Three-dimensional structure of aspartyl protease from human immunodeficiency virus HIV-1
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Estrogen receptor ligands. Part 16: 2-Aryl indoles as highly subtype selective ligands for ERα
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Published in Bioorganic & medicinal chemistry letters (15.04.2007)
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Published in Journal of medicinal chemistry (16.08.1996)
Published in Journal of medicinal chemistry (16.08.1996)
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Estrogen receptor ligands. Part 9: Dihydrobenzoxathiin SERAMs with alkyl substituted pyrrolidine side chains and linkers
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Published in Journal of medicinal chemistry (01.01.1995)
Published in Journal of medicinal chemistry (01.01.1995)
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Structure-Based Design of HIV-1 Protease Inhibitors: Replacement of Two Amides and a 10.pi.-Aromatic System by a Fused Bis-tetrahydrofuran
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Published in Journal of medicinal chemistry (01.08.1994)
Published in Journal of medicinal chemistry (01.08.1994)
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Expression, purification, crystallization and preliminary X-ray analysis of Aeromonas hydrophilia metallo-β-lactamase
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Published in Acta crystallographica. Section F, Structural biology and crystallization communications (01.02.2005)
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A Priori Prediction of Activity for HIV-1 Protease Inhibitors Employing Energy Minimization in the Active Site
Holloway, M. Katharine, Wai, Jenny M, Halgren, Thomas A, Fitzgerald, Paula M. D, Vacca, Joseph P, Dorsey, Bruce D, Levin, Rhonda B, Thompson, Wayne J, Chen, L. Jenny, deSolms, S. Jane, Gaffin, Neil, Ghosh, Arun K, Giuliani, Elizabeth A, Graham, Samuel L, Guare, James P, Hungate, Randall W, Lyle, Terry A, Sanders, William M, Tucker, Thomas J, Wiggins, Mark, Wiscount, Catherine M, Woltersdorf, Otto W, Young, Steven D, Darke, Paul L, Zugay, Joan A
Published in Journal of medicinal chemistry (24.05.1996)
Published in Journal of medicinal chemistry (24.05.1996)
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Synthesis and antiviral activity of a series of HIV-1 protease inhibitors with functionality tethered to the P1 or P1' phenyl design
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Published in Journal of medicinal chemistry (01.05.1992)
Published in Journal of medicinal chemistry (01.05.1992)
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Unanticipated Inhibition of the Metallo-β-lactamase from Bacteroides fragilis by 4-Morpholineethanesulfonic Acid (MES): A Crystallographic Study at 1.85-Å Resolution
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Published in Biochemistry (Easton) (12.05.1998)
Published in Biochemistry (Easton) (12.05.1998)
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Estrogen receptor ligands. Part 16: 2-Aryl indoles as highly subtype selective ligands for ERalpha
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Published in Bioorganic & medicinal chemistry letters (15.04.2007)
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Published in Bioorganic & medicinal chemistry letters (15.04.2007)
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Nonpeptidal P-2 ligands for HIV protease inhibitors: Structure-based design, synthesis, and biological evaluation
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Published in Journal of medicinal chemistry (16.08.1996)
Published in Journal of medicinal chemistry (16.08.1996)
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Estrogen receptor ligands. II. Discovery of benzoxathiins as potent, selective estrogen receptor a modulators
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Published in Journal of medicinal chemistry (2004)
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Published in Journal of medicinal chemistry (2004)
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Succinic Acids as Potent Inhibitors of Plasmid-borne IMP-1 Metallo-β-lactamase
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Published in The Journal of biological chemistry (24.08.2001)
Published in The Journal of biological chemistry (24.08.2001)
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