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Published in Journal of medicinal chemistry (01.02.1993)
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Bradykinin Receptor Antagonists Containing N-Substituted Amino Acids: In Vitro and in Vivo B2 and B1 Receptor Antagonist Activity
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Published in Journal of medicinal chemistry (29.03.1996)
Published in Journal of medicinal chemistry (29.03.1996)
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In vitro and in vivo Activities of Reduced-Size Antagonists of Luteinizing Hormone-Releasing Hormone
Haviv, Fortuna, Fitzpatrick, Timothy D, Nichols, Charles J, Bush, Eugene N, Diaz, Gilbert, Bammert, Gary, Nguyen, A. T, Johnson, Edwin S, Knittle, Judith, Greer, Jonathan
Published in Journal of medicinal chemistry (01.03.1994)
Published in Journal of medicinal chemistry (01.03.1994)
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1E4E-2--NN--8-4--1--3H-[B]-4- SOLID FORMS COMPRISING 1E4E-2-AMINO-NN-DIPROPYL-8-4-PYRROLIDINE-1-CARBONYLPHENYL-3H-BENZO[B]AZEPINE-4-CARBOXAMIDE COMPOSITIONS THEREOF AND USES THEREOF
FRANK ANTHONY, FERRETTI ANTONIO C, FITZPATRICK TIMOTHY D, LI YING, BEAUCHAMPS MARIE G, MAN HON WAH, LU XIAOLING
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Year of Publication 25.10.2017
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OCTAPEPTIDE LHRH ANTAGONISTS
PALABRICA, CHRISTOPHER A, GREER, JONATHAN, HAVIV, FORTUNA, FITZPATRICK, TIMOTHY D
Year of Publication 16.11.1998
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Year of Publication 16.11.1998
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Stabilization of the N-terminal residues of luteinizing hormone-releasing hormone agonists and the effect on pharmacokinetics
Haviv, Fortuna, Fitzpatrick, Timothy D, Nichols, Charles J, Swenson, Rolf E, Bush, Eugene N, Diaz, Gilbert, Nguyen, A, Nellans, Hugh N, Hoffman, Daniel J
Published in Journal of medicinal chemistry (01.10.1992)
Published in Journal of medicinal chemistry (01.10.1992)
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The effect of NMeTyr5 substitution in luteinizing hormone-releasing hormone antagonists
Haviv, Fortuna, Fitzpatrick, Timothy D, Nichols, Charles J, Swenson, Rolf E, Mort, Nicholas A, Bush, Eugene N, Diaz, Gilbert, Nguyen, A. T, Holst, Mark R
Published in Journal of medicinal chemistry (01.04.1993)
Published in Journal of medicinal chemistry (01.04.1993)
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Solid forms comprising (1E, 4E)-2-amino-N,N-dipropyl-8-(4-(pyrrolidine-1-carbonyl)phenyl)-3H-benzo[B]azepine-4-carboxami compositions thereof, and uses thereof
Lu, Xiaoling, Beauchamps, Marie G, Ferretti, Antonio C, Li, Ying, Frank, Anthony, Fitzpatrick, Timothy D, Man, Hon-Wah
Year of Publication 31.03.2020
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Year of Publication 31.03.2020
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Solid forms comprising (1E, 4E)-2-amino-N,N-dipropyl-8-(4-(pyrrolidine-1-carbonyl)phenyl)-3H-benzo(b)azepine-4-carboxamide, compositions thereof, and uses thereof
Lu, Xiaoling, Beauchamps, Marie G, Ferretti, Antonio C, Li, Ying, Frank, Anthony, Fitzpatrick, Timothy D, Man, Hon-Wah
Year of Publication 21.11.2019
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Year of Publication 21.11.2019
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SOLID FORMS COMPRISING (1E, 4E)-2-AMINO-N,N-DIPROPYL-8-(4-(PYRROLIDINE-1-CARBONYL)PHENYL)-3H-BENZO[B]AZEPINE-4-CARBOXAMIDE, COMPOSITIONS THEREOF, AND USES THEREOF
BEAUCHAMPS, Marie G, FITZPATRICK, Timothy D, LI, Ying, MAN, Hon-Wah, LU, Xiaoling, FERRETTI, Antonio C, FRANK, Anthony
Year of Publication 02.01.2020
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Year of Publication 02.01.2020
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SOLID FORMS COMPRISING (1E, 4E)-2-AMINO-N,N-DIPROPYL-8-(4-(PYRROLIDINE-1-CARBONYL)PHENYL)-3H-BENZO[B]AZEPINE-4-CARBOXAMIDE, COMPOSITIONS THEREOF, AND USES THEREOF
