Mechanistic Studies of the Inactivation of TEM-1 and P99 by NXL104, a Novel Non-β-Lactam β-Lactamase Inhibitor
STACHYRA, Thérèse, PECHEREAU, Marie-Claude, BRUNEAU, Jean-Michel, CLAUDON, Monique, FRERE, Jean-Marie, MIOSSEC, Christine, COLEMAN, Kenneth, BLACK, Michael T
Published in Antimicrobial Agents and Chemotherapy (01.12.2010)
Published in Antimicrobial Agents and Chemotherapy (01.12.2010)
Get full text
Journal Article
Interaction of Avibactam with Class B Metallo-β-Lactamases
Abboud, Martine I, Damblon, Christian, Brem, Jürgen, Smargiasso, Nicolas, Mercuri, Paola, Gilbert, Bernard, Rydzik, Anna M, Claridge, Timothy D W, Schofield, Christopher J, Frère, Jean-Marie
Published in Antimicrobial agents and chemotherapy (01.10.2016)
Published in Antimicrobial agents and chemotherapy (01.10.2016)
Get full text
Journal Article
Web Resource
Development of new drugs for an old target: the penicillin binding proteins
Zervosen, Astrid, Sauvage, Eric, Frère, Jean-Marie, Charlier, Paulette, Luxen, André
Published in Molecules (Basel, Switzerland) (24.10.2012)
Published in Molecules (Basel, Switzerland) (24.10.2012)
Get full text
Journal Article
Web Resource
Mercaptophosphonate Compounds as Broad-Spectrum Inhibitors of the Metallo-β-lactamases
Lassaux, Patricia, Hamel, Matthieu, Gulea, Mihaela, Delbrück, Heinrich, Mercuri, Paola Sandra, Horsfall, Louise, Dehareng, Dominique, Kupper, Michaël, Frère, Jean-Marie, Hoffmann, Kurt, Galleni, Moreno, Bebrone, Carine
Published in Journal of medicinal chemistry (08.07.2010)
Published in Journal of medicinal chemistry (08.07.2010)
Get full text
Journal Article
Web Resource
1,2,4‐Triazole‐3‐thione Compounds as Inhibitors of Dizinc Metallo‐β‐lactamases
Sevaille, Laurent, Gavara, Laurent, Bebrone, Carine, De Luca, Filomena, Nauton, Lionel, Achard, Maud, Mercuri, Paola, Tanfoni, Silvia, Borgianni, Luisa, Guyon, Carole, Lonjon, Pauline, Turan‐Zitouni, Gülhan, Dzieciolowski, Julia, Becker, Katja, Bénard, Lionel, Condon, Ciaran, Maillard, Ludovic, Martinez, Jean, Frère, Jean‐Marie, Dideberg, Otto, Galleni, Moreno, Docquier, Jean‐Denis, Hernandez, Jean‐François
Published in ChemMedChem (21.06.2017)
Published in ChemMedChem (21.06.2017)
Get full text
Journal Article
Web Resource
Macrophage-infectivity potentiator of Trypanosoma cruzi (TcMIP) is a new pro-type 1 immuno-stimulating protein for neonatal human cells and vaccines in mice
Radwanska, Magdalena, de Lemos Esteves, Frédéric, Linsen, Loes, Coltel, Nicolas, Cencig, Sabrina, Widart, Joelle, Massart, Anne-Cécile, Colson, Séverine, Di Paolo, Alexandre, Percier, Pauline, Ait Djebbara, Sarra, Guillonneau, François, Flamand, Véronique, De Pauw, Edwin, Frère, Jean-Marie, Carlier, Yves, Truyens, Carine
Published in Frontiers in immunology (23.03.2023)
Published in Frontiers in immunology (23.03.2023)
Get full text
Journal Article
Web Resource
Ir-CPI, a coagulation contact phase inhibitor from the tick Ixodes ricinus, inhibits thrombus formation without impairing hemostasis
Decrem, Yves, Rath, Géraldine, Blasioli, Virginie, Cauchie, Philippe, Robert, Séverine, Beaufays, Jérôme, Frère, Jean-Marie, Feron, Olivier, Dogné, Jean-Michel, Dessy, Chantal, Vanhamme, Luc, Godfroid, Edmond
Published in The Journal of experimental medicine (26.10.2009)
Published in The Journal of experimental medicine (26.10.2009)
Get full text
Journal Article
Mutational Analysis of VIM-2 Reveals an Essential Determinant for Metallo-β-Lactamase Stability and Folding
BORGIANNI, Luisa, VANDENAMEELE, Julie, MATAGNE, André, BINI, Luca, BONOMO, Robert A, FRERE, Jean-Marie, ROSSOLINI, Gian Maria, DOCQUIER, Jean-Denis
Published in Antimicrobial Agents and Chemotherapy (01.08.2010)
Published in Antimicrobial Agents and Chemotherapy (01.08.2010)
Get full text
Journal Article
Web Resource
Activity of Ceftaroline against Enterococcus faecium PBP5
HENRY, Xavier, VERLAINE, Oliver, AMOROSO, Ana, COYETTE, Jacques, FRERE, Jean-Marie, JORIS, Bernard
Published in Antimicrobial Agents and Chemotherapy (01.12.2013)
Published in Antimicrobial Agents and Chemotherapy (01.12.2013)
Get full text
Journal Article
Web Resource
The CebE/MsiK Transporter is a Doorway to the Cello-oligosaccharide-mediated Induction of Streptomyces scabies Pathogenicity
