Continuous inhibition of 20-HETE synthesis by TS-011 improves neurological and functional outcomes after transient focal cerebral ischemia in rats
Tanaka, Yu, Omura, Tomohiro, Fukasawa, Misako, Horiuchi, Nobuko, Miyata, Noriyuki, Minagawa, Toshiya, Yoshida, Shigeru, Nakaike, Shiro
Published in Neuroscience research (01.12.2007)
Published in Neuroscience research (01.12.2007)
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Preclinical disposition of MGS0274 besylate, a prodrug of a potent group II metabotropic glutamate receptor agonist MGS0008 for the treatment of schizophrenia
Kinoshita, Kohnosuke, Ochi, Motoki, Iwata, Katsuya, Fukasawa, Misako, Yamaguchi, Jun‐ichi
Published in Pharmacology research & perspectives (01.10.2019)
Published in Pharmacology research & perspectives (01.10.2019)
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Effect of a new inhibitor of the synthesis of 20-HETE on cerebral ischemia reperfusion injury
OMURA, Tomohiro, TANAKA, Yu, NAKAIKE, Shiro, OKUYAMA, Shigeru, HARDER, Phi David R, ROMAN, Richard J, MIYATA, Noriyuki, KOIZUMI, Chie, SAKURAI, Takanobu, FUKASAWA, Misako, HACHIUMA, Kenji, MINAGAWA, Toshiya, SUSUMU, Teruo, YOSHIDA, Shigeru
Published in Stroke (1970) (01.05.2006)
Published in Stroke (1970) (01.05.2006)
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Safety and pharmacokinetic profiles of MGS0274 besylate (TS‐134), a novel metabotropic glutamate 2/3 receptor agonist prodrug, in healthy subjects
Watanabe, Mai, Marcy, Brian, Kinoshita, Kohnosuke, Fukasawa, Misako, Hikichi, Hirohiko, Chaki, Shigeyuki, Okuyama, Shigeru, Gevorkyan, Hakop, Yoshida, Shigeru
Published in British journal of clinical pharmacology (01.11.2020)
Published in British journal of clinical pharmacology (01.11.2020)
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Discovery of MGS0274, an ester prodrug of a metabotropic glutamate receptor 2/3 agonist with improved oral bioavailability
Urabe, Hiroki, Miyakoshi, Naoki, Ohtake, Norikazu, Nozoe, Akiko, Ochi, Motoki, Fukasawa, Misako, Kinoshita, Kohnosuke, Yamaguchi, Jun-ichi, Marumo, Toshiyuki, Hikichi, Hirohiko, Chaki, Shigeyuki, Hashihayata, Takashi
Published in European journal of medicinal chemistry (01.10.2020)
Published in European journal of medicinal chemistry (01.10.2020)
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Metabolism of N,N-Dipropyl-2-[4-Methoxy-3-(2-Phenyl-Ethoxy)-Phenyl]-Ethyl-Amine-Monohydrochloride (NE-100), A Novel Sigma Ligand: Contribution of Cytochrome P450 Forms Involved in the Formation of Individual Metabolites in Human Liver and Small Intestine
Yamamoto, Takahito, Hagima, Naoko, Fukasawa, Misako, Yamaguchi, Jun-ichi, Nakamura, Masato, Kohno, Yoshiro, Nagata, Kiyoshi, Yamazoe, Yasushi
Published in Drug metabolism and pharmacokinetics (2003)
Published in Drug metabolism and pharmacokinetics (2003)
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