Structure−Activity Relationship Study on Anti-HIV 6-Desfluoroquinolones
Tabarrini, Oriana, Massari, Serena, Daelemans, Dirk, Stevens, Miguel, Manfroni, Giuseppe, Sabatini, Stefano, Balzarini, Jan, Cecchetti, Violetta, Pannecouque, Christophe, Fravolini, Arnaldo
Published in Journal of medicinal chemistry (11.09.2008)
Published in Journal of medicinal chemistry (11.09.2008)
Get full text
Journal Article
New Anti-Human Immunodeficiency Virus Type 1 6-Aminoquinolones: Mechanism of Action
PAROLIN, Cristina, GATTO, Barbara, DEL VECCHIO, Claudia, PECERE, Teresa, TRAMONTANO, Enzo, CECCHETTI, Violetta, FRAVOLINI, Arnaldo, MASIERO, Sara, PALUMBO, Manlio, PALU, Giorgio
Published in Antimicrobial Agents and Chemotherapy (01.03.2003)
Published in Antimicrobial Agents and Chemotherapy (01.03.2003)
Get full text
Journal Article
Novel In Vivo Model for the Study of Human Immunodeficiency Virus Type 1 Transcription Inhibitors: Evaluation of New 6-Desfluoroquinolone Derivatives
STEVENS, Miguel, POLLICITA, Michela, SCHOLS, Dominique, BALZARINI, Jan, PANNECOUQUE, Christophe, VERBEKEN, Erik, TABARRINI, Oriana, CECCHETTI, Violetta, AQUARO, Stefano, PERNO, Carlo Federico, FRAVOLINI, Arnaldo, DE CLERCQ, Erik
Published in Antimicrobial Agents and Chemotherapy (01.04.2007)
Published in Antimicrobial Agents and Chemotherapy (01.04.2007)
Get full text
Journal Article
2‐Phenylquinolones as Inhibitors of the HIV‐1 Tat–TAR Interaction
Gatto, Barbara, Tabarrini, Oriana, Massari, Serena, Giaretta, Giulia, Sabatini, Stefano, Del Vecchio, Claudia, Parolin, Cristina, Fravolini, Arnaldo, Palumbo, Manlio, Cecchetti, Violetta
Published in ChemMedChem (08.06.2009)
Published in ChemMedChem (08.06.2009)
Get full text
Journal Article
Inhibition of Human Immunodeficiency Virus Type 1 Tat-trans-Activation-Responsive Region Interaction by an Antiviral Quinolone Derivative
RICHTER, Sara, PAROLIN, Cristina, GATTO, Barbara, DEL VECCHIO, Claudia, BROCCA-COFANO, Egidio, FRAVOLINI, Arnaldo, PALU, Giorgio, PALUMBO, Manlio
Published in Antimicrobial Agents and Chemotherapy (01.05.2004)
Published in Antimicrobial Agents and Chemotherapy (01.05.2004)
Get full text
Journal Article
From Phenothiazine to 3-Phenyl-1,4-benzothiazine Derivatives as Inhibitors of the Staphylococcus aureus NorA Multidrug Efflux Pump
Sabatini, Stefano, Kaatz, Glenn W, Rossolini, Gian Maria, Brandini, David, Fravolini, Arnaldo
Published in Journal of medicinal chemistry (24.07.2008)
Published in Journal of medicinal chemistry (24.07.2008)
Get full text
Journal Article
Discovery of Novel Inhibitors of the NorA Multidrug Transporter of Staphylococcus aureus
Brincat, Jean Pierre, Carosati, Emanuele, Sabatini, Stefano, Manfroni, Giuseppe, Fravolini, Arnaldo, Raygada, Jose L, Patel, Diixa, Kaatz, Glenn W, Cruciani, Gabriele
Published in Journal of medicinal chemistry (13.01.2011)
Published in Journal of medicinal chemistry (13.01.2011)
Get full text
Journal Article
Inhibition of Subgenomic Hepatitis C Virus RNA Replication by Acridone Derivatives: Identification of an NS3 Helicase Inhibitor
Manfroni, Giuseppe, Paeshuyse, Jan, Massari, Serena, Zanoli, Samantha, Gatto, Barbara, Maga, Giovanni, Tabarrini, Oriana, Cecchetti, Violetta, Fravolini, Arnaldo, Neyts, Johan
Published in Journal of medicinal chemistry (28.05.2009)
Published in Journal of medicinal chemistry (28.05.2009)
Get full text
Journal Article
From 6-Aminoquinolone Antibacterials to 6-Amino-7-thiopyranopyridinylquinolone Ethyl Esters as Inhibitors of Staphylococcus aureus Multidrug Efflux Pumps
Pieroni, Marco, Dimovska, Mirjana, Brincat, Jean Pierre, Sabatini, Stefano, Carosati, Emanuele, Massari, Serena, Kaatz, Glenn W, Fravolini, Arnaldo
Published in Journal of medicinal chemistry (10.06.2010)
Published in Journal of medicinal chemistry (10.06.2010)
Get full text
Journal Article
Synthesis and Anti-BVDV Activity of Acridones As New Potential Antiviral Agents
Tabarrini, Oriana, Manfroni, Giuseppe, Fravolini, Arnaldo, Cecchetti, Violetta, Sabatini, Stefano, De Clercq, Erik, Rozenski, Jef, Canard, Bruno, Dutartre, Hélène, Paeshuyse, Jan, Neyts, Johan
Published in Journal of medicinal chemistry (20.04.2006)
Published in Journal of medicinal chemistry (20.04.2006)
Get full text
Journal Article
A Pharmacophore Hypothesis for P-Glycoprotein Substrate Recognition Using GRIND-Based 3D-QSAR
Cianchetta, Giovanni, Singleton, Robert W, Zhang, Meng, Wildgoose, Marianne, Giesing, Dennis, Fravolini, Arnaldo, Cruciani, Gabriele, Vaz, Roy J
Published in Journal of medicinal chemistry (21.04.2005)
Published in Journal of medicinal chemistry (21.04.2005)
Get full text
Journal Article
Predictive models for hERG potassium channel blockers
Cianchetta, Giovanni, Li, Yi, Kang, Jiesheng, Rampe, David, Fravolini, Arnaldo, Cruciani, Gabriele, Vaz, Roy J.
