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CB1 receptor antagonist rimonabant reverses the diet-induced obesity phenotype through the regulation of lipolysis and energy balance
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Published in The FASEB journal (01.09.2005)
Published in The FASEB journal (01.09.2005)
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Selective inhibition of sucrose and ethanol intake by SR 141716, an antagonist of central cannabinoid (CB1) receptors
ARNONE, M, MARUANI, J, CHAPERON, F, THIEBOT, M.-H, PONCELET, M, SOUBRIE, P, LE FUR, G
Published in Psychopharmacologia (01.07.1997)
Published in Psychopharmacologia (01.07.1997)
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Characterization of (2S,4R)-1-[5-Chloro-1-[(2,4-dimethoxyphenyl)sulfonyl]-3-(2-methoxy-phenyl)-2-oxo-2,3-dihydro-1H-indol-3-yl]-4-hydroxy-N,N-dimethyl-2-pyrrolidine carboxamide (SSR149415), a Selective and Orally Active Vasopressin V1b Receptor Antagonist
Serradeil-Le Gal, Claudine, Wagnon, Jean, Simiand, Jacques, Griebel, Guy, Lacour, Colette, Guillon, Gilles, Barberis, Claude, Brossard, Gabrielle, Soubrié, Philippe, Nisato, Dino, Pascal, Marc, Pruss, Rebecca, Scatton, Bernard, Maffrand, Jean-Pierre, Le Fur, Gérard
Published in The Journal of pharmacology and experimental therapeutics (01.03.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.03.2002)
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The Cannabinoid CB1 Receptor Antagonist Rimonabant (SR141716) Inhibits Cell Proliferation and Increases Markers of Adipocyte Maturation in Cultured Mouse 3T3 F442A Preadipocytes
Gary-Bobo, Magali, Elachouri, Ghizlane, Scatton, Bernard, Le Fur, Gérard, Oury-Donat, Florence, Bensaid, Mohammed
Published in Molecular pharmacology (01.02.2006)
Published in Molecular pharmacology (01.02.2006)
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An Amino-terminal Variant of the Central Cannabinoid Receptor Resulting from Alternative Splicing
Shire, D, Carillon, C, Kaghad, M, Calandra, B, Rinaldi-Carmona, M, Le Fur, G, Caput, D, Ferrara, P
Published in The Journal of biological chemistry (24.02.1995)
Published in The Journal of biological chemistry (24.02.1995)
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Role of Peripheral Benzodiazepine Receptors in Mitochondrial, Cellular, and Cardiac Damage Induced by Oxidative Stress and Ischemia-Reperfusion
Leducq, Nathalie, Bono, Françoise, Sulpice, Thierry, Vin, Val érie, Janiak, Philip, Fur, Gérard Le, O'Connor, Steve E., Herbert, Jean-Marc
Published in The Journal of pharmacology and experimental therapeutics (01.09.2003)
Published in The Journal of pharmacology and experimental therapeutics (01.09.2003)
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In vitro functional evidence of neuronal cannabinoid CB1 receptors in human ileum
Croci, Tiziano, Manara, Luciano, Aureggi, Giulio, Guagnini, Fabio, Rinaldi‐Carmona, Murielle, Maffrand, Jean‐Pierre, Fur, Gérard, Mukenge, Sylvain, Ferla, Gianfranco
Published in British journal of pharmacology (01.12.1998)
Published in British journal of pharmacology (01.12.1998)
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Modulation and Functional Involvement of CB2 Peripheral Cannabinoid Receptors During B-Cell Differentiation
Carayon, Pierre, Marchand, Jean, Dussossoy, Danielle, Derocq, Jean-Marie, Jbilo, Omar, Bord, Annie, Bouaboula, Monsif, Galiègue, Sylvaine, Mondière, Paul, Pénarier, Géraldine, Fur, Gérard Le, Defrance, Thierry, Casellas, Pierre
Published in Blood (15.11.1998)
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Stimulation of the β3-Adrenoceptor as a Novel Treatment Strategy for Anxiety and Depressive Disorders
STEMMELIN, Jeanne, COHEN, Caroline, STAHL, Stephen M, KEANE, Peter, AVENET, Patrick, SCATTON, Bernard, LE FUR, Gérard, GRIEBEL, Guy, TERRANOVA, Jean-Paul, LOPEZ-GRANCHA, Matilde, PICHAT, Philippe, BERGIS, Olivier, DECOBERT, Michel, SANTUCCI, Vincent, FRANCON, Dominique, ALONSO, Richard
