Discovery of 5-[5-Fluoro-2-oxo-1,2- dihydroindol-(3Z)-ylidenemethyl]-2,4- dimethyl-1H-pyrrole-3-carboxylic Acid (2-Diethylaminoethyl)amide, a Novel Tyrosine Kinase Inhibitor Targeting Vascular Endothelial and Platelet-Derived Growth Factor Receptor Tyrosine Kinase
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Published in Journal of medicinal chemistry (27.03.2003)
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Published in Bioorganic & medicinal chemistry letters (01.08.2013)
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Published in Bioorganic & medicinal chemistry letters (01.08.2013)
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Published in Bioorganic & medicinal chemistry letters (01.08.2013)
Published in Bioorganic & medicinal chemistry letters (01.08.2013)
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Pharmacological, Pharmacokinetic, and Primate Analgesic Efficacy Profile of the Novel Bradykinin B 1 Receptor Antagonist ELN441958
Hawkinson, Jon E., Szoke, Balazs G., Garofalo, Albert W., Hom, Dennis S., Zhang, Hongbing, Dreyer, Mark, Fukuda, Juri Y., Chen, Linda, Samant, Bhushan, Simmonds, Stellanie, Zeitz, Karla P., Wadsworth, Angie, Liao, Anna, Chavez, Raymond A., Zmolek, Wes, Ruslim, Lany, Bova, Michael P., Holcomb, Ryan, Butelman, Eduardo R., Ko, Mei-Chuan, Malmberg, Annika B.
Published in The Journal of pharmacology and experimental therapeutics (01.08.2007)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2007)
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Published in 日本呼吸ケア・リハビリテーション学会誌 (31.08.2014)
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Discovery of 5-[5-Fluoro-2-oxo-1,2- dihydroindol-(3 Z )-ylidenemethyl]-2,4- dimethyl-1 H -pyrrole-3-carboxylic Acid (2-Diethylaminoethyl)amide, a Novel Tyrosine Kinase Inhibitor Targeting Vascular Endothelial and Platelet-Derived Growth Factor Receptor Tyrosine Kinase
Sun, Li, Liang, Chris, Shirazian, Sheri, Zhou, Yong, Miller, Todd, Cui, Jean, Fukuda, Juri Y., Chu, Ji-Yu, Nematalla, Asaad, Wang, Xueyan, Chen, Hui, Sistla, Anand, Luu, Tony C., Tang, Flora, Wei, James, Tang, Cho
Published in Journal of medicinal chemistry (01.03.2003)
Published in Journal of medicinal chemistry (01.03.2003)
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ROSSITER KASSANDRA INEZ, SMITH JENIFER LEA, STAPPENBECK FRANK, XU YING-ZI, KONRADI ANDREI W, FUKUDA JURI Y, SEMKO CHRISTOPHER MICHAEL
Year of Publication 05.02.2013
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Year of Publication 05.02.2013
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