SUBSTITUTED TRIAZOLE AND IMIDAZOLE DERIVATIVES AS GAMMA SECRETASE MODULATORS
SVEN FRANCISCUS ANNA VAN BRANDT, WU TONGFEI, MICHEL SURKYN, FREDERIK JAN RITA ROMBOUTS, FRANCOIS PAUL BISCHOFF, GARRETT BERLOND MINNE, SERGE MARIA ALOYSIUS PIETERS, HENRICUS JACOBUS MARIA GIJSEN, DANIEL OEHLRICH, ADRIANA INGRID VELTER, MICHEL ANNA JOZEF DE CLEYN, DIDIER JEAN-CLAUDE BERTHELOT
Year of Publication 16.07.2015
Get full text
Year of Publication 16.07.2015
Patent
N-LINKED MACROCYCLIC 4-(PYRAZOL-5-YL)-INDOLE DERIVATIVES AS INHIBITORS OF MCL-1
VELTER, Adriana-Ingrid, ROMBOUTS, Frederik, Jan, Rita, PESCHIULLI, Aldo
Year of Publication 12.06.2024
Get full text
Year of Publication 12.06.2024
Patent
N-LINKED MACROCYCLIC 4-(PYRAZOL-5-YL)-INDOLE DERIVATIVES AS INHIBITORS OF MCL-1
VELTER, Adriana-Ingrid, ROMBOUTS, Frederik, Jan, Rita, PESCHIULLI, Aldo
Year of Publication 12.06.2024
Get full text
Year of Publication 12.06.2024
Patent
N-LINKED MACROCYCLIC 4-(PYRAZOL-5-YL)-INDOLE DERIVATIVES AS INHIBITORS OF MCL-1
ROMBOUTS, Frederik Jan Rita, VELTER, Adriana-Ingrid, PESCHIULLI, Aldo
Year of Publication 27.07.2023
Get full text
Year of Publication 27.07.2023
Patent
N-LINKED MACROCYCLIC 4-(PYRAZOL-5-YL)-INDOLE DERIVATIVES AS INHIBITORS OF MCL-1
VELTER, Adriana-Ingrid, ROMBOUTS, Frederik, Jan, Rita, PESCHIULLI, Aldo
Year of Publication 26.04.2023
Get full text
Year of Publication 26.04.2023
Patent
N-linked macrocyclic 4-(pyrazol-5-yl)-indole derivatives as inhibitors of MCL-1
ROMBOUTS, Frederik Jan Rita, VELTER, Adriana-Ingrid, PESCHIULLI, Aldo
Year of Publication 23.02.2023
Get full text
Year of Publication 23.02.2023
Patent
MACROCYLIC SULFONYL DERIVATIVES MCL-1 INHIBITORS
ROMBOUTS, Frederik Jan Rita, De BOECK, Benoit Christian Albert Ghislain
Year of Publication 26.01.2023
Get full text
Year of Publication 26.01.2023
Patent
MACROCYCLIC 1,3-BRIDGED 6-CHLORO-7-PYRAZOL-4-YL-1 H-INDOLE-2-CARBOXYLATE AND 6-CHLORO-7-PYRIMIDIN-5-YL-1H-INDOLE-2-CARBOXYLATE DERIVATIVES AS MCL-1 INHIBITORS FOR THE TREATMENT OF CANCER
ROMBOUTS, Frederik Jan Rita, DE BOECK, Benoît Christian Albert Ghislain, JERHAOUI, Soufyan
Year of Publication 13.06.2024
Get full text
Year of Publication 13.06.2024
Patent
MACROCYCLIC BRANCHED 3-FLUORO-BUT-3-ENAMIDES AS INHIBITORS OF MCL-1
ROMBOUTS, Frederik Jan Rita, HSIAO, Meng-Yang, JOUFFROY, Matthieu Dominique, JERHAOUI, Soufyan, SURKYN, Michel
Year of Publication 14.03.2024
Get full text
Year of Publication 14.03.2024
Patent
MACROCYCLIC 1,3-BRIDGED 6-CHLORO-7-PYRAZOL-4-YL-1H-INDOLE-2-CARBOXYLATE AND 6-CHLORO-7-PYRIMIDIN-5-YL-1H-INDOLE-2-CARBOXYLATE DERIVATIVES AS MCL-1 INHIBITORS FOR THE TREATMENT OF CANCER
ROMBOUTS, Frederik, Jan, Rita, JERHAOUI, Soufyan, DE BOECK, Benoît, Christian, Albert, Ghislain
Year of Publication 20.12.2023
Get full text
Year of Publication 20.12.2023
Patent
MACROCYCLIC BRANCHED 3-FLUORO-BUT-3-ENAMIDES AS INHIBITORS OF MCL-1
HSIAO, Meng-Yang, JOUFFROY, Matthieu, Dominique, ROMBOUTS, Frederik, Jan, Rita, JERHAOUI, Soufyan, SURKYN, Michel
Year of Publication 25.10.2023
Get full text
Year of Publication 25.10.2023
Patent