Discovery of Potent Protease-Activated Receptor 4 Antagonists with in Vivo Antithrombotic Efficacy
Miller, Michael M, Banville, Jacques, Friends, Todd J, Gagnon, Mark, Hangeland, Jon J, Lavallée, Jean-François, Martel, Alain, O’Grady, Harold, Rémillard, Roger, Ruediger, Edward, Tremblay, François, Posy, Shana L, Allegretto, Nick J, Guarino, Victor R, Harden, David G, Harper, Timothy W, Hartl, Karen, Josephs, Jonathan, Malmstrom, Sarah, Watson, Carol, Yang, Yanou, Zhang, Ge, Wong, Pancras, Yang, Jing, Bouvier, Michel, Seiffert, Dietmar A, Wexler, Ruth R, Lawrence, R. Michael, Priestley, E. Scott, Marinier, Anne
Published in Journal of medicinal chemistry (22.08.2019)
Published in Journal of medicinal chemistry (22.08.2019)
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Journal Article
Phenylimidazoles as Potent and Selective Inhibitors of Coagulation Factor XIa with in Vivo Antithrombotic Activity
Hangeland, Jon J, Friends, Todd J, Rossi, Karen A, Smallheer, Joanne M, Wang, Cailan, Sun, Zhong, Corte, James R, Fang, Tianan, Wong, Pancras C, Rendina, Alan R, Barbera, Frank A, Bozarth, Jeffrey M, Luettgen, Joseph M, Watson, Carol A, Zhang, Ge, Wei, Anzhi, Ramamurthy, Vidhyashankar, Morin, Paul E, Bisacchi, Gregory S, Subramaniam, Srinath, Arunachalam, Piramanayagam, Mathur, Arvind, Seiffert, Dietmar A, Wexler, Ruth R, Quan, Mimi L
Published in Journal of medicinal chemistry (11.12.2014)
Published in Journal of medicinal chemistry (11.12.2014)
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Journal Article
Pyridine and pyridinone-based factor XIa inhibitors
Corte, James R., Fang, Tianan, Hangeland, Jon J., Friends, Todd J., Rendina, Alan R., Luettgen, Joseph M., Bozarth, Jeffrey M., Barbera, Frank A., Rossi, Karen A., Wei, Anzhi, Ramamurthy, Vidhyashankar, Morin, Paul E., Seiffert, Dietmar A., Wexler, Ruth R., Quan, Mimi L.
Published in Bioorganic & medicinal chemistry letters (15.02.2015)
Published in Bioorganic & medicinal chemistry letters (15.02.2015)
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Journal Article
PK/PD Disconnect Observed with a Reversible Endothelial Lipase Inhibitor
Hangeland, Jon J., Abell, Lynn M., Adam, Leonard P., Jiang, Ji, Friends, Todd J., Haque, Lauren E., Neels, James, Onorato, Joelle M., Chen, Alice Ye A., Taylor, David S., Yin, Xiaohong, Harrity, Thomas W., Basso, Michael D., Yang, Richard, Sleph, Paul G., Gordon, David A., Huang, Christine S., Wexler, Ruth R., Finlay, Heather J., Lawrence, R. Michael
Published in ACS medicinal chemistry letters (12.07.2018)
Published in ACS medicinal chemistry letters (12.07.2018)
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Journal Article
Design and SAR of selective T-type calcium channel antagonists containing a biaryl sulfonamide core
Hangeland, Jon J., Cheney, Daniel L., Friends, Todd J., Swartz, Stephen, Levesque, Paul C., Rich, Adam J., Sun, Lucy, Bridal, Terry R., Adam, Leonard P., Normandin, Diane E., Murugesan, Natesan, Ewing, William R.
Published in Bioorganic & medicinal chemistry (15.01.2008)
Published in Bioorganic & medicinal chemistry (15.01.2008)
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Journal Article
Thyroid receptor ligands. Part 2: Thyromimetics with improved selectivity for the thyroid hormone receptor beta
Hangeland, Jon J., Doweyko, Arthur M., Dejneka, Tamara, Friends, Todd J., Devasthale, Pratik, Mellström, Karin, Sandberg, Johnny, Grynfarb, Marlena, Sack, John S., Einspahr, Howard, Färnegårdh, Mathias, Husman, Bolette, Ljunggren, Jan, Koehler, Konrad, Sheppard, Cheryl, Malm, Johan, Ryono, Denis E.
