS OF HIF-2ALPHA
DREW, Samuel Lawrie, EPPLIN, Matthew, MOON, Hyunyoung, LINDSEY, Erick Allen, LAWSON, Kenneth Victor, POWERS, Jay Patrick, BEATTY, Joel Worley, GAL, Balint, JACOB, Steven Donald, MAILYAN, Artur Karenovich, FOURNIER, Jeremy Thomas Andre, MANDAL, Debashis, LELETI, Manmohan Reddy, WANG, Zhang, KALISIAK, Jaroslaw, MATA, Guillaume, ROSEN, Brandon Reid, JEFFREY, Jenna Leigh, HAELSIG, Karl T, HARDMAN, Clayton, TRAN, Anh Thu, YU, Kai, SU, Yongli, GUNEY, Tezcan, YAN, Xuelei
Year of Publication 01.08.2024
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Year of Publication 01.08.2024
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