HIV-1 Vaccine Development: Constrained Peptide Immunogens Show Improved Binding to the Anti-HIV-1 gp41 MAb
McGaughey, G. B, Citron, M, Danzeisen, R. C, Freidinger, R. M, Garsky, V. M, Hurni, W. M, Joyce, J. G, Liang, X, Miller, M, Shiver, J, Bogusky, M. J
Published in Biochemistry (Easton) (25.03.2003)
Published in Biochemistry (Easton) (25.03.2003)
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Methods for drug discovery: development of potent, selective, orally effective cholecystokinin antagonists
Evans, B. E, Rittle, K. E, Bock, M. G, DiPardo, R. M, Freidinger, R. M, Whitter, W. L, Lundell, G. F, Veber, D. F, Anderson, P. S, Chang, R. S. L, Lotti, V. J, Cerino, D. J, Chen, T. B, Kling, P. J, Kunkel, K. A, Springer, J. P, Hirshfield, J
Published in Journal of medicinal chemistry (01.12.1988)
Published in Journal of medicinal chemistry (01.12.1988)
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The Synthesis of a Prodrug of Doxorubicin Designed to Provide Reduced Systemic Toxicity and Greater Target Efficacy
Garsky, Victor M, Lumma, Patricia K, Feng, Dong-Mei, Wai, Jenny, Ramjit, Harri G, Sardana, Mohinder K, Oliff, Allen, Jones, Raymond E, DeFeo-Jones, Deborah, Freidinger, Roger M
Published in Journal of medicinal chemistry (22.11.2001)
Published in Journal of medicinal chemistry (22.11.2001)
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Journal Article
Design of Highly Potent Noncovalent Thrombin Inhibitors That Utilize a Novel Lipophilic Binding Pocket in the Thrombin Active Site
Tucker, Thomas J, Lumma, William C, Mulichak, Anne M, Chen, Zhongguo, Naylor-Olsen, Adel M, Lewis, S. Dale, Lucas, Robert, Freidinger, Roger M, Kuo, Lawrence C
Published in Journal of medicinal chemistry (14.03.1997)
Published in Journal of medicinal chemistry (14.03.1997)
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In vitro and in vivo evaluation of dihydropyrimidinone C-5 amides as potent and selective alpha(1A) receptor antagonists for the treatment of benign prostatic hyperplasia
Barrow, JC, Nantermet, PG, Selnick, HG, Glass, KL, Rittle, KE, Gilbert, KF, Steele, TG, Homnick, CF, Freidinger, RM, Ransom, RW, Kling, P, Reiss, D, Broten, TP, Schorn, TW, Chang, RSL, O'Malley, SS, Olah, TV, Ellis, JD, Barrish, A, Kassahun, K, Leppert, P, Nagarathnam, D, Forray, C
Published in Journal of medicinal chemistry (13.07.2000)
Published in Journal of medicinal chemistry (13.07.2000)
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Design of Potent, Orally Effective, Nonpeptidal Antagonists of the Peptide Hormone Cholecystokinin
Evans, Ben E., Bock, Mark G., Rittle, Kenneth E., DiPardo, Robert M., Whitter, Willie L., Veber, Daniel F., Anderson, Paul S., Freidinger, Roger M.
Published in Proceedings of the National Academy of Sciences - PNAS (01.07.1986)
Published in Proceedings of the National Academy of Sciences - PNAS (01.07.1986)
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Discovery of a Novel, Selective, and Orally Bioavailable Class of Thrombin Inhibitors Incorporating Aminopyridyl Moieties at the P1 Position
Feng, Dong-Mei, Gardell, Stephen J, Lewis, S. Dale, Bock, Mark G, Chen, Zhongguo, Freidinger, Roger M, Naylor-Olsen, Adel M, Ramjit, Harri G, Woltmann, Richard, Baskin, Elizabeth P, Lynch, Joseph J, Lucas, Robert, Shafer, Jules A, Dancheck, Kimberley B, Chen, I-Wu, Mao, Shi-Shan, Krueger, Julie A, Hare, Timothy R, Mulichak, Anne M, Vacca, Joseph P
Published in Journal of medicinal chemistry (07.11.1997)
Published in Journal of medicinal chemistry (07.11.1997)
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Journal Article
Benzodiazepine gastrin and brain cholecystokinin receptor ligands; L-365,260
Bock, Mark G, DiPardo, Robert M, Evans, Ben E, Rittle, Kenneth E, Whitter, Willie L, Veber, Daniel F, Anderson, Paul S, Freidinger, Roger M
Published in Journal of medicinal chemistry (01.01.1989)
Published in Journal of medicinal chemistry (01.01.1989)
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Characterization of the binding of [3H]L-365,260: a new potent and selective brain cholecystokinin (CCK-B) and gastrin receptor antagonist radioligand
CHANG, R. S. L, CHEN, T. B, BOCK, M. G, FREIDINGER, R. M, CHEN, R, ROSEGAY, A, LOTTI, V. J
Published in Molecular pharmacology (01.06.1989)
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Published in Molecular pharmacology (01.06.1989)
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HIV-1 protease specificity of peptide cleavage is sufficient for processing of gag and pol polyproteins
Darke, Paul L., Nutt, Ruth F., Brady, Stephen F., Garsky, Victor M., Ciccarone, Terrence M., Leu, Chih-Tai, Lumma, Patricia K., Freidinger, Roger M., Veber, Daniel F., Sigal, Irving S.
