Pain inhibition by blocking leukocytic and neuronal opioid peptidases in peripheral inflamed tissue
Schreiter, Anja, Gore, Carmen, Labuz, Dominika, Fournie-Zaluski, Marie-Claude, Roques, Bernard P, Stein, Christoph, Machelska, Halina
Published in The FASEB journal (01.12.2012)
Published in The FASEB journal (01.12.2012)
Get more information
Journal Article
Inhibiting the breakdown of endogenous opioids and cannabinoids to alleviate pain
Roques, Bernard P., Fournié-Zaluski, Marie-Claude, Wurm, Michel
Published in Nature reviews. Drug discovery (01.04.2012)
Published in Nature reviews. Drug discovery (01.04.2012)
Get full text
Journal Article
Intrarenal Aminopeptidase N Inhibition Augments Natriuretic Responses to Angiotensin III in Angiotensin Type 1 Receptor–Blocked Rats
Padia, Shetal H, Kemp, Brandon A, Howell, Nancy L, Siragy, Helmy M, Fournie-Zaluski, Marie-Claude, Roques, Bernard P, Carey, Robert M
Published in Hypertension (Dallas, Tex. 1979) (01.03.2007)
Published in Hypertension (Dallas, Tex. 1979) (01.03.2007)
Get full text
Journal Article
Conference Proceeding
Brain Renin-Angiotensin System Blockade by Systemically Active Aminopeptidase A Inhibitors: A Potential Treatment of Salt-Dependent Hypertension
Fournie-Zaluski, Marie-Claude, Fassot, Celine, Valentin, Bruno, Djordjijevic, Dragan, Goazigo, Annabelle Reaux-Le, Corvol, Pierre, Roques, Bernard P., Llorens-Cortes, Catherine, Baulieu, Etienne-Emile
Published in Proceedings of the National Academy of Sciences - PNAS (18.05.2004)
Published in Proceedings of the National Academy of Sciences - PNAS (18.05.2004)
Get full text
Journal Article
Detection and Quantification of Botulinum Neurotoxin Type A by a Novel Rapid In Vitro Fluorimetric Assay
Poras, Hervé, Ouimet, Tanja, Orng, Sou-Vinh, Fournié-Zaluski, Marie-Claude, Popoff, Michel R, Roques, Bernard P
Published in Applied and Environmental Microbiology (01.07.2009)
Published in Applied and Environmental Microbiology (01.07.2009)
Get full text
Journal Article
Long‐lasting oral analgesic effects of N‐protected aminophosphinic dual ENKephalinase inhibitors (DENKIs) in peripherally controlled pain
Bonnard, Elisabeth, Poras, Hervé, Nadal, Xavier, Maldonado, Rafael, Fournié‐Zaluski, Marie‐Claude, Roques, Bernard P.
Published in Pharmacology research & perspectives (01.03.2015)
Published in Pharmacology research & perspectives (01.03.2015)
Get full text
Journal Article
Conversion of Renal Angiotensin II to Angiotensin III Is Critical for AT2 Receptor-Mediated Natriuresis In Rats
Padia, Shetal H, Kemp, Brandon A, Howell, Nancy L, Fournie-Zaluski, Marie-Claude, Roques, Bernard P, Carey, Robert M
Published in Hypertension (Dallas, Tex. 1979) (01.02.2008)
Published in Hypertension (Dallas, Tex. 1979) (01.02.2008)
Get full text
Journal Article
Conference Proceeding
Toward an Optimal Joint Recognition of the S1‘ Subsites of Endothelin Converting Enzyme-1 (ECE-1), Angiotensin Converting Enzyme (ACE), and Neutral Endopeptidase (NEP)
Inguimbert, Nicolas, Coric, Pascale, Poras, Hervé, Meudal, Hervé, Teffot, Franck, Fournié-Zaluski, Marie-Claude, Roques, Bernard P
Published in Journal of medicinal chemistry (28.03.2002)
Published in Journal of medicinal chemistry (28.03.2002)
Get full text
Journal Article
Metabolism of angiotensin II is required for its in vivo effect on dopamine release in the striatum of the rat
Stragier, Bart, Sarre, Sophie, Vanderheyden, Patrick, Vauquelin, Georges, Fournié‐Zaluski, Marie‐Claude, Ebinger, Guy, Michotte, Yvette
Published in Journal of neurochemistry (01.09.2004)
Published in Journal of neurochemistry (01.09.2004)
Get full text
Journal Article
Aminophosphinic Inhibitors as Transition State Analogues of Enkephalin-Degrading Enzymes: A Class of Central Analgesics
Chen, Huixiong, Noble, Florence, Coric, Pascale, Fournie-Zaluski, Marie-Claude, Roques, Bernard P.
Published in Proceedings of the National Academy of Sciences - PNAS (29.09.1998)
Published in Proceedings of the National Academy of Sciences - PNAS (29.09.1998)
Get full text
Journal Article
삼차 신경통의 예방 및 치료를 위한 NEP 및 APN 의 저해제로서 디술파닐기를 함유하는 아미노산 유도체
WURM MICHEL, PORAS HERVE, ROQUES BERNARD, FOURNIE ZALUSKI MARIE CLAUDE, OUIMET TANJA
Year of Publication 07.10.2020
Get full text
Year of Publication 07.10.2020
Patent
Structure of aminopeptidase N from Escherichia coli complexed with the transition-state analogue aminophosphinic inhibitor PL250
Fournié-Zaluski, Marie-Claude, Poras, Hervé, Roques, Bernard P., Nakajima, Yoshitaka, Ito, Kiyoshi, Yoshimoto, Tadashi
Published in Acta crystallographica. Section D, Biological crystallography. (01.08.2009)
Published in Acta crystallographica. Section D, Biological crystallography. (01.08.2009)
Get full text
Journal Article
Modulation of disulfide dual ENKephalinase inhibitors (DENKIs) activity by a transient N-protection for pain alleviation by oral route
Poras, Hervé, Bonnard, Elisabeth, Fournié-Zaluski, Marie-Claude, Roques, Bernard P.
Published in European journal of medicinal chemistry (18.09.2015)
Published in European journal of medicinal chemistry (18.09.2015)
Get full text
Journal Article
Nouveaux analgésiques par complète inhibition de la dégradation enzymatique des opioïdes endogènes
Roques, Bernard P., Fournié-Zaluski, Marie-Claude, Wurm, Michel
Published in M.S. Médecine sciences (01.05.2012)
Published in M.S. Médecine sciences (01.05.2012)
Get full text
Journal Article