Intrinsic Property Forecast Index (iPFI) as a Rule of Thumb for Medicinal Chemists to Remove a Phototoxicity Liability
Fournier, Jean-François, Bouix-Peter, Claire, Duvert, Denis, Luzy, Anne-Pascale, Ouvry, Gilles
Published in Journal of medicinal chemistry (12.04.2018)
Published in Journal of medicinal chemistry (12.04.2018)
Get full text
Journal Article
Rational Drug Design of Topically Administered Caspase 1 Inhibitors for the Treatment of Inflammatory Acne
Fournier, Jean-François, Clary, Laurence, Chambon, Sandrine, Dumais, Laurence, Harris, Craig Steven, Millois, Corinne, Pierre, Romain, Talano, Sandrine, Thoreau, Étienne, Aubert, Jérome, Aurelly, Michèle, Bouix-Peter, Claire, Brethon, Anne, Chantalat, Laurent, Christin, Olivier, Comino, Catherine, El-Bazbouz, Ghizlane, Ghilini, Anne-Laurence, Isabet, Tatiana, Lardy, Claude, Luzy, Anne-Pascale, Mathieu, Céline, Mebrouk, Kenny, Orfila, Danielle, Pascau, Jonathan, Reverse, Kevin, Roche, Didier, Rodeschini, Vincent, Hennequin, Laurent François
Published in Journal of medicinal chemistry (10.05.2018)
Published in Journal of medicinal chemistry (10.05.2018)
Get full text
Journal Article
New Caspase-1 inhibitor by scaffold hopping into bio-inspired 3D-fragment space
Brethon, Anne, Chantalat, Laurent, Christin, Olivier, Clary, Laurence, Fournier, Jean-François, Gastreich, Marcus, Harris, Craig S., Isabet, Tatiana, Pascau, Jonathan, Thoreau, Etienne, Roche, Didier, Rodeschini, Vincent
Published in Bioorganic & medicinal chemistry letters (15.12.2017)
Published in Bioorganic & medicinal chemistry letters (15.12.2017)
Get full text
Journal Article
Squaramides as novel class I and IIB histone deacetylase inhibitors for topical treatment of cutaneous t-cell lymphoma
Fournier, Jean-François, Bhurruth-Alcor, Yushma, Musicki, Branislav, Aubert, Jérome, Aurelly, Michèle, Bouix-Peter, Claire, Bouquet, Karinne, Chantalat, Laurent, Delorme, Marion, Drean, Bénédicte, Duvert, Gwenaelle, Fleury-Bregeot, Nicolas, Gauthier, Blanche, Grisendi, Karine, Harris, Craig S., Hennequin, Laurent F., Isabet, Tatiana, Joly, Florence, Lafitte, Guillaume, Millois, Corinne, Morgentin, Rémy, Pascau, Jonathan, Piwnica, David, Rival, Yves, Soulet, Catherine, Thoreau, Étienne, Tomas, Loïc
Published in Bioorganic & medicinal chemistry letters (15.09.2018)
Published in Bioorganic & medicinal chemistry letters (15.09.2018)
Get full text
Journal Article
Synthesis and stability evaluation of novel peptidomimetic Caspase-1 inhibitors for topical application
Chambon, Sandrine, Talano, Sandrine, Millois, Corinne, Dumais, Laurence, Pierre, Romain, Tomas, Loic, Mathieu, Céline, Ghilini, Anne-Laurence, Vanthuyne, Nicolas, Reverse, Kevin, Brethon, Anne, Rodeschini, Vincent, Comino, Catherine, Mouis, Grégoire, El-Bazbouz, Ghizlane, Clary, Laurence, Fournier, Jean-François, Bouix-Peter, Claire, Harris, Craig S., Hennequin, Laurent F.
Published in Tetrahedron (13.09.2018)
Published in Tetrahedron (13.09.2018)
Get full text
Journal Article
N-3 alkylation of uracils with unprotected amino alcohols using the Mitsunobu reaction
Lafitte, Guillaume, Beillard, Audrey, Chambon, Sandrine, Soulet, Catherine, Dumais, Laurence, Mouis, Grégoire, Fournier, Jean-François, Clary, Laurence, Bouix-Peter, Claire, Tomas, Loic, Harris, Craig S.