Published in Bioorganic & medicinal chemistry letters (05.07.2004)
Published in Bioorganic & medicinal chemistry letters (05.07.2004)
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Journal Article
A new class of high affinity thyromimetics containing a phenyl-naphthylene core
Hangeland, Jon J., Friends, Todd J., Doweyko, Arthur M., Mellström, Karin, Sandberg, Johnny, Grynfarb, Marlena, Ryono, Denis E.
Published in Bioorganic & medicinal chemistry letters (15.10.2005)
Published in Bioorganic & medicinal chemistry letters (15.10.2005)
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Journal Article
RXFP1 효능제
MATHUR ARVIND, LI JIANQING, CLARKE ADAM JAMES, PASUNOORI LAXMAN, FRIENDS TODD J, WURTZ NICHOLAS R, MYERS MICHAEL C, PINTO DONALD J.P, PABBISETTY KUMAR BALASHANMUGA, SHAW SCOTT A, TORA GEORGE O, SU SHUN, VOKITS BENJAMIN P
Year of Publication 28.06.2024
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Year of Publication 28.06.2024
Patent
Characterization of monoacylglycerol acyltransferase 2 inhibitors by a novel probe in binding assays
Ma, Zhengping, Chao, Hannguang J., Turdi, Huji, Hangeland, Jon J., Friends, Todd, Kopcho, Lisa M., Lawrence, R. Michael, Cheng, Dong
Published in Analytical biochemistry (15.05.2016)
Published in Analytical biochemistry (15.05.2016)
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RXFP1 효능제
MATHUR ARVIND, LI JIANQING, CLARKE ADAM JAMES, FRIENDS TODD J, ORWAT MICHAEL J, BARRE DURGA BUCHI RAJU, MYERS MICHAEL C, PINTO DONALD J.P, KUMAR SREEKANTHA RATNA, PABBISETTY KUMAR BALASHANMUGA, SHAW SCOTT A, SMITH II LEON M, SU SHUN, VOKITS BENJAMIN P, POTTURI HIMA KIRAN
Year of Publication 21.06.2024
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Year of Publication 21.06.2024
Patent
RXFP1 효능제
MATHUR ARVIND, O'MALLEY DANIEL, LI JIANQING, CLARKE ADAM JAMES, LAWRENCE R. MICHAEL, PASUNOORI LAXMAN, FRIENDS TODD J, ORWAT MICHAEL J, WURTZ NICHOLAS R, BHOGADI VIKRAM, MYERS MICHAEL C, PINTO DONALD J.P, KUMAR SREEKANTHA RATNA, PABBISETTY KUMAR BALASHANMUGA, SHAW SCOTT A, SMITH II LEON M, TORA GEORGE O, SU SHUN, SRINIVAS PITANI VEERA VENKATA, FINLAY HEATHER, HEGDE SUBRAMANYA, BILDER DONNA M, VOKITS BENJAMIN P, POTTURI HIMA KIRAN
Year of Publication 28.06.2024
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Year of Publication 28.06.2024
Patent
Corrigendum to “A new class of high affinity thyromimetics containing a phenyl-naphthylene core” [Bioorg. Med. Chem. Lett. 15 (2005) 4579–4584]
Hangeland, Jon J., Friends, Todd J., Doweyko, Arthur M., Mellström, Karin, Sandberg, Johnny, Grynfarb, Marlena, Ryono, Denis E.
