4-(2-Chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]5-methyl-N-(2-propynyl)-1,3-thiazol-2-amine hydrochloride (SSR125543A): a potent and selective corticotrophin-releasing factor(1) receptor antagonist. I. Biochemical and pharmacological characterization
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Effects of the beta3-adrenoceptor (Adrb3) agonist SR58611A (amibegron) on serotonergic and noradrenergic transmission in the rodent: relevance to its antidepressant/anxiolytic-like profile
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Published in Neuroscience (02.10.2008)
Published in Neuroscience (02.10.2008)
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Effects of the beta sub(3)-adrenoceptor (Adrb3) agonist SR58611A (amibegron) on serotonergic and noradrenergic transmission in the rodent: Relevance to its antidepressant/anxiolytic-like profile
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Published in Neuroscience (02.10.2008)
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Binding sites for a peripheral type benzodiazepine antagonist ([3H]PK 11195) in human iris
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Published in Neuropharmacology (01.06.1987)
Published in Neuropharmacology (01.06.1987)
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PK 11195, an antagonist of peripheral type benzodiazepine receptors, modulates Bay K8644 sensitive but not beta- or H2-receptor sensitive voltage operated calcium channels in the guinea pig heart
Mestre, M, Carriot, T, Néliat, G, Uzan, A, Renault, C, Dubroeucq, M C, Guérémy, C, Doble, A, Le Fur, G
Published in Life sciences (1973) (28.07.1986)
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Development of tetrazole bioisosteres in angiotensin II antagonists
Ferrari, B., Taillades, J., Perreaut, P., Bernhart, C., Gougat, J., Guiraudou, P., Cazaubon, C., Roccon, A., Nisato, D., Le Fur, G., Brelière, J.C.
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Neurotensin is an antagonist of the human neurotensin NT2 receptor expressed in Chinese hamster ovary cells
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Decrease in lymphocyte [3H]spiroperidol binding sites in Parkinsonism
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Published in Life sciences (1973) (01.01.1980)
Published in Life sciences (1973) (01.01.1980)
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2-Amino-6-trifluoromethoxy benzothiazole, a possible antagonist of excitatory amino acid neurotransmission--I. Anticonvulsant properties
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Published in Neuropharmacology (1985)
Published in Neuropharmacology (1985)
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Effects of the β 3-adrenoceptor (Adrb3) agonist SR58611A (amibegron) on serotonergic and noradrenergic transmission in the rodent: Relevance to its antidepressant/anxiolytic-like profile
Claustre, Y., Leonetti, M., Santucci, V., Bougault, I., Desvignes, C., Rouquier, L., Aubin, N., Keane, P., Busch, S., Chen, Y., Palejwala, V., Tocci, M., Yamdagni, P., Didier, M., Avenet, P., Le Fur, G., Oury-Donat, F., Scatton, B., Steinberg, R.
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Published in Neuroscience (2008)
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Dual intracellular signaling pathways mediated by the human cannabinoid CB1 receptor
CALANDRA, B, PORTIER, M, KERNEIS, A, DELPECH, M, CARILLON, C, LE FUR, G, FERRARA, P, SHIRE, D
Published in European journal of pharmacology (25.06.1999)
Published in European journal of pharmacology (25.06.1999)
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Mutational analysis and molecular modelling of the antagonist SR 144528 binding site on the human cannabinoid CB2 receptor
GOULDSON, P, CALANDRA, B, LEGOUX, P, KERNEIS, A, RINALDI-CARMONA, M, BARTH, F, LE FUR, G, FERRARA, P, SHIRE, D
Published in European journal of pharmacology (28.07.2000)
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[3H]spiroperidol binding on lymphocytes: changes in two different groups of schizophrenic patients and effect of neuroleptic treatment
Le Fur, G, Zarifian, E, Phan, T, Cuche, H, Flamier, A, Bouchami, F, Burgevin, M C, Loo, H, Gérard, A, Uzan, A
Published in Life sciences (1973) (17.01.1983)
Published in Life sciences (1973) (17.01.1983)
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Expression of Central and Peripheral Cannabinoid Receptors in Human Immune Tissues and Leukocyte Subpopulations
Galiègue, Sylvaine, Mary, Sophie, Marchand, Jean, Dussossoy, Danielle, Carrière, Dominique, Carayon, Pierre, Bouaboula, Monsif, Shire, David, Fur, Gérard, Casellas, Pierre
Published in European journal of biochemistry (15.08.1995)
Published in European journal of biochemistry (15.08.1995)
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Biochemical evidence that 2-phenyl-4[(4-piperidinyl) ethyl]quinoline, a quinoline derivative with pure anticonflict properties, is a partial agonist of benzodiazepine receptors
Benavides, J, Malgouris, C, Flamier, A, Tur, C, Quarteronet, D, Begassat, F, Camelin, J C, Uzan, A, Gueremy, C, Le Fur, G
Published in Neuropharmacology (01.10.1984)
Published in Neuropharmacology (01.10.1984)
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Chapter 15 Nonpeptide vasopressin receptor antagonists: development of selective and orally active V1a, V2 and V1b receptor ligands
Serradeil-Le Gall, C., Wagnon, J., Valette, G., Garcia, G., Pascal, M., Maffrand, J.P., Le Fur, G.
Published in Progress in Brain Research (2002)
Published in Progress in Brain Research (2002)
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Characterization and localization of leptin receptors in the rat kidney
Serradeil-Le Gal, Claudine, Raufaste, Danièle, Brossard, Gabrielle, Pouzet, Brigitte, Marty, Eléonore, Maffrand, Jean-Pierre, Le Fur, Gérard
Published in FEBS letters (10.03.1997)
Published in FEBS letters (10.03.1997)
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