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Anderson, Ethan J, Vistoli, Giulio, Katunga, Lalage A, Funai, Katsuhiko, Regazzoni, Luca, Monroe, T Blake, Gilardoni, Ettore, Cannizzaro, Luca, Colzani, Mara, De Maddis, Danilo, Rossoni, Giuseppe, Canevotti, Renato, Gagliardi, Stefania, Carini, Marina, Aldini, Giancarlo
Published in The Journal of clinical investigation (01.12.2018)
Published in The Journal of clinical investigation (01.12.2018)
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Synthesis of (+)-Dumetorine and Congeners by Using Flow Chemistry Technologies
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Published in Chemistry : a European journal (23.05.2011)
Published in Chemistry : a European journal (23.05.2011)
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Inhibition of Plasmodium falciparum pH regulation by small molecule indole derivatives results in rapid parasite death
van Schalkwyk, Donelly A., Chan, Xie W.A., Misiano, Paola, Gagliardi, Stefania, Farina, Carlo, Saliba, Kevin J.
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Published in Biochemical pharmacology (01.05.2010)
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Synthesis of photoactivable inhibitors of osteoclast vacuolar ATPase
Biasotti, Barbara, Dallavalle, Sabrina, Merlini, Lucio, Farina, Carlo, Gagliardi, Stefania, Parini, Carlo, Belfiore, Pietro
Published in Bioorganic & medicinal chemistry (15.05.2003)
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Synthesis and Structure−Activity Relationships of Bafilomycin A1 Derivatives as Inhibitors of Vacuolar H+-ATPase
Gagliardi, Stefania, Gatti, P. Andrea, Belfiore, Pietro, Zocchetti, Andrea, Clarke, Geoffrey D, Farina, Carlo
Published in Journal of medicinal chemistry (21.05.1998)
Published in Journal of medicinal chemistry (21.05.1998)
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Cinnamic Anilides as New Mitochondrial Permeability Transition Pore Inhibitors Endowed with Ischemia-Reperfusion Injury Protective Effect in Vivo
Fancelli, Daniele, Abate, Agnese, Amici, Raffaella, Bernardi, Paolo, Ballarini, Marco, Cappa, Anna, Carenzi, Giacomo, Colombo, Andrea, Contursi, Cristina, Di Lisa, Fabio, Dondio, Giulio, Gagliardi, Stefania, Milanesi, Eva, Minucci, Saverio, Pain, Gilles, Pelicci, Pier Giuseppe, Saccani, Alessandra, Storto, Mariangela, Thaler, Florian, Varasi, Mario, Villa, Manuela, Plyte, Simon
Published in Journal of medicinal chemistry (26.06.2014)
Published in Journal of medicinal chemistry (26.06.2014)
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Efficient Continuous Flow Synthesis of Hydroxamic Acids and Suberoylanilide Hydroxamic Acid Preparation
Riva, Elena, Gagliardi, Stefania, Mazzoni, Caterina, Passarella, Daniele, Rencurosi, Anna, Vigo, Daniele, Martinelli, Marisa
Published in Journal of organic chemistry (01.05.2009)
Published in Journal of organic chemistry (01.05.2009)
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Synthesis, biological characterization and molecular modeling insights of spirochromanes as potent HDAC inhibitors
Thaler, Florian, Moretti, Loris, Amici, Raffaella, Abate, Agnese, Colombo, Andrea, Carenzi, Giacomo, Fulco, Maria Carmela, Boggio, Roberto, Dondio, Giulio, Gagliardi, Stefania, Minucci, Saverio, Sartori, Luca, Varasi, Mario, Mercurio, Ciro
Published in European journal of medicinal chemistry (27.01.2016)
Published in European journal of medicinal chemistry (27.01.2016)
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Synthesis and biological characterization of spiro[2H-(1,3)-benzoxazine-2,4′-piperidine] based histone deacetylase inhibitors
Thaler, Florian, Varasi, Mario, Abate, Agnese, Carenzi, Giacomo, Colombo, Andrea, Bigogno, Chiara, Boggio, Roberto, Zuffo, Roberto Dal, Rapetti, Daniela, Resconi, Anna, Regalia, Nickolas, Vultaggio, Stefania, Dondio, Giulio, Gagliardi, Stefania, Minucci, Saverio, Mercurio, Ciro
