The significance of chirality in drug design and development
Brooks, W H, Guida, W C, Daniel, K G
Published in Current topics in medicinal chemistry (01.04.2011)
Published in Current topics in medicinal chemistry (01.04.2011)
Get more information
Journal Article
In vitro evaluation of trypanocidal activity in plants used in Argentine traditional medicine
Sülsen, V, Güida, C, Coussio, J, Paveto, C, Muschietti, L, Martino, V
Published in Parasitology research (1987) (01.03.2006)
Published in Parasitology research (1987) (01.03.2006)
Get full text
Journal Article
A Novel Inhibitor of STAT3 Homodimerization Selectively Suppresses STAT3 Activity and Malignant Transformation
XIAOLEI ZHANG, YING SUN, PIREDDU, Roberta, HUA YANG, URLAM, Murali K, LAWRENCE, Harshani R, GUIDA, Wayne C, LAWRENCE, Nicholas J, SEBTI, Saïd M
Published in Cancer research (Chicago, Ill.) (15.03.2013)
Published in Cancer research (Chicago, Ill.) (15.03.2013)
Get full text
Journal Article
Selective chemical probe inhibitor of Stat3, identified through structure-based virtual screening, induces antitumor activity
Siddiquee, Khandaker, Zhang, Shumin, Guida, Wayne C, Blaskovich, Michelle A, Greedy, Benjamin, Lawrence, Harshani R, Yip, M.L. Richard, Jove, Richard, McLaughlin, Mark M, Lawrence, Nicholas J, Sebti, Said M, Turkson, James
Published in Proceedings of the National Academy of Sciences - PNAS (01.05.2007)
Published in Proceedings of the National Academy of Sciences - PNAS (01.05.2007)
Get full text
Journal Article
Discovery of a Novel Shp2 Protein Tyrosine Phosphatase Inhibitor
Chen, Liwei, Sung, Shen-Shu, Yip, M L Richard, Lawrence, Harshani R, Ren, Yuan, Guida, Wayne C, Sebti, Said M, Lawrence, Nicholas J, Wu, Jie
Published in Molecular pharmacology (01.08.2006)
Published in Molecular pharmacology (01.08.2006)
Get full text
Journal Article
Accurate Prediction of Acidity Constants in Aqueous Solution via Density Functional Theory and Self-Consistent Reaction Field Methods
Klicić, Jasna J, Friesner, Richard A, Liu, Shi-Yi, Guida, Wayne C
Published in The journal of physical chemistry. A, Molecules, spectroscopy, kinetics, environment, & general theory (21.02.2002)
Published in The journal of physical chemistry. A, Molecules, spectroscopy, kinetics, environment, & general theory (21.02.2002)
Get full text
Journal Article
Heterozygous IGFALS Gene Variants in Idiopathic Short Stature and Normal Children: Impact on Height and the IGF System
Domené, Horacio M., Scaglia, Paula A., Martínez, Alicia S., Keselman, Ana C., Karabatas, Liliana M., Pipman, Viviana R., Bengolea, Sonia V., Guida, María C., Ropelato, María G., Ballerini, María G., Lescano, Eva M., Blanco, Miguel A., Heinrich, Juan J., Rey, Rodolfo A., Jasper, Héctor G.
Published in Hormone research in paediatrics (01.01.2013)
Published in Hormone research in paediatrics (01.01.2013)
Get full text
Journal Article
Fragment-Based and Structure-Guided Discovery and Optimization of Rho Kinase Inhibitors
Li, Rongshi, Martin, Mathew P, Liu, Yan, Wang, Binglin, Patel, Ronil A, Zhu, Jin-Yi, Sun, Nan, Pireddu, Roberta, Lawrence, Nicholas J, Li, Jiannong, Haura, Eric B, Sung, Shen-Shu, Guida, Wayne C, Schonbrunn, Ernst, Sebti, Said M
Published in Journal of medicinal chemistry (08.03.2012)
Published in Journal of medicinal chemistry (08.03.2012)
Get full text
Journal Article
Inhibitors of Src Homology-2 Domain Containing Protein Tyrosine Phosphatase-2 (Shp2) Based on Oxindole Scaffolds
Lawrence, Harshani R, Pireddu, Roberta, Chen, Liwei, Luo, Yunting, Sung, Shen-Shu, Szymanski, Ann Marie, Yip, M. L. Richard, Guida, Wayne C, Sebti, Saïd M, Wu, Jie, Lawrence, Nicholas J
Published in Journal of medicinal chemistry (28.08.2008)
Published in Journal of medicinal chemistry (28.08.2008)
Get full text
Journal Article
Inhibition of cellular Shp2 activity by a methyl ester analog of SPI-112
Chen, Liwei, Pernazza, Daniele, Scott, Latanya M., Lawrence, Harshani R., Ren, Yuan, Luo, Yunting, Wu, Xin, Sung, Shen-Shu, Guida, Wayne C., Sebti, Said M., Lawrence, Nicholas J., Wu, Jie
Published in Biochemical pharmacology (15.09.2010)
Published in Biochemical pharmacology (15.09.2010)
Get full text
Journal Article
The art and practice of structure-based drug design: A molecular modeling perspective
Bohacek, Regine S., McMartin, Colin, Guida, Wayne C.
Published in Medicinal research reviews (01.01.1996)
Published in Medicinal research reviews (01.01.1996)
Get full text
Journal Article
Docking studies and model development of tea polyphenol proteasome inhibitors: Applications to rational drug design
Smith, David M., Daniel, Kenyon G., Wang, Zhigang, Guida, Wayne C., Chan, Tak-Hang, Dou, Q. Ping
Published in Proteins, structure, function, and bioinformatics (01.01.2004)
Published in Proteins, structure, function, and bioinformatics (01.01.2004)
Get full text
Journal Article
Shp2 protein tyrosine phosphatase inhibitor activity of estramustine phosphate and its triterpenoid analogs
Scott, Latanya M., Chen, Liwei, Daniel, Kenyon G., Brooks, Wesley H., Guida, Wayne C., Lawrence, Harshani R., Sebti, Said M., Lawrence, Nicholas J., Wu, Jie
Published in Bioorganic & medicinal chemistry letters (15.01.2011)
Published in Bioorganic & medicinal chemistry letters (15.01.2011)
Get full text
Journal Article