Published in Neuropsychopharmacology (New York, N.Y.) (25.04.2007)
Published in Neuropsychopharmacology (New York, N.Y.) (25.04.2007)
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Expression of Central and Peripheral Cannabinoid Receptors in Human Immune Tissues and Leukocyte Subpopulations
Galiègue, Sylvaine, Mary, Sophie, Marchand, Jean, Dussossoy, Danielle, Carrière, Dominique, Carayon, Pierre, Bouaboula, Monsif, Shire, David, Fur, Gérard, Casellas, Pierre
Published in European journal of biochemistry (15.08.1995)
Published in European journal of biochemistry (15.08.1995)
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Biochemical and Pharmacological Profile of a Potent and Selective Nonpeptide Antagonist of the Neurotensin Receptor
Gully, Danielle, Canton, Maryse, Boigegrain, Robert, Jeanjean, Francis, Molimard, Jean-Charles, Poncelet, Martine, Gueudet, Christiane, Heaulme, Michel, Leyris, Roger, Brouard, Aline, Pelaprat, Didier, Labbe-Jullie, Catherine, Mazella, Jean, Soubrie, Philippe, Maffrand, Jean-Pierre, Rostene, William, Kitabgi, Patrick, Le Fur, Gerard
Published in Proceedings of the National Academy of Sciences - PNAS (01.01.1993)
Published in Proceedings of the National Academy of Sciences - PNAS (01.01.1993)
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SR141716A, a potent and selective antagonist of the brain cannabinoid receptor
Rinaldi-Carmona, Murielle, Barth, Francis, Héaulme, Michel, Shire, David, Calandra, Bernard, Congy, Christian, Martinez, Serge, Maruani, Jeanne, Néliat, Gervais, Caput, Daniel, Ferrara, Pascual, Soubrié, Philippe, Brelière, Jean Claude, Le Fur, Gérard
Published in FEBS letters (22.08.1994)
Published in FEBS letters (22.08.1994)
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Structural Features of the Central Cannabinoid CB1 Receptor Involved in the Binding of the Specific CB1 Antagonist SR 141716A
Shire, D, Calandra, B, Delpech, M, Dumont, X, Kaghad, M, Le Fur, G, Caput, D, Ferrara, P
Published in The Journal of biological chemistry (22.03.1996)
Published in The Journal of biological chemistry (22.03.1996)
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Role of tachykinins in castor oil diarrhoea in rats
Croci, Tiziano, Landi, Marco, Emonds‐Alt, Xavier, Fur, Gérard, Maffrand, Jean‐Pierre, Manara, Luciano
Published in British journal of pharmacology (01.06.1997)
Published in British journal of pharmacology (01.06.1997)
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Single and multiple doses of rimonabant antagonize acute effects of smoked cannabis in male cannabis users
HUESTIS, Marilyn A, BOYD, Susan J, HEISHMAN, Stephen J, PRESTON, Kenzie L, BONNET, Denis, LE FUR, Gerard, GORELICK, David A
Published in Psychopharmacologia (01.11.2007)
Published in Psychopharmacologia (01.11.2007)
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Permissive role of neurokinin NK3 receptors in NK1 receptor-mediated activation of the locus coeruleus revealed by SR 142801
Bert, Lionel, Rodier, Daniel, Bougault, Isabelle, Allouard, Nathalie, Le-Fur, Gérard, Soubrié, Philippe, Steinberg, Régis
Published in Synapse (New York, N.Y.) (01.01.2002)
Published in Synapse (New York, N.Y.) (01.01.2002)
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Functional identification of rat atypical β‐adrenoceptors by the first β3‐selective antagonists, aryloxypropanolaminotetralins
Manara, Luciano, Badone, Domenico, Baroni, Marco, Boccardi, Giovanni, Cecchi, Roberto, Croci, Tiziano, Giudice, Antonina, Guzzi, Umberto, Landi, Marco, Fur, Gérard
Published in British journal of pharmacology (01.02.1996)
Published in British journal of pharmacology (01.02.1996)
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