Published in European journal of medicinal chemistry (01.06.2013)
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A novel series of metabotropic glutamate receptor 5 negative allosteric modulators based on a 4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine core
Duvey, Guillaume, Perry, Benjamin, Le Poul, Emmanuel, Poli, Sonia, Bonnet, Beatrice, Lambeng, Nathalie, Charvin, Delphine, Donovan-Rodrigues, Tansy, Haddouk, Hasnaà, Gagliardi, Stefania, Rocher, Jean-Philippe
Published in Bioorganic & medicinal chemistry letters (15.08.2013)
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Synthesis and biological evaluation of novel dimiracetam derivatives useful for the treatment of neuropathic pain
Farina, Carlo, Gagliardi, Stefania, Ghelardini, Carla, Martinelli, Marisa, Norcini, Monica, Parini, Carlo, Petrillo, Paola, Ronzoni, Silvano
Published in Bioorganic & medicinal chemistry (15.03.2008)
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Synthesis and Biological Evaluation of N-Hydroxyphenylacrylamides and N-Hydroxypyridin-2-ylacrylamides as Novel Histone Deacetylase Inhibitors
Thaler, Florian, Colombo, Andrea, Mai, Antonello, Amici, Raffaella, Bigogno, Chiara, Boggio, Roberto, Cappa, Anna, Carrara, Simone, Cataudella, Tiziana, Fusar, Fulvia, Gianti, Eleonora, di Ventimiglia, Samuele Joppolo, Moroni, Maurizio, Munari, Davide, Pain, Gilles, Regalia, Nickolas, Sartori, Luca, Vultaggio, Stefania, Dondio, Giulio, Gagliardi, Stefania, Minucci, Saverio, Mercurio, Ciro, Varasi, Mario
Published in Journal of medicinal chemistry (28.01.2010)
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(R) -NIFURATEL, ITS USE FOR THE TREATMENT OF INFECTIONS AND SYNTHESIS OF (R) AND (S)-NIFURATEL
GAGLIARDI STEFANIA, BULGHERONI ANNA, MAILLAND FEDERICO, CONSONNI ALESSANDRA
Year of Publication 23.01.2015
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Year of Publication 23.01.2015
Patent
Chiral Resolution and Pharmacological Characterization of the Enantiomers of the Hsp90 Inhibitor 2-Amino-7-[4-fluoro-2-(3-pyridyl)phenyl]-4-methyl-7,8-dihydro-6H-quinazolin-5-one Oxime
Amici, Raffaella, Bigogno, Chiara, Boggio, Roberto, Colombo, Andrea, Courtney, Stephen M., Dal Zuffo, Roberto, Dondio, Giulio, Fusar, Fulvia, Gagliardi, Stefania, Minucci, Saverio, Molteni, Marco, Montalbetti, Christian A. G. N., Mortoni, Annalisa, Varasi, Mario, Vultaggio, Stefania, Mercurio, Ciro
Published in ChemMedChem (01.07.2014)
Published in ChemMedChem (01.07.2014)
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NIFURATEL SULFOXIDE FOR USE IN THE TREATMENT OF BACTERIAL INFECTIONS
GAGLIARDI STEFANIA, RONZONI SILVANO, BULGHERONI ANNA, CONSONNI ALESSANDRA, CERIANI DANIELA
Year of Publication 04.09.2014
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Year of Publication 04.09.2014
Patent
Chiral Resolution and Pharmacological Characterization of the Enantiomers of the Hsp90 Inhibitor 2‐Amino‐7‐[4‐fluoro‐2‐(3‐pyridyl)phenyl]‐4‐methyl‐7,8‐dihydro‐6 H ‐quinazolin‐5‐one Oxime
Amici, Raffaella, Bigogno, Chiara, Boggio, Roberto, Colombo, Andrea, Courtney, Stephen M., Dal Zuffo, Roberto, Dondio, Giulio, Fusar, Fulvia, Gagliardi, Stefania, Minucci, Saverio, Molteni, Marco, Montalbetti, Christian A. G. N., Mortoni, Annalisa, Varasi, Mario, Vultaggio, Stefania, Mercurio, Ciro
Published in ChemMedChem (01.07.2014)
Published in ChemMedChem (01.07.2014)
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Spiro[chromane-2,4'-piperidine]-Based Histone Deacetylase Inhibitors with Improved invivo Activity
Thaler, Florian, Varasi, Mario, Carenzi, Giacomo, Colombo, Andrea, Abate, Agnese, Bigogno, Chiara, Boggio, Roberto, Carrara, Simone, Cataudella, Tiziana, DalZuffo, Roberto, Reali, Veronica, Vultaggio, Stefania, Dondio, Giulio, Gagliardi, Stefania, Minucci, Saverio, Mercurio, Ciro
Published in ChemMedChem (01.04.2012)
Published in ChemMedChem (01.04.2012)
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