Dynamic modulation of inflammatory pain-related affective and sensory symptoms by optical control of amygdala metabotropic glutamate receptor 4
Zussy, C, Gómez-Santacana, X, Rovira, X, De Bundel, D, Ferrazzo, S, Bosch, D, Asede, D, Malhaire, F, Acher, F, Giraldo, J, Valjent, E, Ehrlich, I, Ferraguti, F, Pin, J-P, Llebaria, A, Goudet, C
Published in Molecular psychiatry (01.03.2018)
Published in Molecular psychiatry (01.03.2018)
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Optical activation of endogenous metabotropic glutamate receptor 4 (mGlu 4 ) in the amygdala dynamically regulates symptoms associated with persistent inflammatory pain
Zussy, C, Gómez-Santacana, X, Rovira, X, De Bundel, D, Ferrazzo, S, Bosch, D, Asede, D, Malhaire, F, Acher, F, Giraldo, J, Valjent, E, Ehrlich, I, Ferraguti, F, Pin, J-P, Llebaria, A, Goudet, C
Published in Molecular Psychiatry (01.03.2018)
Published in Molecular Psychiatry (01.03.2018)
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A double effect molecular switch leads to a novel potent negative allosteric modulator of metabotropic glutamate receptor 5
Gómez-Santacana, X., Rovira, X., Dalton, J. A., Goudet, C., Pin, J. P., Gorostiza, P., Giraldo, J., Llebaria, A.
Published in MedChemComm (01.10.2014)
Published in MedChemComm (01.10.2014)
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A double effect molecular switch leads to a novel potent negative allosteric modulator of metabotropic glutamate receptor 5Electronic supplementary information (ESI) available: NMR spectra and HPLC/PDA, LC/MS and HRMS data. See DOI: 10.1039/c4md00208c
Gómez-Santacana, X, Rovira, X, Dalton, J. A, Goudet, C, Pin, J. P, Gorostiza, P, Giraldo, J, Llebaria, A
Year of Publication 24.09.2014
Year of Publication 24.09.2014
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An allosteric modulator to control endogenous G protein-coupled receptors with light
Pittolo, Silvia, Gómez-Santacana, Xavier, Eckelt, Kay, Rovira, Xavier, Dalton, James, Goudet, Cyril, Pin, Jean-Philippe, Llobet, Artur, Giraldo, Jesús, Llebaria, Amadeu, Gorostiza, Pau
Published in Nature chemical biology (01.10.2014)
Published in Nature chemical biology (01.10.2014)
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