Atypical teratoid/rhabdoid tumoroids reveal subgroup-specific drug vulnerabilities
Paassen, Irene, Williams, Justin, Ríos Arceo, Carla, Ringnalda, Femke, Mercer, Kimberly Shea, Buhl, Juliane L, Moreno, Natalia, Federico, Aniello, Franke, Niels E, Kranendonk, Mariette, Upadhyaya, Santhosh A, Kerl, Kornelius, van de Wetering, Marc, Clevers, Hans, Kool, Marcel, Hoving, Eelco W, Roussel, Martine F, Drost, Jarno
Published in Oncogene (12.05.2023)
Published in Oncogene (12.05.2023)
Get full text
Journal Article
(Immuno)proteasomes as therapeutic target in acute leukemia
Cloos, Jacqueline, Roeten, Margot SF, Franke, Niels E, van Meerloo, Johan, Zweegman, Sonja, Kaspers, Gertjan JL, Jansen, Gerrit
Published in Cancer and metastasis reviews (01.12.2017)
Published in Cancer and metastasis reviews (01.12.2017)
Get full text
Journal Article
Higher ratio immune versus constitutive proteasome level as novel indicator of sensitivity of pediatric acute leukemia cells to proteasome inhibitors
Niewerth, Denise, Franke, Niels E, Jansen, Gerrit, Assaraf, Yehuda G, van Meerloo, Johan, Kirk, Christopher J, Degenhardt, Jeremiah, Anderl, Janet, Schimmer, Aaron D, Zweegman, Sonja, de Haas, Valerie, Horton, Terzah M, Kaspers, Gertjan J L, Cloos, Jacqueline
Published in Haematologica (Roma) (01.12.2013)
Published in Haematologica (Roma) (01.12.2013)
Get full text
Journal Article
Gemcitabine therapeutically disrupts essential SIRT1-mediated p53 repression in atypical teratoid/rhabdoid tumors
Metselaar, Dennis S., Meel, Michaël H., Goulding, Joshua R., du Chatinier, Aimeé, Rigamonti, Leyla, Waranecki, Piotr, Geisemeyer, Neal, de Gooijer, Mark C., Breur, Marjolein, Koster, Jan, Veldhuijzen van Zanten, Sophie E.M., Bugiani, Marianna, Franke, Niels E., Reddy, Alyssa, Wesseling, Pieter, Kaspers, Gertjan J.L., Hulleman, Esther
Published in Cell reports. Medicine (17.09.2024)
Published in Cell reports. Medicine (17.09.2024)
Get full text
Journal Article
Effect of Noncompetitive Proteasome Inhibition on Bortezomib Resistance
Li, Xiaoming, Wood, Tabitha E., Sprangers, Remco, Jansen, Gerrit, Franke, Niels E., Mao, Xinliang, Wang, Xiaoming, Zhang, Yi, Verbrugge, Sue Ellen, Adomat, Hans, Li, Zhi Hua, Trudel, Suzanne, Chen, Christine, Religa, Tomasz L., Jamal, Nazir, Messner, Hans, Cloos, Jacqueline, Rose, David R., Navon, Ami, Guns, Emma, Batey, Robert A., Kay, Lewis E., Schimmer, Aaron D.
Published in JNCI : Journal of the National Cancer Institute (21.07.2010)
Published in JNCI : Journal of the National Cancer Institute (21.07.2010)
Get full text
Journal Article
Exocytosis of polyubiquitinated proteins in bortezomib-resistant leukemia cells: a role for MARCKS in acquired resistance to proteasome inhibitors
Franke, Niels E, Kaspers, Gertjan L, Assaraf, Yehuda G, van Meerloo, Johan, Niewerth, Denise, Kessler, Floortje L, Poddighe, Pino J, Kole, Jeroen, Smeets, Serge J, Ylstra, Bauke, Bi, Chonglei, Chng, Wee Joo, Horton, Terzah M, Menezes, Rene X, Musters, Renée J P, Zweegman, Sonja, Jansen, Gerrit, Cloos, Jacqueline
Published in Oncotarget (15.11.2016)
Published in Oncotarget (15.11.2016)
Get full text
Journal Article
LacdiNAc-Glycans Constitute a Parasite Pattern for Galectin-3-Mediated Immune Recognition
van den Berg, Timo K, Honing, Henk, Franke, Niels, van Remoortere, Alexandra, Schiphorst, Wietske E. C. M, Liu, Fu-Tong, Deelder, Andre M, Cummings, Richard D, Hokke, Cornelis H, van Die, Irma
Published in The Journal of immunology (1950) (01.08.2004)
Published in The Journal of immunology (1950) (01.08.2004)
Get full text
Journal Article
Trabectedin (ET-743, Yondelis) is a substrate for P-glycoprotein, but only high expression of P-glycoprotein confers the multidrug resistance phenotype
Beumer, Jan-Hendrik, Buckle, Tessa, Ouwehand, Mariet, Franke, Niels E F, Lopez-Lazaro, Luis, Schellens, Jan H M, Beijnen, Jos H, van Tellingen, Olaf
Published in Investigational new drugs (01.02.2007)
Published in Investigational new drugs (01.02.2007)
Get full text
Journal Article
Molecular basis of bortezomib resistance: proteasome subunit β5 (PSMB5) gene mutation and overexpression of PSMB5 protein