Published in Bioorganic & medicinal chemistry letters (01.08.2005)
Published in Bioorganic & medicinal chemistry letters (01.08.2005)
Get full text
Journal Article
Synthesis and biological evaluation of 2-phenylquinolones targeted at Tat/TAR recognition
Manfroni, Giuseppe, Gatto, Barbara, Tabarrini, Oriana, Sabatini, Stefano, Cecchetti, Violetta, Giaretta, Giulia, Parolin, Cristina, Del Vecchio, Claudia, Calistri, Arianna, Palumbo, Manlio, Fravolini, Arnaldo
Published in Bioorganic & medicinal chemistry letters (01.02.2009)
Published in Bioorganic & medicinal chemistry letters (01.02.2009)
Get full text
Journal Article
Cell-dependent interference of a series of new 6-aminoquinolone derivatives with viral (HIV/CMV) transactivation
Stevens, Miguel, Balzarini, Jan, Tabarrini, Oriana, Andrei, Graciela, Snoeck, Robert, Cecchetti, Violetta, Fravolini, Arnaldo, De Clercq, Erik, Pannecouque, Christophe
Published in Journal of antimicrobial chemotherapy (01.11.2005)
Published in Journal of antimicrobial chemotherapy (01.11.2005)
Get full text
Journal Article
Correction to From 6-Aminoquinolone Antibacterials to 6-Amino-7-thiopyranopyridinylquinolone Ethyl Esters as Inhibitors of Staphylococcus aureus Multidrug Efflux Pumps
Pieroni, Marco, Dimovska, Mirjana, Brincat, Jean Pierre, Sabatini, Stefano, Carosati, Emanuele, Massari, Serena, Kaatz, Glenn W, Fravolini, Arnaldo
Published in Journal of medicinal chemistry (10.03.2011)
Published in Journal of medicinal chemistry (10.03.2011)
Get full text
Journal Article
Highly Potent 1,4-Benzothiazine Derivatives as KATP-Channel Openers
Cecchetti, Violetta, Calderone, Vincenzo, Tabarrini, Oriana, Sabatini, Stefano, Filipponi, Enrica, Testai, Lara, Spogli, Roberto, Martinotti, Enrica, Fravolini, Arnaldo
Published in Journal of medicinal chemistry (14.08.2003)
Published in Journal of medicinal chemistry (14.08.2003)
Get full text
Journal Article
Highly potent 1,4-benzothiazine derivatives as K-ATP-channel openers
Cecchetti, Calderone, Tabarrini, O, Sabatini, S, Filipponi, E, Testai, L, Spogli, R, Martinotti, E, Fravolini, A
Published in Journal of medicinal chemistry (14.08.2003)
Published in Journal of medicinal chemistry (14.08.2003)
Get full text
Journal Article
Structure Modifications of 6-Aminoquinolones with Potent Anti-HIV Activity
Tabarrini, Oriana, Stevens, Miguel, Cecchetti, Violetta, Sabatini, Stefano, Dell'Uomo, Micaela, Manfroni, Giuseppe, Palumbo, Manlio, Pannecouque, Christophe, De Clercq, Erik, Fravolini, Arnaldo
Published in Journal of medicinal chemistry (21.10.2004)
Published in Journal of medicinal chemistry (21.10.2004)
Get full text
Journal Article
6-Aminoquinolones as New Potential Anti-HIV Agents
Cecchetti, Violetta, Parolin, Cristina, Moro, Stefano, Pecere, Teresa, Filipponi, Enrica, Calistri, Arianna, Tabarrini, Oriana, Gatto, Barbara, Palumbo, Manlio, Fravolini, Arnaldo
Published in Journal of medicinal chemistry (05.10.2000)
Published in Journal of medicinal chemistry (05.10.2000)
Get full text
Journal Article
Antiviral 6-amino-quinolones: Molecular basis for potency and selectivity
Richter, Sara N., Gatto, Barbara, Tabarrini, Oriana, Fravolini, Arnaldo, Palumbo, Manlio
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
Get full text
Journal Article