ERK Inhibitor LY3214996 Targets ERK Pathway-Driven Cancers: A Therapeutic Approach Toward Precision Medicine
Bhagwat, Shripad V, McMillen, William T, Cai, Shufen, Zhao, Baohui, Whitesell, Matthew, Shen, Weihua, Kindler, Lisa, Flack, Robert S, Wu, Wenjuan, Anderson, Bryan, Zhai, Yan, Yuan, Xiu-Juan, Pogue, Meghann, Van Horn, Robert D, Rao, Xi, McCann, Denis, Dropsey, Andrew J, Manro, Jason, Walgren, Jennie, Yuen, Eunice, Rodriguez, Michael J, Plowman, Gregory D, Tiu, Ramon V, Joseph, Sajan, Peng, Sheng-Bin
Published in Molecular cancer therapeutics (01.02.2020)
Published in Molecular cancer therapeutics (01.02.2020)
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Journal Article
Abstract 583: The CDK4/6 inhibitor abemaciclib induces synergistic immune activation and antitumor efficacy in combination with PD-L1 blockade
Dempsey, Jack, Huber, Lysiane, Forest, Amelie, Stephens, Jennifer R., Doman, Thompson N., Manro, Jason, Capen, Andrew, Flack, Robert S., Donoho, Gregory P., Buchanan, Sean, Dios, Alfonso De, Driscoll, Kyla, Kalos, Michael, Novosiadly, Ruslan, Beckmann, Richard P., Schaer, David A.
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
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Journal Article
Abstract 3231: Identifying high quality, potent and selective pyrimidinylthienopyrrolone inhibitors of ERK1/2 kinase: LY3214996
Zhao, Gaiying, McMillen, William T., Cai, Shufen, Zhao, Baohui, Whitesell, Matthew, Wu, Wenjuan, Huss, Karen, Anderson, Bryan, Yuan, Xiu-Juan, Jaken, Susan, Kindler, Lisa, Flack, Robert S., McCann, Denis, Mathes, Brian, Dropsey, Andrew J., Walgren, Jennie, Yuen, Eunice, Manro, Jason, Gong, Xueqian, Cortez, Guillermo, McLean, Johnathan, Rodriguez, Michael J., Tiu, Ramon V., Bhagwat, Shripad V., Joseph, Sajan
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
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Journal Article
Abstract 4973: Discovery of LY3214996, a selective and novel ERK1/2 inhibitor with potent antitumor activities in cancer models with MAPK pathway alterations
Bhagwat, Shripad V., McMillen, William T., Cai, Shufen, Zhao, Baohui, Whitesell, Matthew, Kindler, Lisa, Flack, Robert S., Wu, Wenjuan, Huss, Karen, Anderson, Bryan, Yuan, Xiu-Juan, Jaken, Susan, McCann, Denis, Mathes, Brian, Dropsey, Andrew J., Manro, Jason, Walgren, Jennie, Yuen, Eunice, Gong, Xueqian, Rodriguez, Michael J., Huang, Jianping, Tiu, Ramon V., Joseph, Sajan, Peng, Sheng-Bin
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
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Journal Article
Method of fuel economy
FLACK ROBERT EDWARD, RATNARAJAH RAJ JEBANANDHAN, BROOK DAVID JONATHAN, LLOYD JUSTIN, DAVIS MARCUS TIMOTHY
Year of Publication 28.03.2012
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Year of Publication 28.03.2012
Patent
Method of fuel economy during cold start of a vehicle
FLACK ROBERT EDWARD, RATNARAJAH RAJ JEBANANDHAN, BROOK DAVID JONATHAN, LLOYD JUSTIN, DAVIS MARCUS TIMOTHY
Year of Publication 06.05.2009
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Year of Publication 06.05.2009
Patent