Oerlemans, Ruud, Franke, Niels E., Assaraf, Yehuda G., Cloos, Jacqueline, van Zantwijk, Ina, Berkers, Celia R., Scheffer, George L., Debipersad, Kabir, Vojtekova, Katharina, Lemos, Clara, van der Heijden, Joost W., Ylstra, Bauke, Peters, Godefridus J., Kaspers, Gertjan L., Dijkmans, Ben A.C., Scheper, Rik J., Jansen, Gerrit
Published in Blood (15.09.2008)
Published in Blood (15.09.2008)
Get full text
Journal Article
Marcks Marks Resistance to Proteasome Inhibitors: Exocytosis of Polyubiquitinated Proteins in Bortezomib-Resistant Leukemia Cells
Franke, Niels, Kaspers, Gertjan J.L., Assaraf, Yehuda G, Van Meerloo, Johan, Niewerth, Denise, Horton, Terzah M., Chng, Wee Joo, Bi, Chonglei, Menezes, Rene X., Musters, Renée J., Poddighe, Pino J., Kessler, Floortje, Smeets, Serge, Ylstra, Bauke, Zweegman, Sonja, Jansen, Gerrit, Cloos, Jacqueline
Published in Blood (03.12.2015)
Published in Blood (03.12.2015)
Get full text
Journal Article
Interferon-γ-Induced Upregulation of Immunoproteasome Subunit Assembly Overcomes Bortezomib Resistance of Leukemia Cell Lines Harbouring Bortezomib-Induced Mutations in Constitutive PSMB5
Niewerth, Denise, Franke, Niels, Jansen, Gerrit, Assaraf, Yehuda, van Meerloo, Johan, Kirk, Christopher J, Zweegman, Sonja, Kaspers, Gertjan J.L., Cloos, Jacqueline
Published in Blood (16.11.2012)
Published in Blood (16.11.2012)
Get full text
Journal Article
Sensitivity of Pediatric Acute Leukemia Cells to Bortezomib and Epoxyketone-Based Proteasome Inhibitors: Correlations with Proteasome Subunit Expression
Niewerth, Denise, Franke, Niels, Jansen, Gerrit, van Meerloo, Johan, Assaraf, Yehuda, Kirk, Christopher J, Chan, Elena T, Zweegman, Sonja, Kaspers, Gertjan J., Cloos, Jacqueline
Published in Blood (18.11.2011)
Published in Blood (18.11.2011)
Get full text
Journal Article
Abstract A27: Chronic exposure of malignant hematological cell lines to bortezomib induces de novo hot spot mutations in the PSMB5 gene
Franke, Niels, Niewerth, Denise, van Meerloo, Johan, Vojtekova, Katarina, Verbrugge, Sue Ellen, Schimmer, Aaron, Kaspers, Gertjan, Jansen, Gerrit, Cloos, Jacqueline
Published in Clinical cancer research (01.04.2010)
Published in Clinical cancer research (01.04.2010)
Get full text
Journal Article
Induced Hypotension: Action of Sodium Nitroprusside and Nitroglycerin on the Microcirculation
Endrich, Bernhard, Franke, Niels, Peter, Klaus, Messmer, Konrad
Published in Anesthesiology (Philadelphia) (01.05.1987)
Published in Anesthesiology (Philadelphia) (01.05.1987)
Get full text
Journal Article
Acquisition of Mutations in the PSMB5 Gene during Chronic Exposure of Human Acute Lymphoblastic Leukemia CCRF-CEM Cells to the Proteasome Inhibitor Bortezomib
Franke, Niels E, Oerlemans, Ruud, van Zantwijk, Ina, Vojtekova, Katarina, Kaspers, Gertjan L, Jansen, Gerrit, Cloos, Jacqueline
Published in Blood (16.11.2008)
Published in Blood (16.11.2008)
Get full text
Journal Article
The Novel Proteasome Inhibitor 5-Amino-8-Hydroxyquinole (5AHQ) Overcomes Bortezomib Resistance in Malignant Hematological Cell Line Models Harboring Mutations in the PSMB5 Gene
Franke, Niels E, van Meerloo, Johan, Slot, Linda, Li, Xiaoming, Wood, Tabitha E, Vojtekova, Katarina, Verbrugge, Sue Ellen, Kaspers, Gertjan, Batey, Robert A., Schimmer, Aaron D., Jansen, Gerrit, Cloos, Jacqueline
Published in Blood (20.11.2009)
Published in Blood (20.11.2009)
Get full text
Journal Article
Acquired Resistance to Bortezomib in Human RPMI-8226 Multiple Myeloma Cells: Molecular Characterization, Cross-Resistance with Other Proteasome Inhibitors but Marked Sensitization to Glucocorticoids
Franke, Niels E, Kaspers, Gertjan L, van den Berg, Nynke, van Zantwijk, Ina, Vojtekova, Katarina, Yaqub, Uzma, Smeets, Serge, Ylstra, Bauke, Zweegman, Sonja, Jansen, Gerrit, Cloos, Jacqueline
Published in Blood (16.11.2008)
Published in Blood (16.11.2008)
Get full text
Journal Article
Molecular Mechanisms of Bortezomib Resistance in Acute Lymphoblastic Leukemia Cells in Comparison with Multiple Myeloma Cells
Franke, Niels E., Oerlemans, Ruud, Zweegman, Sonja, van Zantwijk, Ina, Kaspers, Gertjan J., Jansen, Gerrit, Cloos, Jacqueline
Published in Blood (16.11.2007)
Published in Blood (16.11.2007)
Get full text
Journal Article