Discovery and optimization of 3-thiophenylcoumarins as novel agents against Parkinson’s disease: Synthesis, in vitro and in vivo studies
Rodríguez-Enríquez, Fernanda, Viña, Dolores, Uriarte, Eugenio, Fontenla, José Angel, Matos, Maria J.
Published in Bioorganic chemistry (01.08.2020)
Published in Bioorganic chemistry (01.08.2020)
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Gamma-Decanolactone Increases Stress Resistance and Improves Toxicity Parameters on the Caenorhabditis elegans Alternative Model
Campos, Glaucia Maria, Santos, Péterson Alves, Uczay, Mariana, Pflüger, Pricila, Mendes, Thaís Lemos, Fontenla, Jose Angel, Pereira, Patrícia
Published in Journal of applied toxicology (04.10.2024)
Published in Journal of applied toxicology (04.10.2024)
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Journal Article
Novel coumarin-pyridazine hybrids as selective MAO-B inhibitors for the Parkinson’s disease therapy
Rodríguez-Enríquez, Fernanda, Costas-Lago, María Carmen, Besada, Pedro, Alonso-Pena, Miguel, Torres-Terán, Iria, Viña, Dolores, Fontenla, José Ángel, Sturlese, Mattia, Moro, Stefano, Quezada, Elias, Terán, Carmen
Published in Bioorganic chemistry (01.11.2020)
Published in Bioorganic chemistry (01.11.2020)
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Synthesis, pharmacological study and docking calculations of new benzo[f]coumarin derivatives as dual inhibitors of enzymatic systems involved in neurodegenerative diseases
Matos, Maria João, Janeiro, Patricia, González Franco, Rosa María, Vilar, Santiago, Tatonetti, Nicholas P, Santana, Lourdes, Uriarte, Eugenio, Borges, Fernanda, Fontenla, José Angel, Viña, Dolores
Published in Future medicinal chemistry (01.03.2014)
Published in Future medicinal chemistry (01.03.2014)
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Journal Article
Gamma-decanolactone attenuates acute and chronic seizures in mice: a possible role of adenosine A1 receptors
Pflüger, Pricila, Regner, Gabriela Gregory, Luft, Jordana Griebler, Gonçalves, Débora Aguirre, Krebs, Chris, Fontenla, José Angel, Pereira, Patrícia
Published in Behavioural pharmacology (01.09.2020)
Published in Behavioural pharmacology (01.09.2020)
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Journal Article
In vivo effects of new inhibitors of catechol‐O‐methyl transferase
Rivas, Emilia, De Ceballos, Maria L, Nieto, Ofelia, Fontenla, José Angel
Published in British journal of pharmacology (01.04.1999)
Published in British journal of pharmacology (01.04.1999)
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Journal Article
8-Amide and 8-carbamate substitution patterns as modulators of 7-hydroxy-4-methylcoumarin?s antidepressant profile: Synthesis, biological evaluation and docking studies
Matos, Maria J., Novo, Paula, Mayan, Lucia, Torres, Iria, Uriarte, Eugenio, Yanez, Matilde, Fontenla, Jose Angel, Ortuso, Francesco, Alcaro, Stefano, Procopio, Francesca, Rodriguez-Franco, Maria Isabel, Val, Cristina, Loza, Maria I., Brea, Jose, Borges, Fernanda, Vina, Dolores
Published in European journal of medicinal chemistry (15.02.2023)
Published in European journal of medicinal chemistry (15.02.2023)
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Journal Article
8-Amide and 8-carbamate substitution patterns as modulators of 7-hydroxy-4-methylcoumarin's antidepressant profile: Synthesis, biological evaluation and docking studies
Matos, Maria J., Novo, Paula, Mayán, Lucía, Torres, Iria, Uriarte, Eugenio, Yáñez, Matilde, Fontenla, José Ángel, Ortuso, Francesco, Alcaro, Stefano, Procopio, Francesca, Rodríguez-Franco, María Isabel, Val, Cristina, Loza, María I., Brea, José, Borges, Fernanda, Viña, Dolores
Published in European journal of medicinal chemistry (15.02.2023)
Published in European journal of medicinal chemistry (15.02.2023)
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Journal Article
Toxicological assessment of the Achyrocline satureioides aqueous extract in the Caenorhabditis elegans alternative model
Santos, Péterson Alves, Uczay, Mariana, Pflüger, Pricila, Lobo, Larissa Aline Carneiro, Rott, Marilise Brittes, Fontenla, Jose Angel, Rodrigues Siqueira, Ionara, Pereira, Patrícia
Published in Journal of Toxicology and Environmental Health, Part A (16.09.2024)
Published in Journal of Toxicology and Environmental Health, Part A (16.09.2024)
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Pyridazine derivatives, VI. Synthesis and hypotensive activity of 3-hydrazinethieno(2,3-h)cinnoline and its derivatives
García-Dominguez, N, Raviña, E, Santana, L, Terán, C, García-Mera, G, Orallo, F, Crespo, M, Fontenla, J A
Published in Archiv der Pharmazie (Weinheim) (1988)
Published in Archiv der Pharmazie (Weinheim) (1988)
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Synthesis of glycosyl derivatives as dopamine prodrugs: interaction with glucose carrier GLUT-1Electronic supplementary information (ESI) available: experimental details for the preparation of all derivatives and biological assays. See http://www.rsc.org/suppdata/ob/b2/b212066f
Fernández, Caridad, Nieto, Ofelia, Fontenla, José Angel, Rivas, Emilia, de Ceballos, María L., Fernández-Mayoralas, Alfonso
Published in Organic & biomolecular chemistry (27.02.2003)
Published in Organic & biomolecular chemistry (27.02.2003)
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Butyrophenone analogues in the carbazole series as potential atypical antipsychotics: synthesis and determination of affinities at D 2, 5-HT 2A, 5-HT 2B and 5-HT 2C receptors
Masaguer, Christian F., Raviña, Enrique, Fontenla, José Angel, Brea, José, Tristán, Helena, Loza, María Isabel
Published in European journal of medicinal chemistry (2000)
Published in European journal of medicinal chemistry (2000)
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Journal Article
Pyridazine derivatives. XI: Antihypertensive activity of 3-hydrazinocycloheptyl[1,2-c]pyridazine and its hydrazone derivatives
Gil-Longo, J, de los Reyes Laguna, M, Verde, I, Castro, M E, Orallo, F, Fontenla, J A, Calleja, J M, Ravina, E, Teran, C
Published in Journal of pharmaceutical sciences (01.03.1993)
Published in Journal of pharmaceutical sciences (01.03.1993)
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Journal Article
Synthesis and use of perimidinones in disorders of mood and anxiety (Machine-translation by Google Translate, not legally binding)
RODRIGUEZ FIDALGO, BRAIS, CIMADEVILA FONDEVILA, MARTA, SOBARZO SANCHEZ, EDUARDO, URIARTE VILLARES, EUGENIO, FONTENLA GIL, JOSÉ ANGEL
Year of Publication 29.12.2014
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Year of Publication 29.12.2014
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