Published in Tetrahedron letters (17.01.2018)
Published in Tetrahedron letters (17.01.2018)
Get full text
Journal Article
A convenient one-pot synthesis of boroxoles from diboronic acid
Lafitte, Guillaume, Kunihiro, Kana, Bonneaud, Céline, Dréan, Bénédicte, Gaigne, Frédéric, Parnet, Véronique, Pierre, Romain, Raffin, Catherine, Vatinel, Rodolphe, Fournier, Jean-François, Musicki, Branislav, Ouvry, Gilles, Bouix-Peter, Claire, Tomas, Loic, Harris, Craig S.
Published in Tetrahedron letters (27.09.2017)
Published in Tetrahedron letters (27.09.2017)
Get full text
Journal Article
Discovery and Characterization of CD12681, a Potent RORγ Inverse Agonist, Preclinical Candidate for the Topical Treatment of Psoriasis
Ouvry, Gilles, Atrux‐Tallau, Nicolas, Bihl, Franck, Bondu, Aline, Bouix‐Peter, Claire, Carlavan, Isabelle, Christin, Olivier, Cuadrado, Marie‐Josée, Defoin‐Platel, Claire, Deret, Sophie, Duvert, Denis, Feret, Christophe, Forissier, Mathieu, Fournier, Jean‐François, Froude, David, Hacini‐Rachinel, Fériel, Harris, Craig Steven, Hervouet, Catherine, Huguet, Hélène, Lafitte, Guillaume, Luzy, Anne‐Pascale, Musicki, Branislav, Orfila, Danielle, Ozello, Benjamin, Pascau, Coralie, Pascau, Jonathan, Parnet, Véronique, Peluchon, Guillaume, Pierre, Romain, Piwnica, David, Raffin, Catherine, Rossio, Patricia, Spiesse, Delphine, Taquet, Nathalie, Thoreau, Etienne, Vatinel, Rodolphe, Vial, Emmanuel, Hennequin, Laurent François
Published in ChemMedChem (20.02.2018)
Published in ChemMedChem (20.02.2018)
Get full text
Journal Article
An efficient multi-component synthesis of N-1-alkylated 5-nitrouracils from α-amino acids
Boiteau, Jean-Guy, Bouix-Peter, Claire, Chambon, Sandrine, Clary, Laurence, Daver, Sebastien, Dumais, Laurence, Fournier, Jean-François, Harris, Craig S., Mebrouk, Kenny, Millois, Corinne, Pierre, Romain, Rodeville, Nicolas, Talano, Sandrine, Tomas, Loïc
Published in Tetrahedron letters (01.06.2016)
Published in Tetrahedron letters (01.06.2016)
Get full text
Journal Article
Occurrence of an Ascending Aorta Aneurysm 25 Years After Cure of a Tetrology of Fallot
Roux, Nicolas, Doguet, Fabien, Litzler, Pierre‐Yves, Tabley, Alfred, Adde, Jean‐Michel, Fournier, Jean‐François, Redonnet, Michel, Bizet, Catherine Nafeh, Bouchart, François, Hubscher, Catherine Haas, Bessou, Jean‐Paul
Published in Journal of cardiac surgery (01.03.2008)
Published in Journal of cardiac surgery (01.03.2008)
Get full text
Journal Article
An expedient synthesis of non-racemic N-alkylated pyrrolidin-2,5-diones and piperidin-2,6-diones as peptidomimetics
Brethon, Anne, Bouix-Peter, Claire, Clary, Laurence, Fournier, Jean-François, Harris, Craig S., Lardy, Claude, Roche, Didier, Rodeschini, Vincent, Talano, Sandrine
Published in Tetrahedron letters (28.12.2016)
Published in Tetrahedron letters (28.12.2016)
Get full text
Journal Article
Test-retest reliability of posture measurements in adolescents with idiopathic scoliosis
Heitz, Pierre-Henri, Aubin-Fournier, Jean-François, Parent, Éric, Fortin, Carole
Published in The spine journal (01.12.2018)
Published in The spine journal (01.12.2018)
Get full text
Journal Article
Applying the pro-drug approach to afford highly bioavailable antagonists of P2Y
Robichaud, Joël, Fournier, Jean-François, Gagné, Sébastien, Gauthier, Jacques Yves, Hamel, Martine, Han, Yongxin, Hénault, Martin, Kargman, Stacia, Levesque, Jean-François, Mamane, Yaël, Mancini, Joseph, Morin, Nicolas, Mulrooney, Erin, Wu, Jin, Black, W. Cameron
Published in Bioorganic & medicinal chemistry letters (15.07.2011)
Published in Bioorganic & medicinal chemistry letters (15.07.2011)
Get full text
Journal Article