Biological profiling of novel tricyclic inhibitors of bacterial DNA gyrase and topoisomerase IV
Savage, Victoria J, Charrier, Cédric, Salisbury, Anne-Marie, Moyo, Emmanuel, Forward, Henry, Chaffer-Malam, Nathan, Metzger, Richard, Huxley, Anthony, Kirk, Ralph, Uosis-Martin, Mario, Noonan, Gary, Mohmed, Sarfraz, Best, Stuart A, Ratcliffe, Andrew J, Stokes, Neil R
Published in Journal of antimicrobial chemotherapy (01.07.2016)
Published in Journal of antimicrobial chemotherapy (01.07.2016)
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Journal Article
In vitro biological evaluation of novel broad-spectrum isothiazolone inhibitors of bacterial type II topoisomerases
Charrier, Cédric, Salisbury, Anne-Marie, Savage, Victoria J, Moyo, Emmanuel, Forward, Henry, Ooi, Nicola, Cheung, Jonathan, Metzger, Richard, McGarry, David, Walker, Rolf, Cooper, Ian R, Ratcliffe, Andrew J, Stokes, Neil R
Published in Journal of antimicrobial chemotherapy (01.10.2016)
Published in Journal of antimicrobial chemotherapy (01.10.2016)
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Journal Article
Discovery and structure–activity relationships of a novel isothiazolone class of bacterial type II topoisomerase inhibitors
Cooper, Ian R., McCarroll, Andrew J., McGarry, David, Kirkham, James, Pichowicz, Mark, Walker, Rolf, Warrilow, Catherine, Salisbury, Anne-Marie, Savage, Victoria J., Moyo, Emmanuel, Forward, Henry, Cheung, Jonathan, Metzger, Richard, Gault, Zoe, Nelson, Gary, Hughes, Diarmaid, Cao, Sha, Maclean, John, Charrier, Cédric, Craighead, Mark, Best, Stuart, Stokes, Neil R., Ratcliffe, Andrew J.
Published in Bioorganic & medicinal chemistry letters (01.09.2016)
Published in Bioorganic & medicinal chemistry letters (01.09.2016)
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Journal Article