BEAUCHAMPS, Marie G, FITZPATRICK, Timothy D, LI, Ying, MAN, Hon-Wah, LU, Xiaoling, FERRETTI, Antonio C, FRANK, Anthony
Year of Publication 04.04.2019
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Year of Publication 04.04.2019
Patent
Bradykinin receptor antagonists containing N-substituted amino acids: In vitro and in vivo B-2 and B-1 receptor antagonist activity
Goodfellow, VS, Marathe, MV, Kuhlman, KG, Fitzpatrick, TD, Cuadrado, D, Hanson, W, Zuzack, JS, Ross, SE, Wieczorek, M, Burkard, M, Whalley, ET
Published in Journal of medicinal chemistry (29.03.1996)
Published in Journal of medicinal chemistry (29.03.1996)
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SOLID FORMS COMPRISING (1E, 4E)-2-AMINO-N,N-DIPROPYL-8-(4-(PYRROLIDINE-1-CARBONYL)PHENYL)-3H-BENZO[B]AZEPINE-4-CARBOXAMIDE, COMPOSITIONS THEREOF, AND USES THEREOF
FITZPATRICK, Timothy, D, LI, Ying, MAN, Hon-Wah, LU, Xiaoling, FERRETTI, Antonio, C, FRANK, Anthony, BEAUCHAMPS, Marie, G
Year of Publication 19.09.2018
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Year of Publication 19.09.2018
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Solid forms comprising (1E, 4E)-2-amino-N,N-dipropyl-8-(4-(pyrrolidine-1-carbonyl)phenyl)-3H-benzo(b)azepine-4-carboxamide, compositions thereof, and uses thereof
Lu, Xiaoling, Beauchamps, Marie G, Ferretti, Antonio C, Li, Ying, Frank, Anthony, Fitzpatrick, Timothy D, Man, Hon-Wah
Year of Publication 06.07.2017
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Year of Publication 06.07.2017
Patent
SOLID FORMS COMPRISING (1E, 4E)-2-AMINO-N,N-DIPROPYL-8-(4-(PYRROLIDINE-1-CARBONYL)PHENYL)-3H-BENZO[B]AZEPINE-4-CARBOXAMIDE, COMPOSITIONS THEREOF, AND USES THEREOF
FITZPATRICK, Timothy, D, LI, Ying, MAN, Hon-Wah, LU, Xiaoling, FERRETTI, Antonio, C, FRANK, Anthony, BEAUCHAMPS, Marie, G
Year of Publication 25.10.2017
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Year of Publication 25.10.2017
Patent
SOLID FORMS COMPRISING (1E, 4E)-2-AMINO-N,N-DIPROPYL-8-(4-(PYRROLIDINE-1-CARBONYL)PHENYL)-3H-BENZO[B]AZEPINE-4-CARBOXAMIDE, COMPOSITIONS THEREOF, AND USES THEREOF
FITZPATRICK, Timothy, D, LI, Ying, MAN, Hon-Wah, LU, Xiaoling, FERRETTI, Antonio, C, FRANK, Anthony, BEAUCHAMPS, Marie, G
Year of Publication 28.07.2017
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Year of Publication 28.07.2017
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SOLID FORMS COMPRISING (1E, 4E)-2-AMINO-N,N-DIPROPYL-8-(4-(PYRROLIDINE-1-CARBONYL)PHENYL)-3H-BENZO[B]AZEPINE-4-CARBOXAMIDE, COMPOSITIONS THEREOF, AND USES THEREOF
FITZPATRICK, Timothy, D, LI, Ying, MAN, Hon-Wah, LU, Xiaoling, FERRETTI, Antonio, C, FRANK, Anthony, BEAUCHAMPS, Marie, G
Year of Publication 15.09.2016
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Year of Publication 15.09.2016
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SOLID FORMS COMPRISING (1E, 4E)-2-AMINO-N,N-DIPROPYL-8-(4-(PYRROLIDINE-1-CARBONYL)PHENYL)-3H-BENZO[B]AZEPINE-4-CARBOXAMIDE, COMPOSITIONS THEREOF, AND USES THEREOF
FERRETTI, ANTONIO C, LI, YING, FRANK, ANTHONY, BEAUCHAMPS, MARIE G, MAN, HON-WAH, FITZPATRICK, TIMOTHY D, LU, XIAOLING
Year of Publication 23.06.2016
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Year of Publication 23.06.2016
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SOLID FORMS COMPRISING (1E, 4E)-2-AMINO-N,N-DIPROPYL-8-(4-(PYRROLIDINE-1-CARBONYL)PHENYL)-3H-BENZO[B]AZEPINE-4-CARBOXAMIDE, COMPOSITIONS THEREOF, AND USES THEREOF
FITZPATRICK, TIMOTHY, D, FERRETTI, ANTONIO, C, LI, YING, FRANK, ANTHONY, BEAUCHAMPS, MARIE, G, MAN, HON-WAH, LU, XIAOLING
Year of Publication 23.06.2016
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Year of Publication 23.06.2016
Patent
Differential orientation of a GnRH agonist and antagonist in the pituitary GnRH receptor
Janovick, J A, Haviv, F, Fitzpatrick, T D, Conn, P M
Published in Endocrinology (Philadelphia) (01.08.1993)
Published in Endocrinology (Philadelphia) (01.08.1993)
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