Published in Bioorganic & medicinal chemistry letters (2006)
Published in Bioorganic & medicinal chemistry letters (2006)
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Journal Article
RXFP1 AGONISTS
CLARKE, Adam James, WURTZ, Nicholas R, PABBISETTY, Kumar Balashanmuga, MYERS, Michael C, LI, Jianqing, SU, Shun, FRIENDS, Todd J, PASUNOORI, Laxman, PINTO, Donald J.P, SHAW, Scott A, TORA, George O, MATHUR, Arvind, VOKITS, Benjamin P
Year of Publication 04.09.2024
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Year of Publication 04.09.2024
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RXFP1 AGONISTS
CLARKE, Adam James, ORWAT, Michael J, SMITH, II, Leon M, KUMAR, Sreekantha Ratna, PABBISETTY, Kumar Balashanmuga, MYERS, Michael C, LI, Jianqing, SU, Shun, FRIENDS, Todd J, PINTO, Donald J.P, BARRE, Durga Buchi Raju, SHAW, Scott A, POTTURI, Hima Kiran, MATHUR, Arvind, VOKITS, Benjamin P
Year of Publication 04.09.2024
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Year of Publication 04.09.2024
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RXFP1 AGONISTS
CLARKE, Adam James, WURTZ, Nicholas R, PABBISETTY, Kumar Balashanmuga, MYERS, Michael C, LI, Jianqing, SU, Shun, FRIENDS, Todd J, PASUNOORI, Laxman, PINTO, Donald J.P, SHAW, Scott A, TORA, George O, MATHUR, Arvind, VOKITS, Benjamin P
Year of Publication 04.05.2023
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Year of Publication 04.05.2023
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BHOGADI, Vikram, CLARKE, Adam James, ORWAT, Michael J, WURTZ, Nicholas R, KUMAR, Sreekantha Ratna, HEGDE, Subramanya, FINLAY, Heather, PABBISETTY, Kumar Balashanmuga, MYERS, Michael C, O'MALLEY, Daniel, LI, Jianqing, SU, Shun, FRIENDS, Todd J, SMITH II, Leon M, PASUNOORI, Laxman, PINTO, Donald J.P, LAWRENCE, R. Michael, SRINIVAS, Pitani Veera Venkata, SHAW, Scott A, POTTURI, Hima Kiran, TORA, George O, BILDER, Donna M, MATHUR, Arvind, VOKITS, Benjamin P
Year of Publication 04.09.2024
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Year of Publication 04.09.2024
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BHOGADI, Vikram, CLARKE, Adam James, ORWAT, Michael J, WURTZ, Nicholas R, KUMAR, Sreekantha Ratna, HEGDE, Subramanya, FINLAY, Heather, PABBISETTY, Kumar Balashanmuga, MYERS, Michael C, O'MALLEY, Daniel, LI, Jianqing, SU, Shun, FRIENDS, Todd J, SMITH II, Leon M, PASUNOORI, Laxman, PINTO, Donald J.P, LAWRENCE, R. Michael, SRINIVAS, Pitani Veera Venkata, SHAW, Scott A, POTTURI, Hima Kiran, TORA, George O, BILDER, Donna M, MATHUR, Arvind, VOKITS, Benjamin P
Year of Publication 13.06.2024
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Year of Publication 13.06.2024
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Rxfp1 agonists
PINTO Donald J.P, FINLAY Heather, BHOGADI Vikram, PASUNOORI Laxman, KUMAR Sreekantha Ratna, MATHUR Arvind, POTTURI Hima Kiran, SMITH II Leon M, SU Shun, VOKITS Benjamin P, O'MALLEY Daniel, SHAW Scott A, FRIENDS Todd J, CLARKE Adam James, MYERS Michael C, BRISTOL-MYERS SQUIBB COMPANY, TORA George O, ORWAT Michael J, BILDER Donna M, LI Jianqing, HEGDE Subramanya, LAWRENCE R. Michael, PABBISETTY Kumar Balashanmuga, SRINIVAS Pitani Veera Venkata
Year of Publication 01.06.2024
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Year of Publication 01.06.2024
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RXFP1 AGONISTS
CLARKE, Adam James, ORWAT, Michael J, KUMAR, Sreekantha Ratna, PABBISETTY, Kumar Balashanmuga, MYERS, Michael C, LI, Jianqing, SU, Shun, FRIENDS, Todd J, PINTO, Donald J.P, SMITH, II, BARRE, Durga Buchi Raju, SHAW, Scott A, POTTURI, Hima Kiran, MATHUR, Arvind, VOKITS, Benjamin P
Year of Publication 04.05.2023
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Year of Publication 04.05.2023
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RXFP1 AGONISTS
BHOGADI, Vikram, CLARKE, Adam James, ORWAT, Michael J, WURTZ, Nicholas R, KUMAR, Sreekantha Ratna, HEGDE, Subramanya, FINLAY, Heather, PABBISETTY, Kumar Balashanmuga, MYERS, Michael C, O'MALLEY, Daniel, LI, Jianqing, SU, Shun, FRIENDS, Todd J, SMITH II, Leon M, PASUNOORI, Laxman, PINTO, Donald J.P, LAWRENCE, R. Michael, SRINIVAS, Pitani Veera Venkata, SHAW, Scott A, POTTURI, Hima Kiran, TORA, George O, BILDER, Donna M, MATHUR, Arvind, VOKITS, Benjamin P
Year of Publication 04.05.2023
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Year of Publication 04.05.2023
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