Published in Biochemical and biophysical research communications (14.10.1988)
Published in Biochemical and biophysical research communications (14.10.1988)
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Journal Article
Synthesis and Biological Activities of Potent Peptidomimetics Selective for Somatostatin Receptor Subtype 2
Yang, Lihu, Berk, Scott C., Rohrer, Susan P., Mosley, Ralph T., Guo, Liangqin, Underwood, Dennis J., Arison, Byron H., Birzin, Elizabeth T., Hayes, Edward C., Mitra, Sudha W., Parmar, Rupa M., Cheng, Kang, Wu, Tsuei-Ju, Butler, Bridgette S., Foor, Forrest, Pasternak, Alexander, Pan, Yanping, Silva, Maria, Freidinger, Roger M., Smith, Roy G., Chapman, Kevin, Schaeffer, James M., Patchett, Arthur A.
Published in Proceedings of the National Academy of Sciences - PNAS (01.09.1998)
Published in Proceedings of the National Academy of Sciences - PNAS (01.09.1998)
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Chemical Synthesis of Echistatin, a Potent Inhibitor of Platelet Aggregation from Echis carinatus: Synthesis and Biological Activity of Selected Analogs
Garsky, Victor M., Lumma, Patricia K., Freidinger, Roger M., Pitzenberger, Steven M., Randall, William C., Veber, Daniel F., Gould, Robert J., Friedman, Paul A.
Published in Proceedings of the National Academy of Sciences - PNAS (01.06.1989)
Published in Proceedings of the National Academy of Sciences - PNAS (01.06.1989)
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Journal Article
Nonpeptide oxytocin antagonists: Analogs of L-371,257 with improved potency
Williams, Peter D., Bock, Mark G., Evans, Ben E., Freidinger, Roger M., Gallicchio, Steven N., Guidotti, Maribeth T., Jacobson, Marlene A., Kuo, Michelle S., Levy, Michelle R., Lis, Edward V., Michelson, Stuart R., Pawluczyk, Joseph M., Perlow, Debra S., Pettibone, Douglas J., Quigley, Amy G., Reiss, Duane R., Salvatore, Christopher, Stauffer, Kenneth J., Woyden, Carla J.
Published in Bioorganic & medicinal chemistry letters (03.05.1999)
Published in Bioorganic & medicinal chemistry letters (03.05.1999)
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Journal Article
Progress towards the development of a HIV-1 gp41-directed vaccine
McGaughey, Georgia B, Barbato, Gaetano, Bianchi, Elisabetta, Freidinger, Roger M, Garsky, Victor M, Hurni, William M, Joyce, Joseph G, Liang, Xiaoping, Miller, Michael D, Pessi, Antonello, Shiver, John W, Bogusky, Michael J
Published in Current HIV research (01.04.2004)
Published in Current HIV research (01.04.2004)
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Identification of a Series of CCK-2 Receptor Nonpeptide Agonists: Sensitivity to Stereochemistry and a Receptor Point Mutation
Kopin, Alan S., McBride, Edward W., Chen, Ci, Freidinger, Roger M., Chen, Duan, Zhao, Chun-Mei, Beinborn, Martin
Published in Proceedings of the National Academy of Sciences - PNAS (29.04.2003)
Published in Proceedings of the National Academy of Sciences - PNAS (29.04.2003)
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Identification of an orally active, nonpeptidyl oxytocin antagonist
PETTIBONE, D. J, CLINESCHMIDT, B. V, HALUSKA, G. J, NOVY, M. J, LOWENSOHN, R. I, KISHEL, M. T, LIS, E. V, REISS, D. R, WOYDEN, C. J, EVANS, B. E, FREIDINGER, R. M, VEBER, D. F, COOK, M. J
Published in The Journal of pharmacology and experimental therapeutics (01.01.1993)
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Published in The Journal of pharmacology and experimental therapeutics (01.01.1993)
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Spontaneous Assembly of Soda Straws
Campbell, D. J, Freidinger, E. R, Hastings, J. M, Querns, M. K
Published in Journal of chemical education (01.02.2002)
Published in Journal of chemical education (01.02.2002)
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