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Published in Chemistry : a European journal (02.01.2013)
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Published in Organic & biomolecular chemistry (14.08.2012)
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Published in Angewandte Chemie (01.07.2014)
Published in Angewandte Chemie (01.07.2014)
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Optimization of Triazine Nitriles as Rhodesain Inhibitors: Structure-Activity Relationships, Bioisosteric Imidazopyridine Nitriles, and X-ray Crystal Structure Analysis with Human CathepsinL
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Published in ChemMedChem (01.06.2013)
Published in ChemMedChem (01.06.2013)
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Tuning and predicting biological affinity: aryl nitriles as cysteine protease inhibitorsDedicated to Professor Wilfred van Gunsteren on the occasion of his 65th birthday.This article is part of the Organic & Biomolecular Chemistry 10th Anniversary issue.Electronic supplementary information (ESI) available: Detailed experimental procedures and spectroscopic data for all compounds, biological assays and additional figures and tables. See DOI: 10.1039/c2ob00034b
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Year of Publication 14.08.2012
Year of Publication 14.08.2012
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Journal Article
Optimization of Triazine Nitriles as Rhodesain Inhibitors: Structure-Activity Relationships, Bioisosteric Imidazopyridine Nitriles, and X-ray Crystal Structure Analysis with Human Cathepsin L
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Published in ChemMedChem (01.06.2013)
Published in ChemMedChem (01.06.2013)
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Identifizierung von Pyrrolopyrazinen als polypotente Liganden mit Antimalariawirkung
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Published in Angewandte Chemie (01.07.2014)
Published in Angewandte Chemie (01.07.2014)
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Identifizierung von Pyrrolopyrazinen als polypotente Liganden mit Antimalariawirkung
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Published in Angewandte Chemie (01.07.2014)
Published in Angewandte Chemie (01.07.2014)
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