Jourdan, Samuel, Francis, Isolde Maria, Kim, Min Jung, Salazar, Joren Jeico C, Planckaert, Sören, Frère, Jean-Marie, Matagne, André, Kerff, Frédéric, Devreese, Bart, Loria, Rosemary, Rigali, Sébastien
Published in Scientific reports (02.06.2016)
Published in Scientific reports (02.06.2016)
Get full text
Journal Article
Web Resource
Biochemical and Structural Characterization of the Subclass B1 Metallo-β-Lactamase VIM-4
LASSAUX, Patricia, TRAORE, Daouda A. K, GALLENI, Moreno, LOISEL, Elodie, FAVIER, Adrien, DOCQUIER, Jean-Denis, SOHIER, Jean Sébastien, LAURENT, Clémentine, BEBRONE, Carine, FRERE, Jean-Marie, FERRER, Jean-Luc
Published in Antimicrobial Agents and Chemotherapy (01.03.2011)
Published in Antimicrobial Agents and Chemotherapy (01.03.2011)
Get full text
Journal Article
Web Resource
Kinetic analysis of N-alkylaryl carboxamide hexitol nucleotides as substrates for evolved polymerases
Renders, Marleen, Dumbre, Shrinivas, Abramov, Mikhail, Kestemont, Donaat, Margamuljana, Lia, Largy, Eric, Cozens, Christopher, Vandenameele, Julie, Pinheiro, Vitor B, Toye, Dominique, Frère, Jean-Marie, Herdewijn, Piet
Published in Nucleic acids research (18.03.2019)
Published in Nucleic acids research (18.03.2019)
Get full text
Journal Article
Web Resource
The Structure of the Dizinc Subclass B2 Metallo-β-Lactamase CphA Reveals that the Second Inhibitory Zinc Ion Binds in the Histidine Site
Bebrone, Carine, Delbrück, Heinrich, Kupper, Michaël B, Schlömer, Philipp, Willmann, Charlotte, Frère, Jean-Marie, Fischer, Rainer, Galleni, Moreno, Hoffmann, Kurt M V
Published in Antimicrobial Agents and Chemotherapy (01.10.2009)
Published in Antimicrobial Agents and Chemotherapy (01.10.2009)
Get full text
Journal Article
An Extended Reservoir of Class-D Beta-Lactamases in Non-Clinical Bacterial Strains
Lupo, Valérian, Mercuri, Paola Sandra, Frère, Jean-Marie, Joris, Bernard, Galleni, Moreno, Baurain, Denis, Kerff, Frédéric
Published in Microbiology spectrum (27.04.2022)
Published in Microbiology spectrum (27.04.2022)
Get full text
Journal Article
Web Resource
Unexpected Tricovalent Binding Mode of Boronic Acids within the Active Site of a Penicillin-Binding Protein
Zervosen, Astrid, Herman, Raphael, Kerff, Frédéric, Herman, Alexandre, Bouillez, André, Prati, Fabio, Pratt, R. F, Frère, Jean-Marie, Joris, Bernard, Luxen, André, Charlier, Paulette, Sauvage, Eric
Published in Journal of the American Chemical Society (20.07.2011)
Published in Journal of the American Chemical Society (20.07.2011)
Get full text
Journal Article
Web Resource
Interactions between Avibactam and Ceftazidime-Hydrolyzing Class D β-Lactamases
Frère, Jean-Marie, Bogaerts, Pierre, Huang, Te-Din, Stefanic, Patrick, Moray, Joël, Bouillenne, Fabrice, Brans, Alain
Published in Biomolecules (Basel, Switzerland) (23.03.2020)
Published in Biomolecules (Basel, Switzerland) (23.03.2020)
Get full text
Journal Article
Web Resource
NH-1,2,3-Triazole Inhibitors of the VIM-2 Metallo-β-Lactamase
Weide, Timo, Saldanha, S. Adrian, Minond, Dmitriy, Spicer, Timothy P, Fotsing, Joseph R, Spaargaren, Michael, Frère, Jean-Marie, Bebrone, Carine, Sharpless, K. Barry, Hodder, Peter S, Fokin, Valery V
Published in ACS medicinal chemistry letters (08.07.2010)
Published in ACS medicinal chemistry letters (08.07.2010)
Get full text
Journal Article
Structural basis for the broad-spectrum inhibition of metallo-beta-lactamases by thiols
Lienard, Benoit M. R., Garau, Gianpiero, Horsfall, Louise, Karsisiotis, Andreas I., Damblon, Christian, Lassaux, Patricia, Papamicael, Cyril, Roberts, Gordon C. K., Galleni, Moreno, Dideberg, Otto, Frere, Jean-Marie, Schofield, Christopher J.
Published in Organic & biomolecular chemistry (01.01.2008)
Published in Organic & biomolecular chemistry (01.01.2008)
Get full text
Journal Article
Web Resource
β-Lactamase Inhibitors Derived from Single-Domain Antibody Fragments Elicited in the Camelidae
CONRATH, Katja E, LAUWEREYS, Marc, GALLENI, Moreno, MATAGNE, André, FRERE, Jean-Marie, KINNE, Jörg, WYNS, Lode, MUYLDERMANS, Serge
Published in Antimicrobial Agents and Chemotherapy (01.10.2001)
Published in Antimicrobial Agents and Chemotherapy (01.10.2001)
Get full text
Journal Article
Web Resource