Discovery of (3-(4-(2-Oxa-6-azaspiro[3.3]heptan-6-ylmethyl)phenoxy)azetidin-1-yl)(5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-yl)methanone (AZD1979), a Melanin Concentrating Hormone Receptor 1 (MCHr1) Antagonist with Favorable Physicochemical Properties
Johansson, Anders, Löfberg, Christian, Antonsson, Madeleine, von Unge, Sverker, Hayes, Martin A, Judkins, Robert, Ploj, Karolina, Benthem, Lambertus, Lindén, Daniel, Brodin, Peter, Wennerberg, Marie, Fredenwall, Marléne, Li, Lanna, Persson, Joachim, Bergman, Rolf, Pettersen, Anna, Gennemark, Peter, Hogner, Anders
Published in Journal of medicinal chemistry (24.03.2016)
Published in Journal of medicinal chemistry (24.03.2016)
Get full text
Journal Article
Oxetane Substrates of Human Microsomal Epoxide Hydrolase
Toselli, Francesca, Fredenwall, Marlene, Svensson, Peder, Li, Xue-Qing, Johansson, Anders, Weidolf, Lars, Hayes, Martin A
Published in Drug metabolism and disposition (01.08.2017)
Published in Drug metabolism and disposition (01.08.2017)
Get full text
Journal Article
Structure‐Based Drug Design of Mineralocorticoid Receptor Antagonists to Explore Oxosteroid Receptor Selectivity
Nordqvist, Anneli, O'Mahony, Gavin, Fridén‐Saxin, Maria, Fredenwall, Marlene, Hogner, Anders, Granberg, Kenneth L., Aagaard, Anna, Bäckström, Stefan, Gunnarsson, Anders, Kaminski, Tim, Xue, Yafeng, Dellsén, Anita, Hansson, Eva, Hansson, Pia, Ivarsson, Ida, Karlsson, Ulla, Bamberg, Krister, Hermansson, Majlis, Georgsson, Jennie, Lindmark, Bo, Edman, Karl
Published in ChemMedChem (05.01.2017)
Published in ChemMedChem (05.01.2017)
Get full text
Journal Article
agentes terapêuticos 976
Per oskar Sverker Von Unge, Robert Anderw Judkins, Lanna Li, Susanne Doris Margit Bökman-Winiwarter, Anders Carls Hogner, Marlene Fredenwall, Björn Christian Ingvar Löfberg
Year of Publication 24.09.2019
Get full text
Year of Publication 24.09.2019
Patent
(3-(4-(aminomethyl)phenoxy or phenylthio)azetidin-1-yl)(5-phenyl-1,3,4-oxadiazol-2-yl)methanone compounds
JUDKINS ROBERT ANDREW, BOEKMAN-WINIWARTER SUSANNE DORIS MARGIT, JOHANSSON LARS ANDERS MIKAEL, VON UNGE SVERKER, LOEFBERG BJOERN CHRISTIAN INGVAR, LI LANNA, HOGNER CARL ANDERS, FREDENWALL MARLENE
Year of Publication 01.10.2013
Get full text
Year of Publication 01.10.2013
Patent